17gs A 1.9 BS01 GTX A 1 Y7 F8 R13 W38 K44 Q51 L52 Q64 S65 G205 Y8 F9 R14 W39 K45 Q52 L53 Q65 S66 G206 Y7 R13 Y8 R14 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 P09211 210 MPPYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPAFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 17gs B 1.9 BS01 GTX B 1 Y7 F8 R13 W38 K44 Q51 L52 Q64 S65 G205 Y6 F7 R12 W37 K43 Q50 L51 Q63 S64 G204 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 P09211 210 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPAFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 1bh5 A 2.2 BS02 GTX A 1 R122 M157 F162 R116 M151 F156 E33 E99 H126 Q172 E27 E93 H120 Q166 4.4.1.5 0004462,0005515,0005654,0005737,0005829,0005886,0005975,0006357,0006749,0008270,0009438,0016829,0030316,0043066,0046872,0070062 Q04760 9705294 200 SGGLTDEAALSCCSDADPSTKDFLLQETMLRVKDPKKSLDFYTRVLGMTLIQKCDFPIMKFSLYFLAYEDKNDIPKEKDEKIAWALSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIQILNPNKMATLM 1bh5 A 2.2 BS04 GTX B 1 R37 F67 L69 T101 N103 R31 F61 L63 T95 N97 E33 E99 H126 Q172 E27 E93 H120 Q166 4.4.1.5 0004462,0005515,0005654,0005737,0005829,0005886,0005975,0006357,0006749,0008270,0009438,0016829,0030316,0043066,0046872,0070062 Q04760 9705294 200 SGGLTDEAALSCCSDADPSTKDFLLQETMLRVKDPKKSLDFYTRVLGMTLIQKCDFPIMKFSLYFLAYEDKNDIPKEKDEKIAWALSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIQILNPNKMATLM 1bh5 B 2.2 BS02 GTX A 1 R37 F67 T101 N103 R36 F66 T100 N102 E33 E99 H126 Q172 E32 E98 H125 Q171 4.4.1.5 0004462,0005515,0005654,0005737,0005829,0005886,0005975,0006357,0006749,0008270,0009438,0016829,0030316,0043066,0046872,0070062 Q04760 9705294 200 EPQPPSGGLTDEAALSCCSDADPSTKDFLLQETMLRVKDPKKSLDFYTRVLGMTLIQKCDFPIMKFSLYFLAYEDKNDIPKEKDEKIAWALSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIQILNPNKMATLM 1bh5 B 2.2 BS04 GTX B 1 R122 M157 F162 M183 R121 M156 F161 M182 E33 E99 H126 Q172 E32 E98 H125 Q171 4.4.1.5 0004462,0005515,0005654,0005737,0005829,0005886,0005975,0006357,0006749,0008270,0009438,0016829,0030316,0043066,0046872,0070062 Q04760 9705294 200 EPQPPSGGLTDEAALSCCSDADPSTKDFLLQETMLRVKDPKKSLDFYTRVLGMTLIQKCDFPIMKFSLYFLAYEDKNDIPKEKDEKIAWALSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIQILNPNKMATLM 1bh5 C 2.2 BS02 GTX C 1 R122 F162 M179 R116 F156 M173 E33 E99 H126 Q172 E27 E93 H120 Q166 4.4.1.5 0004462,0005515,0005654,0005737,0005829,0005886,0005975,0006357,0006749,0008270,0009438,0016829,0030316,0043066,0046872,0070062 Q04760 9705294 200 SGGLTDEAALSCCSDADPSTKDFLLQETMLRVKDPKKSLDFYTRVLGMTLIQKCDFPIMKFSLYFLAYEDKNDIPKEKDEKIAWALSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIQILNPNKMATLM 1bh5 C 2.2 BS04 GTX D 1 R37 F67 L69 T101 N103 R31 F61 L63 T95 N97 E33 E99 H126 Q172 E27 E93 H120 Q166 4.4.1.5 0004462,0005515,0005654,0005737,0005829,0005886,0005975,0006357,0006749,0008270,0009438,0016829,0030316,0043066,0046872,0070062 Q04760 9705294 200 SGGLTDEAALSCCSDADPSTKDFLLQETMLRVKDPKKSLDFYTRVLGMTLIQKCDFPIMKFSLYFLAYEDKNDIPKEKDEKIAWALSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIQILNPNKMATLM 1bh5 D 2.2 BS02 GTX C 1 R37 F67 N103 R36 F66 N102 E33 E99 H126 Q172 E32 E98 H125 Q171 4.4.1.5 0004462,0005515,0005654,0005737,0005829,0005886,0005975,0006357,0006749,0008270,0009438,0016829,0030316,0043066,0046872,0070062 Q04760 9705294 200 EPQPPSGGLTDEAALSCCSDADPSTKDFLLQETMLRVKDPKKSLDFYTRVLGMTLIQKCDFPIMKFSLYFLAYEDKNDIPKEKDEKIAWALSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIQILNPNKMATLM 1bh5 D 2.2 BS04 GTX D 1 R122 F162 M183 R121 F161 M182 E33 E99 H126 Q172 E32 E98 H125 Q171 4.4.1.5 0004462,0005515,0005654,0005737,0005829,0005886,0005975,0006357,0006749,0008270,0009438,0016829,0030316,0043066,0046872,0070062 Q04760 9705294 200 EPQPPSGGLTDEAALSCCSDADPSTKDFLLQETMLRVKDPKKSLDFYTRVLGMTLIQKCDFPIMKFSLYFLAYEDKNDIPKEKDEKIAWALSRKATLELTHNWGTEDDETQSYHNGNSDPRGFGHIGIAVPDVYSACKRFEELGVKFVKKPDDGKMKGLAFIQDPDGYWIQILNPNKMATLM 1gnw A 2.2 BS01 GTX A 1 L35 K41 Q53 V54 E66 S67 L34 K40 Q52 V53 E65 S66 2.5.1.18 0000325,0002239,0004364,0004601,0005737,0005783,0005829,0005886,0006952,0009407,0009409,0009506,0009507,0009570,0009636,0009734,0010043,0016740,0019904,0043231,0043295,0046686,0048046,0098869,1901149,2001147,2001227 P46422 8551521 212 GIKVFGHPASIATRRVLIALHEKNLDFELVHVELKDGEHKKEPFLSRNPFGQVPAFEDGDLKLFESRAITQYIAHRYENQGTNLLQTDSKNISQYAIMAIGMQVEDHQFDPVASKLAFEQIFKSIYGLTTDEAVVAEEEAKLAKVLDVYEARLKEFKYLAGETFTLTDLHHIPAIQYLLGTPTKKLFTERPRVNEWVAEITKRPASEKVQ 1gnw A 2.2 BS02 GTX A 2 S11 I12 A13 Q53 I122 S10 I11 A12 Q52 I121 2.5.1.18 0000325,0002239,0004364,0004601,0005737,0005783,0005829,0005886,0006952,0009407,0009409,0009506,0009507,0009570,0009636,0009734,0010043,0016740,0019904,0043231,0043295,0046686,0048046,0098869,1901149,2001147,2001227 P46422 8551521 213 GIKVFGHPASIATRRVLIALHEKNLDFELVHVELKDGEHKKEPFLSRNPFGQVPAFEDGDLKLFESRAITQYIAHRYENQGTNLLQTDSKNISQYAIMAIGMQVEDHQFDPVASKLAFEQIFKSIYGLTTDEAVVAEEEAKLAKVLDVYEARLKEFKYLAGETFTLTDLHHIPAIQYLLGTPTKKLFTERPRVNEWVAEITKRPASEKVQ 1gnw B 2.2 BS01 GTX B 1 L35 K41 Q53 V54 E66 S67 L34 K40 Q52 V53 E65 S66 2.5.1.18 0000325,0002239,0004364,0004601,0005737,0005783,0005829,0005886,0006952,0009407,0009409,0009506,0009507,0009570,0009636,0009734,0010043,0016740,0019904,0043231,0043295,0046686,0048046,0098869,1901149,2001147,2001227 P46422 8551521 212 GIKVFGHPASIATRRVLIALHEKNLDFELVHVELKDGEHKKEPFLSRNPFGQVPAFEDGDLKLFESRAITQYIAHRYENQGTNLLQTDSKNISQYAIMAIGMQVEDHQFDPVASKLAFEQIFKSIYGLTTDEAVVAEEEAKLAKVLDVYEARLKEFKYLAGETFTLTDLHHIPAIQYLLGTPTKKLFTERPRVNEWVAEITKRPASEKVQ 1gnw B 2.2 BS02 GTX B 2 S11 I12 A13 S10 I11 A12 2.5.1.18 0000325,0002239,0004364,0004601,0005737,0005783,0005829,0005886,0006952,0009407,0009409,0009506,0009507,0009570,0009636,0009734,0010043,0016740,0019904,0043231,0043295,0046686,0048046,0098869,1901149,2001147,2001227 P46422 8551521 213 GIKVFGHPASIATRRVLIALHEKNLDFELVHVELKDGEHKKEPFLSRNPFGQVPAFEDGDLKLFESRAITQYIAHRYENQGTNLLQTDSKNISQYAIMAIGMQVEDHQFDPVASKLAFEQIFKSIYGLTTDEAVVAEEEAKLAKVLDVYEARLKEFKYLAGETFTLTDLHHIPAIQYLLGTPTKKLFTERPRVNEWVAEITKRPASEKVQ 1gsu A 1.94 BS01 GTX A 1 Y6 W7 W45 K49 N58 L59 Q71 S72 Y115 W209 Y6 W7 W45 K49 N58 L59 Q71 S72 Y115 W209 Y6 L12 R17 Y6 L12 R17 2.5.1.18 0004364,0005737,0006629,0016740,0042802 P20136 9571047 220 VVTLGYWDIRGLAHAIRLLLEYTETPYQERRYKAGPAPDFDPSDWTNEKEKLGLDFPNLPYLIDGDVKLTQSNAILRYIARKHNMCGETEVEKQRVDVLENHLMDLRMAFARLCYSPDFEKLKPAYLEQLPGKLRQLSRFLGSRSWFVGDKLTFVDFLAYDVLDQQRMFVPDCPELQGNLSQFLQRFEALEKISAYMRSGRFMKAPIFWYTALWNNK 1gsu B 1.94 BS01 GTX B 1 Y6 G11 L12 W45 N58 L59 Q71 S72 R107 Y6 G11 L12 W45 N58 L59 Q71 S72 R107 Y6 L12 R17 Y6 L12 R17 2.5.1.18 0004364,0005737,0006629,0016740,0042802 P20136 9571047 220 VVTLGYWDIRGLAHAIRLLLEYTETPYQERRYKAGPAPDFDPSDWTNEKEKLGLDFPNLPYLIDGDVKLTQSNAILRYIARKHNMCGETEVEKQRVDVLENHLMDLRMAFARLCYSPDFEKLKPAYLEQLPGKLRQLSRFLGSRSWFVGDKLTFVDFLAYDVLDQQRMFVPDCPELQGNLSQFLQRFEALEKISAYMRSGRFMKAPIFWYTALWNNK 1gwc A 2.25 BS01 GTX A 1 S15 F17 K42 K55 I56 E68 S69 S12 F14 K39 K52 I53 E65 S66 2.5.1.18 0004364,0005737,0006749,0016740 O04941 12033934 1225 GDDLKLLGAWPSPFVTRVKLALALKGLSYEDVEEDLYKKSELLLKSNPVHKKIPVLIHNGAPVCESMIILQYIDEVFASTGPSLLPADPYERAIARFWVAYVDDKLVAPWRQWLRGKTEEEKSEGKKQAFAAVGVLEGALRECSKGGGFFGGDGVGLVDVALGGVLSWMKVTEALSGDKIFDAAKTPLLAAWVERFIELDAAKAALPDVGRLLEFAKAREA 1gwc B 2.25 BS01 GTX B 1 S15 F17 K42 K55 I56 E68 S69 S12 F14 K39 K52 I53 E65 S66 2.5.1.18 0004364,0005737,0006749,0016740 O04941 12033934 1225 GDDLKLLGAWPSPFVTRVKLALALKGLSYEDVEEDLYKKSELLLKSNPVHKKIPVLIHNGAPVCESMIILQYIDEVFASTGPSLLPADPYERAIARFWVAYVDDKLVAPWRQWLRGKTEEEKSEGKKQAFAAVGVLEGALRECSKGGGFFGGDGVGLVDVALGGVLSWMKVTEALSGDKIFDAAKTPLLAAWVERFIELDAAKAALPDVGRLLEFAKAREA 1gwc C 2.25 BS01 GTX C 1 S15 F17 K42 K55 I56 E68 S69 S12 F14 K39 K52 I53 E65 S66 2.5.1.18 0004364,0005737,0006749,0016740 O04941 12033934 1226 GDDLKLLGAWPSPFVTRVKLALALKGLSYEDVEEDLYKKSELLLKSNPVHKKIPVLIHNGAPVCESMIILQYIDEVFASTGPSLLPADPYERAIARFWVAYVDDKLVAPWRQWLRGKTEEEKSEGKKQAFAAVGVLEGALRECSKGGGFFGGDGVGLVDVALGGVLSWMKVTEALSGDKIFDAAKTPLLAAWVERFIELDAAKAALPDVGRLLEFAKAREAA 1k0a A 2.5 BS01 GTX A 1 A122 P123 N124 F146 R164 V165 E180 S181 L231 W316 A23 P24 N25 F47 R65 V66 E81 S82 L132 W196 A122 A23 1.11.1.9,1.8.4.- 0003714,0006808 P23202 11695904 355 SRITKFFQEQPLEGYTLFSHRSAPNGFKVAIVLSELGFHYNTIFLDFNLGEHRAPEFVSVNPNARVPALIDHGMDNLSIWESGAILLHLVNKYYKETGNPLLWSDDLADQSQINAWLFFQTSGHAPMIGQALHFRYFHSQKIASAVERYTDEVRRVYGVVEMALAERREALVMEFDYPVWLVGDKLTIADLAFVPWNNVVDRIGINIKIEFPEVYKWTKHMMRRPAVIKALRGE 1k3l A 1.5 BS01 GTX A 1 Y9 R15 R45 Q54 V55 Q67 T68 V111 L213 F220 Y8 R14 R44 Q53 V54 Q66 T67 V110 L212 F219 Y9 R15 R20 Y8 R14 R19 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 12211029 5100 AEKPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 1k3l A 1.5 BS02 GTX B 1 D101 R131 D100 R130 Y9 R15 R20 Y8 R14 R19 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 12211029 5200 AEKPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 1k3l B 1.5 BS01 GTX A 1 D101 R131 D98 R128 Y9 R15 R20 Y6 R12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 12211029 5100 KPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 1k3l B 1.5 BS02 GTX B 1 R15 R45 Q54 V55 Q67 T68 F220 R12 R42 Q51 V52 Q64 T65 F217 Y9 R15 R20 Y6 R12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 12211029 5200 KPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 1k3y A 1.3 BS01 GTX A 1 Y9 R15 R45 Q54 V55 Q67 T68 V111 F220 Y8 R14 R44 Q53 V54 Q66 T67 V110 F219 Y9 R15 R20 Y8 R14 R19 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 12211029 5100 AEKPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 1k3y A 1.3 BS04 GTX B 1 D101 R131 D100 R130 Y9 R15 R20 Y8 R14 R19 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 12211029 5200 AEKPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 1k3y B 1.3 BS01 GTX A 1 D101 R131 D100 R130 Y9 R15 R20 Y8 R14 R19 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 12211029 5100 AEKPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 1k3y B 1.3 BS02 GTX B 1 R15 R45 Q54 V55 Q67 T68 F220 R14 R44 Q53 V54 Q66 T67 F219 Y9 R15 R20 Y8 R14 R19 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 12211029 5200 AEKPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 1m9a A 2.1 BS01 GTX A 1 Y7 W8 L13 W41 K45 N54 L55 Q67 S68 R103 S107 Q204 Y7 W8 L13 W41 K45 N54 L55 Q67 S68 R103 S107 Q204 Y7 L13 Y7 L13 2.5.1.18 0004364,0006749,0016740 P08515 12596270 220 MSPILGYWKIKGLVQPTRLLLEYLEEKYEEHLYERDEGDKWRNKKFELGLEFPNLPYYIDGDVKLTQSMAIIRYIADKHNMLGGCPKERAEISMLEGAVLDIRYGVSRIAYSKDFETLKVDFLSKLPEMLKMFEDRLCHKTYLNGDHVTHPDFMLYDALDVVLYMDPMCLDAFPKLVCFKKRIEAIPQIDKYLKSSKYIAWPLQGWQATFGGGDHP 1pgt A 1.8 BS01 GTX A 1 Y7 F8 R13 W38 K44 Q51 L52 Q64 S65 Y8 F9 R14 W39 K45 Q52 L53 Q65 S66 Y7 R13 Y8 R14 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 P09211 9245401 210 MPPYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYVSLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 1pgt B 1.8 BS01 GTX B 1 F8 R13 W38 K44 Q51 L52 Q64 S65 Y108 F8 R13 W38 K44 Q51 L52 Q64 S65 Y108 Y7 R13 Y7 R13 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 P09211 9245401 210 PPYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYVSLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 1pn9 A 2.0 BS01 GTX A 1 S9 P11 L33 H50 C51 I52 E64 S65 F207 S9 P11 L33 H50 C51 I52 E64 S65 F207 S9 S9 2.5.1.18,4.5.1.1 0003824,0004364,0006749,0016740,0016829,0018833 Q93113 14646079 301 MDFYYLPGSAPCRAVQMTAAAVGVELNLKLTDLMKGEHMKPEFLKLNPQHCIPTLVDNGFALWESRAIQIYLAEKYGKDDKLYPKDPQKRAVVNQRLYFDMGTLYQRFADYHYPQIFAKQPANPENEKKMKDAVGFLNTFLEGQEYAAGNDLTIADLSLAATIATYEVAGFDFAPYPNVAAWFARCKANAPGYALNQAGADEFKAKFLS 1pn9 B 2.0 BS01 GTX B 1 S9 L33 H50 C51 I52 E64 S65 Y113 S9 L33 H50 C51 I52 E64 S65 Y113 S9 S9 2.5.1.18,4.5.1.1 0003824,0004364,0006749,0016740,0016829,0018833 Q93113 14646079 302 MDFYYLPGSAPCRAVQMTAAAVGVELNLKLTDLMKGEHMKPEFLKLNPQHCIPTLVDNGFALWESRAIQIYLAEKYGKDDKLYPKDPQKRAVVNQRLYFDMGTLYQRFADYHYPQIFAKQPANPENEKKMKDAVGFLNTFLEGQEYAAGNDLTIADLSLAATIATYEVAGFDFAPYPNVAAWFARCKANAPGYALNQAGADEFKAKFLS 1q4j A 2.2 BS01 GTX A 1 Y9 F10 K15 F45 Q58 V59 Q71 S72 N111 Y7 F8 K13 F43 Q56 V57 Q69 S70 N109 Y9 K15 R20 Y7 K13 R18 2.5.1.18 0004364,0016740 Q8ILQ7 12972411 212 DNIVLYYFDARGKAELIRLIFAYLGIEYTDKRFGVNGDAFVEFKNFKKEKDTPFEQVPILQIGDLILAQSQAIVRYLSKKYNICGESELNEFYADMIFCGVQDIHYKFNNTNLFKQNETTFLNEDLPKWSGYFEKLLKKNHTNNNNDKYYFVGNNLTYADLAVFNLYDDIETKYPSSLKNFPLLKAHNEFISNLPNIKNYITNRKESVY 1q4j A 2.2 BS02 GTX B 1 F116 K117 E120 T121 F114 K115 E118 T119 Y9 K15 R20 Y7 K13 R18 2.5.1.18 0004364,0016740 Q8ILQ7 12972411 212 DNIVLYYFDARGKAELIRLIFAYLGIEYTDKRFGVNGDAFVEFKNFKKEKDTPFEQVPILQIGDLILAQSQAIVRYLSKKYNICGESELNEFYADMIFCGVQDIHYKFNNTNLFKQNETTFLNEDLPKWSGYFEKLLKKNHTNNNNDKYYFVGNNLTYADLAVFNLYDDIETKYPSSLKNFPLLKAHNEFISNLPNIKNYITNRKESVY 1q4j B 2.2 BS01 GTX A 1 F116 K117 T121 F114 K115 T119 Y9 K15 R20 Y7 K13 R18 2.5.1.18 0004364,0016740 Q8ILQ7 12972411 212 DNIVLYYFDARGKAELIRLIFAYLGIEYTDKRFGVNGDAFVEFKNFKKEKDTPFEQVPILQIGDLILAQSQAIVRYLSKKYNICGESELNEFYADMIFCGVQDIHYKFNNTNLFKQNETTFLNEDLPKWSGYFEKLLKKNHTNNNNDKYYFVGNNLTYADLAVFNLYDDIETKYPSSLKNFPLLKAHNEFISNLPNIKNYITNRKESVY 1q4j B 2.2 BS02 GTX B 1 Y9 F45 Q58 V59 Q71 S72 N111 Y7 F43 Q56 V57 Q69 S70 N109 Y9 K15 R20 Y7 K13 R18 2.5.1.18 0004364,0016740 Q8ILQ7 12972411 212 DNIVLYYFDARGKAELIRLIFAYLGIEYTDKRFGVNGDAFVEFKNFKKEKDTPFEQVPILQIGDLILAQSQAIVRYLSKKYNICGESELNEFYADMIFCGVQDIHYKFNNTNLFKQNETTFLNEDLPKWSGYFEKLLKKNHTNNNNDKYYFVGNNLTYADLAVFNLYDDIETKYPSSLKNFPLLKAHNEFISNLPNIKNYITNRKESVY 1tu8 A 1.8 BS01 GTX A 1 Y7 F8 L13 F38 K42 Q49 L50 Q62 S63 Y106 Y7 F8 L13 F38 K42 Q49 L50 Q62 S63 Y106 Y7 L13 R18 Y7 L13 R18 2.5.1.18 0004364,0005829,0006749,0016740 P46427 15640152 2001 MSYKLTYFSIRGLAEPIRLFLVDQDIKFIDDRIAKDDFSSIKSQFQFGQLPCLYDGDQQIVQSGAILRHLARKYNLNGENEMETTYIDMFCEGVRDLHVKYTRMIYMAYETEKDPYIKSILPGELAKFEKLLATRGNGRNLILGDKISYADYALFEELDVHQILDPHCLDKFPLLKVFHQRMKDRPKLKEYCEKRDAAKVPVNGNGKQ 1tu8 B 1.8 BS01 GTX B 1 Y7 F8 L13 K35 F38 Q49 L50 Q62 S63 Y106 Y7 F8 L13 K35 F38 Q49 L50 Q62 S63 Y106 Y7 L13 R18 Y7 L13 R18 2.5.1.18 0004364,0005829,0006749,0016740 P46427 15640152 2002 MSYKLTYFSIRGLAEPIRLFLVDQDIKFIDDRIAKDDFSSIKSQFQFGQLPCLYDGDQQIVQSGAILRHLARKYNLNGENEMETTYIDMFCEGVRDLHVKYTRMIYMAYETEKDPYIKSILPGELAKFEKLLATRGNGRNLILGDKISYADYALFEELDVHQILDPHCLDKFPLLKVFHQRMKDRPKLKEYCEKRDAAKVPVNGNGKQ 1tu8 C 1.8 BS01 GTX C 1 Y7 F8 L13 F38 K42 Q49 L50 Q62 S63 Y106 Y7 F8 L13 F38 K42 Q49 L50 Q62 S63 Y106 Y7 L13 R18 Y7 L13 R18 2.5.1.18 0004364,0005829,0006749,0016740 P46427 15640152 2004 MSYKLTYFSIRGLAEPIRLFLVDQDIKFIDDRIAKDDFSSIKSQFQFGQLPCLYDGDQQIVQSGAILRHLARKYNLNGENEMETTYIDMFCEGVRDLHVKYTRMIYMAYETEKDPYIKSILPGELAKFEKLLATRGNGRNLILGDKISYADYALFEELDVHQILDPHCLDKFPLLKVFHQRMKDRPKLKEYCEKRDAAKVPVNGNGKQ 1tu8 D 1.8 BS01 GTX D 1 Y7 F8 L13 F38 Q49 L50 Q62 S63 Y106 Y7 F8 L13 F38 Q49 L50 Q62 S63 Y106 Y7 L13 R18 Y7 L13 R18 2.5.1.18 0004364,0005829,0006749,0016740 P46427 15640152 2003 MSYKLTYFSIRGLAEPIRLFLVDQDIKFIDDRIAKDDFSSIKSQFQFGQLPCLYDGDQQIVQSGAILRHLARKYNLNGENEMETTYIDMFCEGVRDLHVKYTRMIYMAYETEKDPYIKSILPGELAKFEKLLATRGNGRNLILGDKISYADYALFEELDVHQILDPHCLDKFPLLKVFHQRMKDRPKLKEYCEKRDAAKVPVNGNGKQ 1vf2 A 2.15 BS01 GTX A 1 Y9 K15 Q54 V55 Q67 T68 L220 M222 Y223 Y6 K12 Q51 V52 Q64 T65 L217 M219 Y220 2.5.1.18 0004364,0005737,0006749,0006805,0016740 P26697 2457 KPVLYYFNGRGKMESIRWLLAAAGVEFEEVFLETREQYEKLLQSGILMFQQVPMVEIDGMKLVQTRAILNYIAGKYNLYGKDLKERALIDMYVGGTDDLMGFLLSFPFLSAEDKVKQCAFVVEKATSRYFPAYEKVLKDHGQDFLVGNRLSWADIHLLEAILMVEEKKSDALSGFPLLQAFKKRISSIPTIKKFLAPGSKRKPISDDKYVETVRRVLRMYYDVKP 1vf2 A 2.15 BS02 GTX B 1 D101 R131 D98 R128 2.5.1.18 0004364,0005737,0006749,0006805,0016740 P26697 3468 KPVLYYFNGRGKMESIRWLLAAAGVEFEEVFLETREQYEKLLQSGILMFQQVPMVEIDGMKLVQTRAILNYIAGKYNLYGKDLKERALIDMYVGGTDDLMGFLLSFPFLSAEDKVKQCAFVVEKATSRYFPAYEKVLKDHGQDFLVGNRLSWADIHLLEAILMVEEKKSDALSGFPLLQAFKKRISSIPTIKKFLAPGSKRKPISDDKYVETVRRVLRMYYDVKP 1vf2 B 2.15 BS01 GTX A 1 D1101 R1131 D98 R128 Y1009 K1015 R1020 Y6 K12 R17 2.5.1.18 0004364,0005737,0006749,0006805,0016740 P26697 2457 KPVLYYFNGRGKMESIRWLLAAAGVEFEEVFLETREQYEKLLQSGILMFQQVPMVEIDGMKLVQTRAILNYIAGKYNLYGKDLKERALIDMYVGGTDDLMGFLLSFPFLSAEDKVKQCAFVVEKATSRYFPAYEKVLKDHGQDFLVGNRLSWADIHLLEAILMVEEKKSDALSGFPLLQAFKKRISSIPTIKKFLAPGSKRKPISDDKYVETVRRVLRMYYDVKP 1vf2 B 2.15 BS02 GTX B 1 K1015 Q1054 V1055 Q1067 T1068 F1111 M1222 Y1223 K12 Q51 V52 Q64 T65 F108 M219 Y220 Y1009 K1015 R1020 Y6 K12 R17 2.5.1.18 0004364,0005737,0006749,0006805,0016740 P26697 3468 KPVLYYFNGRGKMESIRWLLAAAGVEFEEVFLETREQYEKLLQSGILMFQQVPMVEIDGMKLVQTRAILNYIAGKYNLYGKDLKERALIDMYVGGTDDLMGFLLSFPFLSAEDKVKQCAFVVEKATSRYFPAYEKVLKDHGQDFLVGNRLSWADIHLLEAILMVEEKKSDALSGFPLLQAFKKRISSIPTIKKFLAPGSKRKPISDDKYVETVRRVLRMYYDVKP 1ydk A 1.95 BS01 GTX A 1 R15 R45 Q54 V55 Q67 T68 L107 R13 R43 Q52 V53 Q65 T66 L105 Y9 R15 R20 Y7 R13 R18 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 Kd=1.3uM -logKd/Ki=5.89, Kd=1.3uM P08263 15893769 5100 EKPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMD 1ydk A 1.95 BS02 GTX B 1 D101 R131 D99 R129 Y9 R15 R20 Y7 R13 R18 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 Kd=1.3uM -logKd/Ki=5.89, Kd=1.3uM P08263 15893769 5200 EKPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMD 1ydk B 1.95 BS01 GTX A 1 D101 R131 D98 R128 Y9 R15 R20 Y6 R12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 Kd=1.3uM -logKd/Ki=5.89, Kd=1.3uM P08263 15893769 5100 KPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKAFRF 1ydk B 1.95 BS02 GTX B 1 R15 Q54 V55 Q67 T68 L107 F220 R12 Q51 V52 Q64 T65 L104 F217 Y9 R15 R20 Y6 R12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 Kd=1.3uM -logKd/Ki=5.89, Kd=1.3uM P08263 15893769 5200 KPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKAFRF 2aaw A 2.4 BS01 GTX A 1 Y9 Q58 V59 Q71 S72 F116 Y9 Q58 V59 Q71 S72 F116 Y9 K15 R20 Y9 K15 R20 2.5.1.18 0004364,0016740 Ki=35uM Q8ILQ7 16385005 220 MGDNIVLYYFDARGKAELIRLIFAYLGIEYTDKRFGVNGDAFVEFKNFKKEKDTPFEQVPILQIGDLILAQSQAIVRYLSKKYNICGESELNEFYADMIFCGVQDIHYKFNNTNLFKQNETTFLNEDLPKWSGYFEKLLKKNHKYYFVGNNLTYADLAVFNLYDDIETKYPSSLKNFPLLKAHNEFISNLPNIKNYITNRKESVY 2aaw C 2.4 BS01 GTX C 1 Q58 V59 Q71 S72 Q58 V59 Q71 S72 2.5.1.18 0004364,0016740 Ki=35uM Q8ILQ7 16385005 221 MGDNIVLYYFDARGKAELIRLIFAYLGIEYTDKRFGVNGDAFVEFKNFKKEKDTPFEQVPILQIGDLILAQSQAIVRYLSKKYNICGESELNEFYADMIFCGVQDIHYKFNNTNLFKQNETTFLNEDLPKWSGYFEKLLKKNHTNNNNDKYYFVGNNLTYADLAVFNLYDDIETKYPSSLKNFPLLKAHNEFISNLPNIKNYITNRKESVY 2c3q A 1.85 BS01 GTX A 1 S11 H40 K53 V54 E66 S67 W115 R234 M238 S10 H39 K52 V53 E65 S66 W114 R233 M237 S11 S10 2.5.1.18 0004364,0004602,0005515,0005737,0005829,0006749,0016740,0070062,0098869 P30711 16298388 301 GLELYLDLLSQPCRAVYIFAKKNDIPFELRIVDLIKGQHLSDAFAQVNPLKKVPALKDGDFTLTESVAILLYLTRKYKVPDYWYPQDLQARARVDEYLAWQHTTLRRSCLRALWHKVMFPVFLGEPVSPQTLAATLAELDVTLQLLEDKFLQNKAFLTGPHISLADLVAITELMHPVGAGCQVFEGRPKLATWRQRVEAAVGEDLFQEAHEVILKAKDFPPADPTIKQKLMPRVLAMIR 2c3q B 1.85 BS01 GTX B 1 L35 H40 K53 V54 E66 S67 R234 M238 L34 H39 K52 V53 E65 S66 R233 M237 S11 S10 2.5.1.18 0004364,0004602,0005515,0005737,0005829,0006749,0016740,0070062,0098869 P30711 16298388 301 GLELYLDLLSQPCRAVYIFAKKNDIPFELRIVDLIKGQHLSDAFAQVNPLKKVPALKDGDFTLTESVAILLYLTRKYKVPDYWYPQDLQARARVDEYLAWQHTTLRRSCLRALWHKVMFPVFLGEPVSPQTLAATLAELDVTLQLLEDKFLQNKAFLTGPHISLADLVAITELMHPVGAGCQVFEGRPKLATWRQRVEAAVGEDLFQEAHEVILKAKDFPPADPTIKQKLMPRVLAMIR 2c3q C 1.85 BS01 GTX C 1 S11 L35 H40 K53 V54 E66 S67 R234 M238 S10 L34 H39 K52 V53 E65 S66 R233 M237 S11 S10 2.5.1.18 0004364,0004602,0005515,0005737,0005829,0006749,0016740,0070062,0098869 P30711 16298388 301 GLELYLDLLSQPCRAVYIFAKKNDIPFELRIVDLIKGQHLSDAFAQVNPLKKVPALKDGDFTLTESVAILLYLTRKYKVPDYWYPQDLQARARVDEYLAWQHTTLRRSCLRALWHKVMFPVFLGEPVSPQTLAATLAELDVTLQLLEDKFLQNKAFLTGPHISLADLVAITELMHPVGAGCQVFEGRPKLATWRQRVEAAVGEDLFQEAHEVILKAKDFPPADPTIKQKLMPRVLAMIR 2c3q D 1.85 BS01 GTX D 1 S11 L35 H40 K53 V54 E66 S67 R234 M238 S10 L34 H39 K52 V53 E65 S66 R233 M237 S11 S10 2.5.1.18 0004364,0004602,0005515,0005737,0005829,0006749,0016740,0070062,0098869 P30711 16298388 301 GLELYLDLLSQPCRAVYIFAKKNDIPFELRIVDLIKGQHLSDAFAQVNPLKKVPALKDGDFTLTESVAILLYLTRKYKVPDYWYPQDLQARARVDEYLAWQHTTLRRSCLRALWHKVMFPVFLGEPVSPQTLAATLAELDVTLQLLEDKFLQNKAFLTGPHISLADLVAITELMHPVGAGCQVFEGRPKLATWRQRVEAAVGEDLFQEAHEVILKAKDFPPADPTIKQKLMPRVLAMIR 2c80 A 2.3 BS01 GTX A 1 Y10 R16 W41 K45 R52 L53 E70 S71 Y110 L113 Y7 R13 W38 K42 R49 L50 E67 S68 Y107 L110 Y10 R16 R21 Y7 R13 R18 2.5.1.18 0004364,0006749,0016740 Kd=4.7uM -logKd/Ki=5.33, Kd=4.7uM P30113 16777141 1212 DHIKVIYFNGRGRAESIRMTLVAAGVNYEDERISFQDWPKIKPTIPGGRLPAVKITDNHGHVKWMVESLAIARYMAKKHHMMGGTEEEYYNVEKLIGQAEDLEHEYYKTLMKPEEEKQKIIKEILNGKVPVLLDIICESLKASTGKLAVGDKVTLADLVLIAVIDHVTDLDKEFLTGKYPEIHKHRENLLASSPRLAKYLSDRAATPF 2c80 B 2.3 BS01 GTX B 1 Y10 F11 R16 W41 K45 R52 L53 E70 S71 Y110 F211 Y7 F8 R13 W38 K42 R49 L50 E67 S68 Y107 F208 Y10 R16 R21 Y7 R13 R18 2.5.1.18 0004364,0006749,0016740 Kd=4.7uM -logKd/Ki=5.33, Kd=4.7uM P30113 16777141 1213 DHIKVIYFNGRGRAESIRMTLVAAGVNYEDERISFQDWPKIKPTIPGGRLPAVKITDNHGHVKWMVESLAIARYMAKKHHMMGGTEEEYYNVEKLIGQAEDLEHEYYKTLMKPEEEKQKIIKEILNGKVPVLLDIICESLKASTGKLAVGDKVTLADLVLIAVIDHVTDLDKEFLTGKYPEIHKHRENLLASSPRLAKYLSDRAATPF 2glr A 2.2 BS01 GTX A 1 F8 I35 W38 K44 Q51 L52 Q64 S65 F8 I35 W38 K44 Q51 L52 Q64 S65 Y7 R13 R18 Y7 R13 R18 2.5.1.18 0000302,0002674,0004364,0005634,0005737,0005739,0005829,0006629,0006693,0006749,0006805,0008432,0009636,0014003,0016740,0019207,0031100,0031667,0032355,0032691,0032720,0032869,0032872,0032873,0032930,0032991,0033591,0035726,0043066,0043124,0043200,0045471,0048147,0051122,0051771,0070372,0070373,0070664,0071222,0071364,0071385,0071460,0071638,1901687,2000429,2001237 P19157 8145243 210 PPYTIVYFPVRGRCEAMRMLLADQGQSWKEEVVTIDTWMQGLLKPTCLYGQLPKFEDGDLTLYQSNAILRHLGRSLGLYGKNQREAAQMDMVNDGVEDLRGKYVTLIYTNYENGKNDYVKALPGHLKPFETLLSQNQGGKAFIVGDQISFADYNLLDLLLIHQVLAPGCLDNFPLLSAYVARLSARPKIKAFLSSPEHVNRPINGNGKQ 2glr B 2.2 BS01 GTX B 1 Y7 F8 R13 W38 K44 Q51 L52 Q64 S65 Y7 F8 R13 W38 K44 Q51 L52 Q64 S65 Y7 R13 R18 Y7 R13 R18 2.5.1.18 0000302,0002674,0004364,0005634,0005737,0005739,0005829,0006629,0006693,0006749,0006805,0008432,0009636,0014003,0016740,0019207,0031100,0031667,0032355,0032691,0032720,0032869,0032872,0032873,0032930,0032991,0033591,0035726,0043066,0043124,0043200,0045471,0048147,0051122,0051771,0070372,0070373,0070664,0071222,0071364,0071385,0071460,0071638,1901687,2000429,2001237 P19157 8145243 210 PPYTIVYFPVRGRCEAMRMLLADQGQSWKEEVVTIDTWMQGLLKPTCLYGQLPKFEDGDLTLYQSNAILRHLGRSLGLYGKNQREAAQMDMVNDGVEDLRGKYVTLIYTNYENGKNDYVKALPGHLKPFETLLSQNQGGKAFIVGDQISFADYNLLDLLLIHQVLAPGCLDNFPLLSAYVARLSARPKIKAFLSSPEHVNRPINGNGKQ 2imk A 1.9 BS01 GTX A 1 S12 P14 L36 H41 H53 T54 I55 E67 S68 F108 R112 L207 S11 P13 L35 H40 H52 T53 I54 E66 S67 F107 R111 L206 S12 S11 2.5.1.18 0003824,0004364,0006749 Q7PVS6 18778777 302 SNLVLYTLHLSPPCRAVELTAKALGLELEQKTINLLTGDHLKPEFVKLNPQHTIPVLDDNGTIITESHAIMIYLVTKYGKDDSLYPKDPVKQARVNSALHFESGVLFARMRFIFERILFFGKSDIPEDRVEYVQKSYELLEDTLVDDFVAGPTMTIADFSCISTISSIMGVVPLEQSKHPRIYAWIDRLKQLPYYEEANGGGGTDLGKFVLAKKEENAKA 2imk B 1.9 BS01 GTX B 1 S12 P14 L36 H41 H53 T54 I55 E67 S68 F108 R112 S12 P14 L36 H41 H53 T54 I55 E67 S68 F108 R112 S12 S12 2.5.1.18 0003824,0004364,0006749 Q7PVS6 18778777 301 MSNLVLYTLHLSPPCRAVELTAKALGLELEQKTINLLTGDHLKPEFVKLNPQHTIPVLDDNGTIITESHAIMIYLVTKYGKDDSLYPKDPVKQARVNSALHFESGVLFARMRFIFERILFFGKSDIPEDRVEYVQKSYELLEDTLVDDFVAGPTMTIADFSCISTISSIMGVVPLEQSKHPRIYAWIDRLKQLPYYEEANGGGGTDLGKFVLAKKEENA 2j9h A 2.4 BS01 GTX A 1 F9 R14 W39 K45 Q52 L53 Q65 S66 F8 R13 W38 K44 Q51 L52 Q64 S65 Y8 R14 Y7 R13 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 Ki=410uM -logKd/Ki=3.39, Ki=410uM P09211 18177897 300 PPYTVVYFPVRGRSAALRMLLADQGQSWKEEVVTVETWQEGSLKASALYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRAKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGSLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 2j9h B 2.4 BS01 GTX B 1 F9 R14 W39 K45 G51 Q52 L53 Q65 S66 F8 R13 W38 K44 G50 Q51 L52 Q64 S65 Y8 R14 Y7 R13 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 Ki=410uM -logKd/Ki=3.39, Ki=410uM P09211 18177897 300 PPYTVVYFPVRGRSAALRMLLADQGQSWKEEVVTVETWQEGSLKASALYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRAKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGSLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 2oa7 A 2.2 BS01 GTX A 1 F8 V10 R13 I35 K44 Q51 L52 Q64 G205 F8 V10 R13 I35 K44 Q51 L52 Q64 G205 Y7 R13 R18 Y7 R13 R18 2.5.1.18 0000302,0002674,0004364,0005634,0005737,0005739,0005829,0006629,0006693,0006749,0006805,0008432,0009636,0014003,0016740,0019207,0031100,0031667,0032355,0032691,0032720,0032869,0032872,0032873,0032930,0032991,0033591,0035726,0043066,0043124,0043200,0045471,0048147,0051122,0051771,0070372,0070373,0070664,0071222,0071364,0071385,0071460,0071638,1901687,2000429,2001237 P19157 301 PPYTIVYFPVRGRAEAMRMLLADQGQSWKEEVVTIDTWMQGLLKPTCLYGQLPKFEDGDLTLYQSNAILRHLGRSLGLYGKNQREAAQMDMVNDGVEDLRGKYVTLIYTNYENGKNDYVKALPGHLKPFETLLSQNQGGKAFIVGDQISFADYNLLDLLLIHQVLAPGCLDNFPLLSAYVARLSARPKIKAFLSSPEHVNRPINGNGKQ 2oa7 B 2.2 BS01 GTX B 1 F8 V10 R13 I35 W38 K44 Q51 L52 Q64 S65 G205 F8 V10 R13 I35 W38 K44 Q51 L52 Q64 S65 G205 Y7 R13 R18 Y7 R13 R18 2.5.1.18 0000302,0002674,0004364,0005634,0005737,0005739,0005829,0006629,0006693,0006749,0006805,0008432,0009636,0014003,0016740,0019207,0031100,0031667,0032355,0032691,0032720,0032869,0032872,0032873,0032930,0032991,0033591,0035726,0043066,0043124,0043200,0045471,0048147,0051122,0051771,0070372,0070373,0070664,0071222,0071364,0071385,0071460,0071638,1901687,2000429,2001237 P19157 302 PPYTIVYFPVRGRAEAMRMLLADQGQSWKEEVVTIDTWMQGLLKPTCLYGQLPKFEDGDLTLYQSNAILRHLGRSLGLYGKNQREAAQMDMVNDGVEDLRGKYVTLIYTNYENGKNDYVKALPGHLKPFETLLSQNQGGKAFIVGDQISFADYNLLDLLLIHQVLAPGCLDNFPLLSAYVARLSARPKIKAFLSSPEHVNRPINGNGKQ 2r3x A 1.8 BS01 GTX A 1 Y9 L15 R45 Q54 V55 Q67 T68 F220 Y8 L14 R44 Q53 V54 Q66 T67 F219 Y9 L15 R20 Y8 L14 R19 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 19959275 5100 AEKPKLHYFNARGLMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 2r3x A 1.8 BS02 GTX B 1 D101 R131 D100 R130 Y9 L15 R20 Y8 L14 R19 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 19959275 5200 AEKPKLHYFNARGLMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 2r3x B 1.8 BS01 GTX A 1 D101 R131 D98 R128 Y9 L15 R20 Y6 L12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 19959275 5100 KPKLHYFNARGLMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 2r3x B 1.8 BS02 GTX B 1 Y9 L15 R45 Q54 V55 Q67 T68 L107 F220 Y6 L12 R42 Q51 V52 Q64 T65 L104 F217 Y9 L15 R20 Y6 L12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 19959275 5200 KPKLHYFNARGLMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 2r6k A 2.51 BS01 GTX A 1 Y9 R45 Q54 V55 Q67 T68 F220 Y8 R44 Q53 V54 Q66 T67 F219 Y9 R15 R20 Y8 R14 R19 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 20606271 5100 AEKPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAVLNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 2r6k A 2.51 BS02 GTX B 1 D101 R131 D100 R130 Y9 R15 R20 Y8 R14 R19 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 20606271 5200 AEKPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAVLNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 2r6k B 2.51 BS01 GTX A 1 D101 R131 D98 R128 Y9 R15 R20 Y6 R12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 20606271 5100 KPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAVLNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 2r6k B 2.51 BS02 GTX B 1 Y9 R15 R45 Q54 V55 Q67 T68 L107 F220 Y6 R12 R42 Q51 V52 Q64 T65 L104 F217 Y9 R15 R20 Y6 R12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 20606271 5200 KPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAVLNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 3f63 A 1.8 BS01 GTX A 1 S9 P11 L33 H50 C51 I52 E65 S66 Y119 F123 S9 P11 L33 H50 C51 I52 E65 S66 Y119 F123 S9 S9 2.5.1.18 0004364,0006749,0016740 Q9GN60 20196771 220 MDFYYLPGSAPCRAVQMTAAAVGVELNLKLTNLMAGEHMKPEFLKLNPQHCIPTLVDEDGFVLWESRAIQIYLVEKYGAHDADLAERLYPSDPRRRAVVHQRLFFDVAVLYQRFAEYYYPQIFGQKVPVGDPGRLRSMEQALEFLNTFLEGEQYVAGGDDPTIADLSILATIATYEVAGYDLRRYENVQRWYERTSAIVPGADKNVEGAKVFGRYFTQ 3f63 B 1.8 BS01 GTX B 1 S9 P11 L33 H50 C51 I52 E65 S66 F212 Y215 S9 P11 L33 H50 C51 I52 E65 S66 F212 Y215 S9 S9 2.5.1.18 0004364,0006749,0016740 Q9GN60 20196771 220 MDFYYLPGSAPCRAVQMTAAAVGVELNLKLTNLMAGEHMKPEFLKLNPQHCIPTLVDEDGFVLWESRAIQIYLVEKYGAHDADLAERLYPSDPRRRAVVHQRLFFDVAVLYQRFAEYYYPQIFGQKVPVGDPGRLRSMEQALEFLNTFLEGEQYVAGGDDPTIADLSILATIATYEVAGYDLRRYENVQRWYERTSAIVPGADKNVEGAKVFGRYF 3f6d A 1.7 BS01 GTX A 1 S9 P11 L33 H50 C51 I52 E65 S66 Y119 I122 Y215 S9 P11 L33 H50 C51 I52 E65 S66 Y119 I122 Y215 S9 S9 2.5.1.18 0004364,0006749,0016740 Q9GN60 20196771 220 MDFYYLPGSAPCRAVQMTAAAVGVELNLKLTNLMAGEHMKPEFLKLNPQHCIPTLVDEDGFVLWESRAIQIYLVEKYGAHDADLAERLYPSDPRRRAVVHQRLFFDVAVLYQRFAEYYYPQIAGQKVPVGDPGRLRSMEQALEFLNTFLEGEQYVAGGDDPTIADLSILATIATYEVAGYDLRRYENVQRWYERTSAIVPGADKNVEGAKVFGRYFTQ 3f6d B 1.7 BS01 GTX B 1 S9 P11 L33 H50 C51 I52 E65 S66 S9 P11 L33 H50 C51 I52 E65 S66 S9 S9 2.5.1.18 0004364,0006749,0016740 Q9GN60 20196771 220 MDFYYLPGSAPCRAVQMTAAAVGVELNLKLTNLMAGEHMKPEFLKLNPQHCIPTLVDEDGFVLWESRAIQIYLVEKYGAHDADLAERLYPSDPRRRAVVHQRLFFDVAVLYQRFAEYYYGDPGRLRSMEQALEFLNTFLEGEQYVAGGDDPTIADLSILATIATYEVAGYDLRRYENVQRWYERTSAIVPGADKNVEGAKVFG 3g7j A 2.2 BS01 GTX A 1 G8 S9 P11 L33 H38 H50 C51 I52 E65 S66 Y215 G8 S9 P11 L33 H38 H50 C51 I52 E65 S66 Y215 S9 S9 2.5.1.18 0004364,0006749,0016740 Q9GN60 20196771 220 MDFYYLPGSAPCRAVQMTAAAVGVELNLKLTNLMAGEHMKPEFLKLNPQHCIPTLVDEDGFVLWESRAIQIYLVEKYGAHDADLAERLYPSDPRRRAVVHQRLFFDVAVLYQRFAEYYEPQIFGQKVPVGDPGRLRSMEQALEFLNTFLEGEQYVAGGDDPTIADLSILATIATYEVAGYDLRRYENVQRWYERTSAIVPGADKNVEGAKVFGRYFT 3g7j B 2.2 BS01 GTX B 1 G8 S9 P11 H50 C51 I52 E65 S66 G8 S9 P11 H50 C51 I52 E65 S66 S9 S9 2.5.1.18 0004364,0006749,0016740 Q9GN60 20196771 220 MDFYYLPGSAPCRAVQMTAAAVGVELNLKLTNLMAGEHMKPEFLKLNPQHCIPTLVDEDGFVLWESRAIQIYLVEKYGAHDADLAERLYPSDPRRRAVVHQRLFFDVAVLYQRFAEYYEPQIFGQKVPVGDPGRLRSMEQALEFLNTFLEGEQYVAGGDDPTIADLSILATIATYEVAGYDLRRYENVQRWYERTSAIVPGADKNVEGAKVFGRYF 3ktl A 1.75 BS01 GTX A 1 Y9 R15 Q54 V55 Q67 T68 V111 F220 Y8 R14 Q53 V54 Q66 T67 V110 F219 Y9 R15 R20 Y8 R14 R19 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 20606271 5100 AEKPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAALNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 3ktl A 1.75 BS02 GTX B 1 D101 R131 D100 R130 Y9 R15 R20 Y8 R14 R19 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 20606271 5200 AEKPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAALNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 3ktl B 1.75 BS01 GTX A 1 D101 R131 D98 R128 Y9 R15 R20 Y6 R12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 20606271 5100 KPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAALNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 3ktl B 1.75 BS02 GTX B 1 R15 R45 Q54 V55 Q67 T68 M208 F220 R12 R42 Q51 V52 Q64 T65 M205 F217 Y9 R15 R20 Y6 R12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 20606271 5200 KPKLHYFNARGRMESTRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAALNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 3l0h A 2.13 BS01 GTX A 1 R15 Q54 V55 Q67 T68 F220 R14 Q53 V54 Q66 T67 F219 Y9 R15 R20 Y8 R14 R19 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 20833278 5100 AEKPKLHYFNARGRMESTRALLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 3l0h A 2.13 BS02 GTX B 1 D101 R131 D100 R130 Y9 R15 R20 Y8 R14 R19 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 20833278 5200 AEKPKLHYFNARGRMESTRALLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 3l0h B 2.13 BS01 GTX A 1 D101 R131 D98 R128 Y9 R15 R20 Y6 R12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 20833278 5100 KPKLHYFNARGRMESTRALLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 3l0h B 2.13 BS02 GTX B 1 R45 Q54 V55 Q67 T68 L107 F220 R42 Q51 V52 Q64 T65 L104 F217 Y9 R15 R20 Y6 R12 R17 1.11.1.-,2.5.1.18,5.3.3.- 0004364,0004601,0004602,0004769,0005504,0005515,0005737,0005829,0006629,0006693,0006749,0006805,0016740,0016853,0030855,0043651,0070062,0098869,1901687 P08263 20833278 5200 KPKLHYFNARGRMESTRALLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEIDGMKLVQTRAILNYIASKYNLYGKDIKERALIDMYIEGIADLGEMILLLPVCPPEEKDAKLALIKEKIKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPLLKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEEARKIFRF 3rpn A 1.9 BS01 GTX A 1 L15 S16 P17 Y18 N53 P56 M66 G182 L183 F198 G199 S200 D201 L14 S15 P16 Y17 N52 P55 M65 G181 L182 F197 G198 S199 D200 2.5.1.18 0004364,0004602,0005515,0005737,0005739,0005759,0005777,0005782,0005829,0006749,0016020,0016491,0016740,0030855,0043231,0070062,0098869 Q9Y2Q3 21728995 302 GPLPRTVELFYDVLSPYSWLGFEILCRYQNIWNINLQLRPSLITGIMKDSGNKPPGLLPRKGLYMANDLKLLRHHLQIPIHFPKDFLSVMLEKGSLSAMRFLTAVNLEHPEMLEKASRELWMRVWSRNEDITEPQSILAAAEKAGMSAEQAQGLLEKIATPKVKNQLKETTEAACRYGAFGLPITVAHVDGQTHMLFGSDRMELLAHLLGEKWMGPIPPA 3rpn B 1.9 BS01 GTX B 1 L15 S16 P17 Y18 N53 P56 M91 L92 G182 L183 F198 G199 S200 D201 L14 S15 P16 Y17 N52 P55 M90 L91 G181 L182 F197 G198 S199 D200 2.5.1.18 0004364,0004602,0005515,0005737,0005739,0005759,0005777,0005782,0005829,0006749,0016020,0016491,0016740,0030855,0043231,0070062,0098869 Q9Y2Q3 21728995 301 GPLPRTVELFYDVLSPYSWLGFEILCRYQNIWNINLQLRPSLITGIMKDSGNKPPGLLPRKGLYMANDLKLLRHHLQIPIHFPKDFLSVMLEKGSLSAMRFLTAVNLEHPEMLEKASRELWMRVWSRNEDITEPQSILAAAEKAGMSAEQAQGLLEKIATPKVKNQLKETTEAACRYGAFGLPITVAHVDGQTHMLFGSDRMELLAHLLGEKWMGPIPPA 3rpn C 1.9 BS01 GTX C 1 L15 S16 P17 Y18 I44 N53 P56 M91 G182 L183 F198 G199 S200 D201 L14 S15 P16 Y17 I43 N52 P55 M90 G181 L182 F197 G198 S199 D200 2.5.1.18 0004364,0004602,0005515,0005737,0005739,0005759,0005777,0005782,0005829,0006749,0016020,0016491,0016740,0030855,0043231,0070062,0098869 Q9Y2Q3 21728995 301 GPLPRTVELFYDVLSPYSWLGFEILCRYQNIWNINLQLRPSLITGIMKDSGNKPPGLLPRKGLYMANDLKLLRHHLQIPIHFPKDFLSVMLEKGSLSAMRFLTAVNLEHPEMLEKASRELWMRVWSRNEDITEPQSILAAAEKAGMSAEQAQGLLEKIATPKVKNQLKETTEAACRYGAFGLPITVAHVDGQTHMLFGSDRMELLAHLLGEKWMGPIPPA 3rpn D 1.9 BS01 GTX D 1 S16 P17 Y18 N53 M66 L70 L88 G182 L183 F198 G199 S200 D201 S15 P16 Y17 N52 M65 L69 L87 G181 L182 F197 G198 S199 D200 2.5.1.18 0004364,0004602,0005515,0005737,0005739,0005759,0005777,0005782,0005829,0006749,0016020,0016491,0016740,0030855,0043231,0070062,0098869 Q9Y2Q3 21728995 302 GPLPRTVELFYDVLSPYSWLGFEILCRYQNIWNINLQLRPSLITGIMKDSGNKPPGLLPRKGLYMANDLKLLRHHLQIPIHFPKDFLSVMLEKGSLSAMRFLTAVNLEHPEMLEKASRELWMRVWSRNEDITEPQSILAAAEKAGMSAEQAQGLLEKIATPKVKNQLKETTEAACRYGAFGLPITVAHVDGQTHMLFGSDRMELLAHLLGEKWMGPIPPA 3rpn E 1.9 BS01 GTX E 1 S16 P17 Y18 N53 M66 L88 G182 L183 F198 G199 S200 D201 S15 P16 Y17 N52 M65 L87 G181 L182 F197 G198 S199 D200 2.5.1.18 0004364,0004602,0005515,0005737,0005739,0005759,0005777,0005782,0005829,0006749,0016020,0016491,0016740,0030855,0043231,0070062,0098869 Q9Y2Q3 21728995 302 GPLPRTVELFYDVLSPYSWLGFEILCRYQNIWNINLQLRPSLITGIMKDSGNKPPGLLPRKGLYMANDLKLLRHHLQIPIHFPKDFLSVMLEKGSLSAMRFLTAVNLEHPEMLEKASRELWMRVWSRNEDITEPQSILAAAEKAGMSAEQAQGLLEKIATPKVKNQLKETTEAACRYGAFGLPITVAHVDGQTHMLFGSDRMELLAHLLGEKWMGPIPPA 3rpn F 1.9 BS01 GTX C 1 K62 R202 K61 R201 2.5.1.18 0004364,0004602,0005515,0005737,0005739,0005759,0005777,0005782,0005829,0006749,0016020,0016491,0016740,0030855,0043231,0070062,0098869 Q9Y2Q3 21728995 301 GPLPRTVELFYDVLSPYSWLGFEILCRYQNIWNINLQLRPSLITGIMKDSGNKPPGLLPRKGLYMANDLKLLRHHLQIPIHFPKDFLSVMLEKGSLSAMRFLTAVNLEHPEMLEKASRELWMRVWSRNEDITEPQSILAAAEKAGMSAEQAQGLLEKIATPKVKNQLKETTEAACRYGAFGLPITVAHVDGQTHMLFGSDRMELLAHLLGEKWMGPIPPA 3rpn F 1.9 BS02 GTX F 1 S16 P17 Y18 N53 P56 M66 L88 W126 G182 L183 F198 G199 S200 D201 S15 P16 Y17 N52 P55 M65 L87 W125 G181 L182 F197 G198 S199 D200 2.5.1.18 0004364,0004602,0005515,0005737,0005739,0005759,0005777,0005782,0005829,0006749,0016020,0016491,0016740,0030855,0043231,0070062,0098869 Q9Y2Q3 21728995 302 GPLPRTVELFYDVLSPYSWLGFEILCRYQNIWNINLQLRPSLITGIMKDSGNKPPGLLPRKGLYMANDLKLLRHHLQIPIHFPKDFLSVMLEKGSLSAMRFLTAVNLEHPEMLEKASRELWMRVWSRNEDITEPQSILAAAEKAGMSAEQAQGLLEKIATPKVKNQLKETTEAACRYGAFGLPITVAHVDGQTHMLFGSDRMELLAHLLGEKWMGPIPPA 4gss A 2.5 BS01 GTX A 1 F8 R13 W38 K44 Q51 L52 Q64 S65 G205 F7 R12 W37 K43 Q50 L51 Q63 S64 G204 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 P09211 9166793 210 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIFTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 4gss B 2.5 BS01 GTX B 1 F8 R13 W38 K44 Q51 L52 Q64 S65 G205 F7 R12 W37 K43 Q50 L51 Q63 S64 G204 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 P09211 9166793 210 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIFTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 4jc7 A 2.7 BS01 GTX A 1 N55 E58 Y59 Y93 R104 L108 A116 N60 E63 Y64 Y98 R109 L113 A121 2.5.1.-,4.4.1.20 0004364,0004464,0004602,0005515,0005634,0005635,0005640,0005783,0005789,0006629,0006691,0008047,0008289,0016020,0016740,0016829,0019370,0031965,0042759,0042802,0043231,0098869 Q16873 24366866 211 HHHHHHKDEVALLAAVTLLGVLLQAYFSLQVISARRAFRVSPPLTTGPPEFERVYRAQVNCSEYFPLFLATLWVAGIFFHEGAAALCGLVYLFARLRYFQGYARSAQLRLAPLYASARALALLVALAALGLLAHFLPAALRAALLGRLRTLLPW 4jcz A 2.75 BS01 GTX A 1 N55 E58 Y59 Y93 R104 L108 L115 W116 N56 E59 Y60 Y94 R105 L109 L116 W117 2.5.1.-,4.4.1.20 0004364,0004464,0004602,0005515,0005634,0005635,0005640,0005783,0005789,0006629,0006691,0008047,0008289,0016020,0016740,0016829,0019370,0031965,0042759,0042802,0043231,0098869 Q16873 24366866 209 HHKDEVALLAAVTLLGVLLQAYFSLQVISARRAFRVSPPLTTGPPEFERVYRAQVNCSEYFPLFLATLWVAGIFFHEGAAALCGLVYLFARLRYFQGYARSAQLRLAPLYASARALWLLVALAALGLLAHFLPAALRAALLGRLRTL 4jrz A 2.4 BS01 GTX A 1 N55 E58 Y59 Y93 R104 L108 F116 N61 E64 Y65 Y99 R110 L114 F122 2.5.1.-,4.4.1.20 0004364,0004464,0004602,0005515,0005634,0005635,0005640,0005783,0005789,0006629,0006691,0008047,0008289,0016020,0016740,0016829,0019370,0031965,0042759,0042802,0043231,0098869 Q16873 24366866 211 MHHHHHHKDEVALLAAVTLLGVLLQAYFSLQVISARRAFRVSPPLTTGPPEFERVYRAQVNCSEYFPLFLATLWVAGIFFHEGAAALCGLVYLFARLRYFQGYARSAQLRLAPLYASARALFLLVALAALGLLAHFLPAALRAALLGRLRTLLPW 4ntf A 2.65 BS01 GTX A 1 N55 E58 Y59 R104 L108 W116 N55 E58 Y59 R104 L108 W116 2.5.1.-,4.4.1.20 0004464,0005634,0005635,0005640,0005783,0005789,0006629,0006691,0008047,0008289,0016020,0016740,0016829,0019370,0031965 Q60860 201 HKDEVALLATVTLVGVLLQAYFSLQVISARRAFHVSPPLTSGPPEFERVFRAQVNCSEYFPLFLATLWVAGIFFHEGAAALCGLFYLFARLRYFQGYARSAQLRLTPLYASARALWLLVAMAALGLLVHFLPGTLRTALFRWLQM 5kej A 2.35 BS01 GTX A 1 S14 Y16 K54 I55 E67 S68 S13 Y15 K53 I54 E66 S67 2.5.1.18 0004364,0005737,0005829,0006749,0009407,0009636,0016740 Kd=7.8uM -logKd/Ki=5.11, Kd=7.8uM A0A1P8NWC2 28104507 301 AKSDVKLLGAWPSPYVMRARITLNVKSVDYELLEETLGSKSDLLLKSNPVHKKIPVLIHNDKPICESLIIVHYIDEFWSSGPSILPSDPYDRAIARFWAAYLDEKWYPSLKGIASAQGEEAKKAAVDQVGESLALIEDTYVKLSKGKPFFGGEKIGYLDIAFGCFLGWLRVTEKTSGVKFLNEAKTPHLAKWAVRFCADPAVKDVMPETEKLAEFAKLLAKF 5kej B 2.35 BS01 GTX B 1 S14 Y16 K54 I55 E67 S68 Y108 S13 Y15 K53 I54 E66 S67 Y107 2.5.1.18 0004364,0005737,0005829,0006749,0009407,0009636,0016740 Kd=7.8uM -logKd/Ki=5.11, Kd=7.8uM A0A1P8NWC2 28104507 301 AKSDVKLLGAWPSPYVMRARITLNVKSVDYELLEETLGSKSDLLLKSNPVHKKIPVLIHNDKPICESLIIVHYIDEFWSSGPSILPSDPYDRAIARFWAAYLDEKWYPSLKGIASAQGEEAKKAAVDQVGESLALIEDTYVKLSKGKPFFGGEKIGYLDIAFGCFLGWLRVTEKTSGVKFLNEAKTPHLAKWAVRFCADPAVKDVMPETEKLAEFAKLLAKF 6f4k A 1.55 BS01 GTX A 1 S15 Y17 K55 I56 E80 S81 S12 Y14 K52 I53 E77 S78 2.5.1.18 0004364,0005737,0046872 A0A384E145 29855494 300 TKQITLYTATFSPYAHRVRIALEEAGAEYTTYDVDILRNMPDWFPLVNPLKKIPAMTFGGPEVPPDQPSPESAKIAESLAMLEFIADLFPDAKLLPTDPVLRARARTFMALYENYVNGQFRDVWFLGTPADPLLQALEMLQGALPPDGGFAAGEWSIADAAVIPFLARMFPYLEAGLGLYSKEDGVKMRKAMASERFARIRQYVRDCRARPSFANTWAGDAEQVEAAKTVPMLRVGEHHHH 6f4k A 1.55 BS02 GTX A 2 Y17 N120 R124 F128 F168 M172 Y14 N117 R121 F125 F165 M169 2.5.1.18 0004364,0005737,0046872 A0A384E145 29855494 301 TKQITLYTATFSPYAHRVRIALEEAGAEYTTYDVDILRNMPDWFPLVNPLKKIPAMTFGGPEVPPDQPSPESAKIAESLAMLEFIADLFPDAKLLPTDPVLRARARTFMALYENYVNGQFRDVWFLGTPADPLLQALEMLQGALPPDGGFAAGEWSIADAAVIPFLARMFPYLEAGLGLYSKEDGVKMRKAMASERFARIRQYVRDCRARPSFANTWAGDAEQVEAAKTVPMLRVGEHHHH 6f4k B 1.55 BS01 GTX B 1 F14 S15 P16 Y17 K55 I56 E80 S81 Y175 F11 S12 P13 Y14 K52 I53 E77 S78 Y172 2.5.1.18 0004364,0005737,0046872 A0A384E145 29855494 301 TKQITLYTATFSPYAHRVRIALEEAGAEYTTYDVDILRNMPDWFPLVNPLKKIPAMTFGGPEVPPDQPSPESAKIAESLAMLEFIADLFPDAKLLPTDPVLRARARTFMALYENYVNGQFRDVWFLGTPADPLLQALEMLQGALPPDGGFAAGEWSIADAAVIPFLARMFPYLEAGLGLYSKEDGVKMRKAMASERFARIRQYVRDCRARPSFANTWAGDAEQVEAAKTVPMLRVGEHHHH 9gss A 1.97 BS01 GTX A 1 F8 R13 W38 Q51 L52 Q64 S65 G205 F7 R12 W37 Q50 L51 Q63 S64 G204 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 P09211 9398518 211 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ 9gss B 1.97 BS01 GTX B 1 Y7 F8 R13 W38 Q51 L52 Q64 S65 G205 Y6 F7 R12 W37 Q50 L51 Q63 S64 G204 Y7 R13 Y6 R12 2.5.1.18 0000302,0002674,0004364,0004602,0005504,0005515,0005576,0005615,0005634,0005737,0005739,0005829,0006469,0006629,0006693,0006749,0006805,0007417,0008432,0009890,0010804,0016740,0019207,0031982,0032691,0032720,0032872,0032873,0032930,0034774,0035726,0035730,0035731,0035732,0043066,0043124,0043407,0043409,0043508,0043651,0048147,0051122,0051771,0070026,0070062,0070372,0070373,0070664,0071222,0071638,0097057,0098869,1901687,1904813,2001237 P09211 9398518 210 PYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGDLTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYVKALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAYVGRLSARPKLKAFLASPEYVNLPINGNGKQ