2cma A 2.3 BS01 F20 A 1 Y46 R47 D48 D181 F182 C215 S216 A217 I219 G220 R221 Q262 D298 Y44 R45 D46 D179 F180 C213 S214 A215 I217 G218 R219 Q260 D296 D181 C215 R221 S222 Q262 D179 C213 R219 S220 Q260 3.1.3.48 0004725,0006470,0016311 ic50=185nM -logKd/Ki=6.73, IC50=185nM P18031 16916797 1299 MEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHED