2giu A 2.2 BS01 FBR A 1 L298 E305 I373 I376 F377 L33 E40 I107 I110 F111 ? 0003677,0004879,0006355 ic50=1.5nM -logKd/Ki=8.82, IC50=1.5nM IC50=1.8nM, EC50=4nM Q92731 16632357 600 LDALSPEQLVLTLLEAEPPHVLISRPASMMMSLTKLADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDLVLDRDEGKCEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMYPLVADSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMVVPVYDLLLEMLNAHVL