3fxz A 1.64 BS01 FLL A 1 I276 G277 Q278 V284 A297 R299 M344 E345 Y346 L347 A348 G350 D393 L396 I28 G29 Q30 V36 A49 R51 M96 E97 Y98 L99 A100 G102 D145 L148 D389 K391 D393 N394 D407 P416 T427 D141 K143 D145 N146 D159 P168 T179 2.7.11.1 0004672,0005524,0006468 ic50=130nM -logKd/Ki=6.89, IC50=130nM Q13153 18973295 1 SDEEILEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIRQMNLQQQPKKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRDIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEAT