2uw0 A 2.0 BS02 GVK A 1 G50 T51 G52 G55 R56 V57 A70 E121 Y122 A123 E127 E170 N171 M173 T183 D184 F327 G37 T38 G39 G42 R43 V44 A57 E108 Y109 A110 E114 E157 N158 M160 T170 D171 F314 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0001669,0001707,0004672,0004674,0004679,0004691,0005515,0005524,0005634,0005737,0005739,0005829,0005886,0005952,0006468,0010737,0016310,0018105,0019904,0031594,0034237,0034605,0036126,0048471,0106310,1904262 -logKd/Ki=7.70, IC50=20nM P00517 17451235 1351 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLTKLEFSFKDNSNLYMVMEYAPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLMIDQQGYIKVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF