4cp5 A 2.32 BS01 EOI A 1 K16 H59 F64 L68 R92 T98 R109 V116 N119 K12 H55 F60 L64 R88 T94 R105 V112 N115 K16 Y56 N119 G122 E133 K12 Y52 N115 G118 E129 2.7.4.6 0004550,0005524,0005737,0005840,0005856,0005886,0006183,0006187,0006228,0006241,0006414,0007186,0009117,0009142,0009617,0015629,0016301,0016310,0019954,0030036,0030141,0045335,0045920,0046872,0048550,0050765 Kd=452uM P22887 25766862 1156 KVNKERTFLAVKPDGVARGLVGEIIARYEKKGFVLVGLKQLVPTKDLAESHYAEHKERPFFGGLVSFITSGPVVAMVFEGKGVVASARLMIGVTNPLASAPGSIRGDFGVDVGRNIIGGSDSVESANREIALWFKPEELLTEVKPNPNLYE 4cp5 B 2.32 BS01 EOI B 1 K16 Y56 H59 F64 R92 T98 R109 V116 N119 K12 Y52 H55 F60 R88 T94 R105 V112 N115 K16 Y56 N119 G122 E133 K12 Y52 N115 G118 E129 2.7.4.6 0004550,0005524,0005737,0005840,0005856,0005886,0006183,0006187,0006228,0006241,0006414,0007186,0009117,0009142,0009617,0015629,0016301,0016310,0019954,0030036,0030141,0045335,0045920,0046872,0048550,0050765 Kd=452uM P22887 25766862 1156 KVNKERTFLAVKPDGVARGLVGEIIARYEKKGFVLVGLKQLVPTKDLAESHYAEHKERPFFGGLVSFITSGPVVAMVFEGKGVVASARLMIGVTNPLASAPGSIRGDFGVDVGRNIIGGSDSVESANREIALWFKPEELLTEVKPNPNLYE 4cp5 C 2.32 BS01 EOI C 1 K16 H59 F64 R92 T98 R109 K12 H55 F60 R88 T94 R105 K16 Y56 N119 G122 E133 K12 Y52 N115 G118 E129 2.7.4.6 0004550,0005524,0005737,0005840,0005856,0005886,0006183,0006187,0006228,0006241,0006414,0007186,0009117,0009142,0009617,0015629,0016301,0016310,0019954,0030036,0030141,0045335,0045920,0046872,0048550,0050765 Kd=452uM P22887 25766862 1156 KVNKERTFLAVKPDGVARGLVGEIIARYEKKGFVLVGLKQLVPTKDLAESHYAEHKERPFFGGLVSFITSGPVVAMVFEGKGVVASARLMIGVTNPLASAPGSIRGDFGVDVGRNIIGGSDSVESANREIALWFKPEELLTEVKPNPNLYE 4cp5 D 2.32 BS01 EOI D 1 K16 H59 F64 L68 R92 T98 R109 V116 K12 H55 F60 L64 R88 T94 R105 V112 K16 Y56 N119 G122 E133 K12 Y52 N115 G118 E129 2.7.4.6 0004550,0005524,0005737,0005840,0005856,0005886,0006183,0006187,0006228,0006241,0006414,0007186,0009117,0009142,0009617,0015629,0016301,0016310,0019954,0030036,0030141,0045335,0045920,0046872,0048550,0050765 Kd=452uM -logKd/Ki=3.34, Kd=452uM P22887 25766862 1156 KVNKERTFLAVKPDGVARGLVGEIIARYEKKGFVLVGLKQLVPTKDLAESHYAEHKERPFFGGLVSFITSGPVVAMVFEGKGVVASARLMIGVTNPLASAPGSIRGDFGVDVGRNIIGGSDSVESANREIALWFKPEELLTEVKPNPNLYE 4cp5 E 2.32 BS01 EOI E 1 K16 H59 F64 R92 T98 R109 V116 N119 K12 H55 F60 R88 T94 R105 V112 N115 K16 Y56 N119 G122 E133 K12 Y52 N115 G118 E129 2.7.4.6 0004550,0005524,0005737,0005840,0005856,0005886,0006183,0006187,0006228,0006241,0006414,0007186,0009117,0009142,0009617,0015629,0016301,0016310,0019954,0030036,0030141,0045335,0045920,0046872,0048550,0050765 Kd=452uM P22887 25766862 1156 KVNKERTFLAVKPDGVARGLVGEIIARYEKKGFVLVGLKQLVPTKDLAESHYAEHKERPFFGGLVSFITSGPVVAMVFEGKGVVASARLMIGVTNPLASAPGSIRGDFGVDVGRNIIGGSDSVESANREIALWFKPEELLTEVKPNPNLYE 4cp5 F 2.32 BS01 EOI F 1 K16 H59 F64 R92 T98 R109 V116 N119 K12 H55 F60 R88 T94 R105 V112 N115 K16 Y56 N119 G122 E133 K12 Y52 N115 G118 E129 2.7.4.6 0004550,0005524,0005737,0005840,0005856,0005886,0006183,0006187,0006228,0006241,0006414,0007186,0009117,0009142,0009617,0015629,0016301,0016310,0019954,0030036,0030141,0045335,0045920,0046872,0048550,0050765 Kd=452uM -logKd/Ki=3.34, Kd=452uM P22887 25766862 1156 KVNKERTFLAVKPDGVARGLVGEIIARYEKKGFVLVGLKQLVPTKDLAESHYAEHKERPFFGGLVSFITSGPVVAMVFEGKGVVASARLMIGVTNPLASAPGSIRGDFGVDVGRNIIGGSDSVESANREIALWFKPEELLTEVKPNPNLYE