3jut A 2.25 BS01 GTQ A 1 N10 K105 K110 Q119 N10 K105 K110 Q119 ? 0008083 P05230 20145243 131 KKPKLLYCSNGGHFLRILPDGTVDGTRDRSDQHIQLQLSAESVGEVYIKSTETGQYLAMDTDGLLYGSQTPNEECLFLERLEENHYNTYISKKHAEKNWFVGLKKNGSCKRGPRTHYGQKAILFLPLPVS 3jut B 2.25 BS01 GTQ B 1 N10 K110 Q119 K120 N10 K110 Q119 K120 ? 0008083 P05230 20145243 131 KKPKLLYCSNGGHFLRILPDGTVDGTRDRSDQHIQLQLSAESVGEVYIKSTETGQYLAMDTDGLLYGSQTPNEECLFLERLEENHYNTYISKKHAEKNWFVGLKKNGSCKRGPRTHYGQKAILFLPLPVS 3nl1 A 2.155 BS02 GTQ A 1 R83 W104 Q108 H119 R127 H160 H162 D174 L176 R82 W103 Q107 H118 R126 H159 H161 D173 L175 1.13.11.4 0046872,0051213 Q67FT0 22155290 370 QNEKLDHESVTQAMQPKDTPELRALYKSFEEESIIPLWTQLGDLMPIHPKSKAVPHVWKWSTLLRLARKSGELVPVGRGGERRALGLANPGLGGNAYISPTMWAGIQYLGPRETAPEHRHSQNAFRFVVEGEGVWTVVNGDPVRMSRGDLLLTPGWCFHGHMNDTDQPMAWIDGLDIPFSQQMDVGFFEFGSDRVTDYATPNFSRGERLWCHPGLRPLSGLQNTVASPIGAYRWEFTDRALTEQLLLEDEGQPATVAPGHAAIRYVNPTTGGDVMPTLRCEFHRLRAGTETATRNEVGSTVFQVFEGAGAVVMNGETTKLEKGDMFVVPSWVPWSLQAETQFDLFRFSDAPIMEALSFMRTKIEGQ 3nw4 A 2.0 BS02 GTQ A 1 R83 W104 Q108 H119 R127 H160 H162 D174 L176 R79 W100 Q104 H115 R123 H156 H158 D170 L172 1.13.11.4 0046872,0051213 Q67FT0 23384287 370 KLDHESVTQAMQPKDTPELRALYKSFEEESIIPLWTQLGDLMPIHPKSKAVPHVWKWSTLLRLARKSGELVPVGRGGERRALGLANPGLGGNAYISPTMWAAIQYLGPRETAPEHRHSQNAFRFVVEGEGVWTVVNGDPVRMSRGDLLLTPGWCFHGHMNDTDQPMAWIDGLDIPFSQQMDVGFFEFGSDRVTDYATPNFSRGERLWCHPGLRPLSGLQNTVASPIGAYRWEFTDRALTEQLLLEDEGQPATVAPGHAAIRYVNPTTGGDVMPTLRCEFHRLRAGTETATRNEVGSTVFQVFEGAGAVVMNGETTKLEKGDMFVVPSWVPWSLQAETQFDLFRFSDAPIMEALSFMRTKIEGQ 4e3d A 1.6 BS02 GTQ A 1 H94 L198 T200 H91 L194 T196 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=5mM -logKd/Ki=2.30, IC50=5mM IC50=5000000nM, Ki=4100nM P00918 22531842 303 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4e3d A 1.6 BS03 GTQ A 2 G6 Y7 G8 F231 E239 G3 Y4 G5 F227 E235 H64 H94 H96 E106 H119 T199 H61 H91 H93 E103 H116 T195 4.2.1.1,4.2.1.69 0002009,0004064,0004089,0005515,0005737,0005829,0005886,0006730,0008270,0015670,0016829,0018820,0032230,0032849,0038166,0043209,0044070,0045177,0046872,0046903,0051453,0070050,0070062,2001150,2001225 ic50=5mM -logKd/Ki=2.30, IC50=5mM IC50=5000000nM, Ki=4100nM P00918 22531842 304 HWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK 4fag A 2.5 BS02 GTQ A 1 R83 Y104 H119 H121 R127 H160 D174 L176 R78 Y99 H114 H116 R122 H155 D169 L171 1.13.11.4 0046872,0051213 Q67FT0 22960182 402 LDHESVTQAMQPKDTPELRALYKSFEEESIIPLWTQLGDLMPIHPKSKAVPHVWKWSTLLRLARKSGELVPVGRGGERRALGLANPGLGGNAYISPTMYAGIQYLGPRETAPEHRHSQNAFRFVVEGEGVWTVVNGDPVRMSRGDLLLTPGWCFHGHMNDTDQPMAWIDGLDIPFSQQMDVGFFEFGSDRVTDYATPNFSRGERLWCHPGLRPLSGLQNTVASPIGAYRWEFTDRALTEQLLLEDEGQPATVAPGHAAIRYVNPTTGGDVMPTLRCEFHRLRAGTETATRNEVGSTVFQVFEGAGAVVMNGETTKLEKGDMFVVPSWVPWSLQAETQFDLFRFSDAPIMEALSFMRTKIEGQ 7bpc A 2.45 BS01 GTQ A 1 W24 F28 A64 F194 F295 W23 F27 A63 F193 F294 ? 0005737,0005829,0016787,0016831,0019748,0046872 N1S495 32421914 401 MLGKVALEEAFALPRHKERTRWWAGLFAIDPDKHAAEINDITEQRIKYMNEHGVGYTILSYTAPGVQDVWDPKEAQALAVEVNDYIADAIKAHPDRLGAFATLSMHDPKEAAEELRRVVTKYGFKGALVNDTQRAGADGDDMIFYDGPEWDVFWSTVTDLDVPFYLHPRNPTGSIHEKLWAKRSWLIGPPLSFAQGVSLHALGMVTNGVFDRHPKLQIVLGHLGEHIPFDMWRINHWFEDIKKPLGLSCKLTIREYFARNLWITTSGHFSTSTLQFCLGEVGADRILFSIDYPFENFSDACTWYDGLAINDVDKRKIGKDNAKKLFKLPQFYQS 7bpc C 2.45 BS01 GTQ C 1 A64 R170 N171 P190 S193 A63 R169 N170 P189 S192 ? 0005737,0005829,0016787,0016831,0019748,0046872 N1S495 32421914 401 MLGKVALEEAFALPRHKERTRWWAGLFAIDPDKHAAEINDITEQRIKYMNEHGVGYTILSYTAPGVQDVWDPKEAQALAVEVNDYIADAIKAHPDRLGAFATLSMHDPKEAAEELRRVVTKYGFKGALVNDTQRAGADGDDMIFYDGPEWDVFWSTVTDLDVPFYLHPRNPTGSIHEKLWAKRSWLIGPPLSFAQGVSLHALGMVTNGVFDRHPKLQIVLGHLGEHIPFDMWRINHWFEDIKKPLGLSCKLTIREYFARNLWITTSGHFSTSTLQFCLGEVGADRILFSIDYPFENFSDACTWYDGLAINDVDKRKIGKDNAKKLFKLPQFYQSEDH 7bpc C 2.45 BS02 GTQ C 2 L27 F28 K183 I188 L26 F27 K182 I187 ? 0005737,0005829,0016787,0016831,0019748,0046872 N1S495 32421914 402 MLGKVALEEAFALPRHKERTRWWAGLFAIDPDKHAAEINDITEQRIKYMNEHGVGYTILSYTAPGVQDVWDPKEAQALAVEVNDYIADAIKAHPDRLGAFATLSMHDPKEAAEELRRVVTKYGFKGALVNDTQRAGADGDDMIFYDGPEWDVFWSTVTDLDVPFYLHPRNPTGSIHEKLWAKRSWLIGPPLSFAQGVSLHALGMVTNGVFDRHPKLQIVLGHLGEHIPFDMWRINHWFEDIKKPLGLSCKLTIREYFARNLWITTSGHFSTSTLQFCLGEVGADRILFSIDYPFENFSDACTWYDGLAINDVDKRKIGKDNAKKLFKLPQFYQSEDH 8zi8 A 2.65 BS01 GTQ A 1 L144 H159 H255 H259 K263 L144 H159 H255 H259 K263 B7WRJ7 402 MTIVHRRLALAIGDPHGIGPEIALKALQQLSATERSLIKVYGPWSALEQAAQICQMESLLQDLIHEEAGSLAQPVQCGEITPQAGLSTVQSATAAIRACESGEVDAVIACPHHETAIHRAGIAFSGYPSLLANVLGMNEDEVFLMLVGAGLRIVHVTLHESVRSALERLSPQLVINAVDAAVQTCTLLGVPKPQVAVFGINPHASEGQLFGLEDSQITVPAVETLRKRGLTVDGPMGADMVLAQRKHDLYVAMLHDQGHIPIKLLAPNGASALSIGGRVVLSSVGHGSAMDIAGRGVADATALLRTIALLGAQP 8zi8 D 2.65 BS01 GTQ D 1 H159 H255 H259 K263 H159 H255 H259 K263 B7WRJ7 401 MTIVHRRLALAIGDPHGIGPEIALKALQQLSATERSLIKVYGPWSALEQAAQICQMESLLQDLIHEEAGSLAQPVQCGEITPQAGLSTVQSATAAIRACESGEVDAVIACPHHETAIHRAGIAFSGYPSLLANVLGMNEDEVFLMLVGAGLRIVHVTLHESVRSALERLSPQLVINAVDAAVQTCTLLGVPKPQVAVFGINPHASEGQLFGLEDSQITVPAVETLRKRGLTVDGPMGADMVLAQRKHDLYVAMLHDQGHIPIKLLAPNGASALSIGGRVVLSSVGHGSAMDIAGRGVADATALLRTIALLGAQP