2xp4 A 1.8 BS01 G14 A 1 H59 L61 K63 R68 C113 L122 F134 S154 H157 H40 L42 K44 R49 C94 L103 F115 S135 H138 H59 C113 Q131 S154 H157 H40 C94 Q112 S135 H138 5.2.1.8 0000413,0001666,0001932,0001934,0003755,0003774,0005515,0005634,0005654,0005737,0005829,0007088,0008013,0010468,0016607,0016859,0030182,0030496,0030512,0031434,0031647,0032091,0032092,0032465,0032794,0035307,0036064,0042177,0043547,0045944,0046785,0048156,0050808,0050815,0050816,0050821,0051219,0060255,0060392,0070373,0080090,0090263,0098978,0099524,1900180,1902430,1990757,2000146 ic50=180uM -logKd/Ki=3.74, IC50=180uM Q13526 20932746 1165 LPPGWEKAMSRSSGRVYYFNHITNASQWERPEPARVRCSHLLVKHSQSRRPSSWRQEKITRTKEEALELINGYIQKIKSGEEDFESLASQFSDCSSAKARGDLGAFSRGQMQKPFEDASFALRTGEMSGPVFTDSGIHIILRTE 3grj A 2.49 BS01 G14 A 1 S166 G167 L168 S163 G164 L165 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K309 A312 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=1mM -logKd/Ki=3.00, Ki=1mM P00811 19416920 365 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNLAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 3grj B 2.49 BS01 G14 B 1 S64 Q120 S61 Q117 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 Ki=1mM P00811 19416920 363 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ