5l9l A 1.8 BS01 GOP A 1 S37 W41 Q67 Q87 Y130 W235 R238 D261 T297 S8 W12 Q38 Q58 Y101 W206 R209 D232 T268 Kd=79.4nM -logKd/Ki=7.10, Kd=79.4nM 27609514 401 MDVVIASSGGGWQEAQDKALWAPAAKALNITYTQDTFQNWAEARAQVESGSVTWDIIQIGIADEPQAKAAGVLEKLDPDIVNKADFPPGSVTDSFVANSNYSTLIAWNKKTYGDNGPKSMADFFDVKKFPGKRALWNQPIGMIEAAALALGTPRDKVYEFLSTEEGRKAAIAKLTELAPSVSVWWESGAQAAQLIKDGEVDMIITWGGRVQGAINDGANFAYTFNDAQLGTDGYAIVKGAPHRDAAMRFLKEMSKAEYQKDLPNSFATAPANMKAYDLAKYTPEKMATMASAPENVAVQYSVDPNFWAKHAKWASEAYDNVRL 5l9l B 1.8 BS01 GOP B 1 S37 W41 F66 Q67 Q87 Y130 W235 R238 D261 T297 S8 W12 F37 Q38 Q58 Y101 W206 R209 D232 T268 Kd=79.4nM 27609514 401 MDVVIASSGGGWQEAQDKALWAPAAKALNITYTQDTFQNWAEARAQVESGSVTWDIIQIGIADEPQAKAAGVLEKLDPDIVNKADFPPGSVTDSFVANSNYSTLIAWNKKTYGDNGPKSMADFFDVKKFPGKRALWNQPIGMIEAAALALGTPRDKVYEFLSTEEGRKAAIAKLTELAPSVSVWWESGAQAAQLIKDGEVDMIITWGGRVQGAINDGANFAYTFNDAQLGTDGYAIVKGAPHRDAAMRFLKEMSKAEYQKDLPNSFATAPANMKAYDLAKYTPEKMATMASAPENVAVQYSVDPNFWAKHAKWASEAYDNVR 5l9o A 1.84 BS01 GOP A 1 F96 A113 A114 G116 R121 A133 G134 T162 L163 Q164 D201 S223 A226 F61 A78 A79 G81 R86 A98 G99 T127 L128 Q129 D166 S188 A191 ? 0015276,0016020,0034220,0042597 Kd=4uM -logKd/Ki=5.40, Kd=4uM Q7D447 27609514 301 DNPLGLIDPTTISVGTMGDAKPYAFTTADGNFTGFDIELFLNVAGRLGFKKEQVVFTGQEFSALMPSVANGRFDVAAAAIGTTAKRKETVDFSDGYLAGFLSVLTSEAGITDAAGLKGKRLGVVQGTLQEIYAEKNFAGTDLVKFPDNNSAVSALNNGTVDAHFLDFEAAKDYSARYPALKIAVNIPSFDAPAGFVIRKGNDALRNALDKGLKEAMQDGTWKKLHEKWFPGTPMPAAYLPK 5l9o B 1.84 BS01 GOP B 1 F96 A113 A114 G116 R121 A133 G134 T162 L163 Q164 D201 S223 A226 F62 A79 A80 G82 R87 A99 G100 T128 L129 Q130 D167 S189 A192 ? 0015276,0016020,0034220,0042597 Kd=4uM Q7D447 27609514 301 MDNPLGLIDPTTISVGTMGDAKPYAFTTADGNFTGFDIELFLNVAGRLGFKKEQVVFTGQEFSALMPSVANGRFDVAAAAIGTTAKRKETVDFSDGYLAGFLSVLTSEAGITDAAGLKGKRLGVVQGTLQEIYAEKNFAGTDLVKFPDNNSAVSALNNGTVDAHFLDFEAAKDYSARYPALKIAVNIPSFDAPAGFVIRKGNDALRNALDKGLKEAMQDGTWKKLHEKWFPGTPMPAAYLPKQ