3bki B 1.87 BS01 FQX B 1 Y16 Y61 P89 L90 T91 R96 E193 M196 Y220 Y12 Y57 P85 L86 T87 R92 E189 M192 Y216 ? 0015276,0016020 ic50=7.6uM P19491 18754610 264 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3bki C 1.87 BS01 FQX C 1 Y16 Y61 P89 L90 T91 R96 E193 M196 Y220 Y12 Y57 P85 L86 T87 R92 E189 M192 Y216 ? 0015276,0016020 ic50=7.6uM P19491 18754610 264 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3bki D 1.87 BS01 FQX D 1 Y16 Y61 P89 L90 T91 R96 E193 M196 Y220 Y12 Y57 P85 L86 T87 R92 E189 M192 Y216 ? 0015276,0016020 ic50=7.6uM P19491 18754610 264 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3bki P 1.87 BS01 FQX P 1 Y16 Y61 P89 L90 T91 R96 E193 M196 Y220 Y12 Y57 P85 L86 T87 R92 E189 M192 Y216 ? 0015276,0016020 ic50=7.6uM -logKd/Ki=5.12, IC50=7.6uM P19491 18754610 264 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC