1ixn A 2.3 BS01 DXP A 1 D11 H12 H45 R47 H52 E72 T102 T103 F133 H193 D10 H11 H44 R46 H51 E71 T101 T102 F132 H192 N9 H12 H45 R47 R51 E72 T103 E153 H193 N8 H11 H44 R46 R50 E71 T102 E152 H192 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856,0042802 P0A794 12206776 2001 AELLLGVNIDHIATLRNARGTAYPDPVQAAFIAEQAGADGITVHLREDRRHITDRDVRILRQTLDTRMNLEMAVTEEMLAIAVETKPHFCCLVPEKRQEVTTEGGLDVAGQRDKMRDACKRLADAGIQVSLFIDADEEQIKAAAEVGAPFIEIHTGCYADAKTDAEQAQELARIAKAATFAASLGLKVNAGHGLTYHNVKAIAAIPEMHELNIGHAIIGRAVMTGLKDAVAEMKRLMLEARG 1ixn B 2.3 BS01 DXP B 1 D11 H12 H45 R47 H52 E72 T102 T103 F133 H193 D10 H11 H44 R46 H51 E71 T101 T102 F132 H192 N9 H12 H45 R47 R51 E72 T103 E153 H193 N8 H11 H44 R46 R50 E71 T102 E152 H192 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856,0042802 P0A794 12206776 2002 AELLLGVNIDHIATLRNARGTAYPDPVQAAFIAEQAGADGITVHLREDRRHITDRDVRILRQTLDTRMNLEMAVTEEMLAIAVETKPHFCCLVPEKRQEVTTEGGLDVAGQRDKMRDACKRLADAGIQVSLFIDADEEQIKAAAEVGAPFIEIHTGCYADAKTDAEQAQELARIAKAATFAASLGLKVNAGHGLTYHNVKAIAAIPEMHELNIGHAIIGRAVMTGLKDAVAEMKRLMLEARG 1ixn C 2.3 BS01 DXP C 1 D11 H12 H45 R47 H52 E72 T102 T103 F133 H193 D10 H11 H44 R46 H51 E71 T101 T102 F132 H192 N9 H12 H45 R47 R51 E72 T103 E153 H193 N8 H11 H44 R46 R50 E71 T102 E152 H192 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856,0042802 P0A794 12206776 2003 AELLLGVNIDHIATLRNARGTAYPDPVQAAFIAEQAGADGITVHLREDRRHITDRDVRILRQTLDTRMNLEMAVTEEMLAIAVETKPHFCCLVPEKRQEVTTEGGLDVAGQRDKMRDACKRLADAGIQVSLFIDADEEQIKAAAEVGAPFIEIHTGCYADAKTDAEQAQELARIAKAATFAASLGLKVNAGHGLTYHNVKAIAAIPEMHELNIGHAIIGRAVMTGLKDAVAEMKRLMLEARG 1ixn D 2.3 BS01 DXP D 1 D11 H12 H45 H52 E72 T102 T103 F133 H193 D10 H11 H44 H51 E71 T101 T102 F132 H192 N9 H12 H45 R47 R51 E72 T103 E153 H193 N8 H11 H44 R46 R50 E71 T102 E152 H192 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856,0042802 P0A794 12206776 2004 AELLLGVNIDHIATLRNARGTAYPDPVQAAFIAEQAGADGITVHLREDRRHITDRDVRILRQTLDTRMNLEMAVTEEMLAIAVETKPHFCCLVPEKRQEVTTEGGLDVAGQRDKMRDACKRLADAGIQVSLFIDADEEQIKAAAEVGAPFIEIHTGCYADAKTDAEQAQELARIAKAATFAASLGLKVNAGHGLTYHNVKAIAAIPEMHELNIGHAIIGRAVMTGLKDAVAEMKRLMLEARG 1m5w A 1.96 BS01 DXP A 1 D11 H12 R47 E72 T102 T103 H193 D10 H11 R46 E71 T101 T102 H192 N9 H12 H45 R47 R51 E72 T103 E153 H193 N8 H11 H44 R46 R50 E71 T102 E152 H192 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856,0042802 Kd=54uM -logKd/Ki=4.27, Kd=54uM P0A794 12269807 1001 AELLLGVNIDHIATLRNARGTAYPDPVQAAFIAEQAGADGITVHLREDRRHITDRDVRILRQTLDTRMNLEMAVTEEMLAIAVETKPHFCCLVPEKRQEVTTEGGLDVAGQRDKMRDACKRLADAGIQVSLFIDADEEQIKAAAEVGAPFIEIHTGCYADAKTDAEQAQELARIAKAATFAASLGLKVNAGHGLTYHNVKAIAAIPEMHELNIGHAIIGRAVMTGLKDAVAEMKRLMLEARG 1m5w B 1.96 BS01 DXP B 1 N9 D11 H52 G215 H216 N8 D10 H51 G214 H215 N9 H12 H45 R47 R51 E72 T103 E153 H193 N8 H11 H44 R46 R50 E71 T102 E152 H192 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856,0042802 Kd=54uM P0A794 12269807 1002 AELLLGVNIDHIATLRNARGTAYPDPVQAAFIAEQAGADGITVHLREDRRHITDRDVRILRQTLDTRMNLEMAVTEEMLAIAVETKPHFCCLVPEKRQEVTTEGGLDVAGQRDKMRDACKRLADAGIQVSLFIDADEEQIKAAAEVGAPFIEIHTGCYADAKTDAEQAQELARIAKAATFAASLGLKVNAGHGLTYHNVKAIAAIPEMHELNIGHAIIGRAVMTGLKDAVAEMKRLMLEARG 1m5w C 1.96 BS01 DXP C 1 D11 H52 E72 T102 T103 H193 D10 H51 E71 T101 T102 H192 N9 H12 H45 R47 R51 E72 T103 E153 H193 N8 H11 H44 R46 R50 E71 T102 E152 H192 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856,0042802 Kd=54uM P0A794 12269807 1003 AELLLGVNIDHIATLRNARGTAYPDPVQAAFIAEQAGADGITVHLREDRRHITDRDVRILRQTLDTRMNLEMAVTEEMLAIAVETKPHFCCLVPEKRQEVTTEGGLDVAGQRDKMRDACKRLADAGIQVSLFIDADEEQIKAAAEVGAPFIEIHTGCYADAKTDAEQAQELARIAKAATFAASLGLKVNAGHGLTYHNVKAIAAIPEMHELNIGHAIIGRAVMTGLKDAVAEMKRLMLEARG 1m5w E 1.96 BS01 DXP E 1 D11 H52 K97 H193 G215 H216 D10 H51 K96 H192 G214 H215 N9 H12 H45 R47 R51 E72 T103 E153 H193 N8 H11 H44 R46 R50 E71 T102 E152 H192 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856,0042802 Kd=54uM -logKd/Ki=4.27, Kd=54uM P0A794 12269807 1005 AELLLGVNIDHIATLRNARGTAYPDPVQAAFIAEQAGADGITVHLREDRRHITDRDVRILRQTLDTRMNLEMAVTEEMLAIAVETKPHFCCLVPEKRQEVTTEGGLDVAGQRDKMRDACKRLADAGIQVSLFIDADEEQIKAAAEVGAPFIEIHTGCYADAKTDAEQAQELARIAKAATFAASLGLKVNAGHGLTYHNVKAIAAIPEMHELNIGHAIIGRAVMTGLKDAVAEMKRLMLEARG 1m5w F 1.96 BS01 DXP F 1 D11 H45 H52 G215 H216 D10 H44 H51 G214 H215 N9 H12 H45 R47 R51 E72 T103 E153 H193 N8 H11 H44 R46 R50 E71 T102 E152 H192 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856,0042802 Kd=54uM P0A794 12269807 1006 AELLLGVNIDHIATLRNARGTAYPDPVQAAFIAEQAGADGITVHLREDRRHITDRDVRILRQTLDTRMNLEMAVTEEMLAIAVETKPHFCCLVPEKRQEVTTEGGLDVAGQRDKMRDACKRLADAGIQVSLFIDADEEQIKAAAEVGAPFIEIHTGCYADAKTDAEQAQELARIAKAATFAASLGLKVNAGHGLTYHNVKAIAAIPEMHELNIGHAIIGRAVMTGLKDAVAEMKRLMLEARG 1m5w G 1.96 BS01 DXP G 1 N9 D11 H45 H52 H193 G215 H216 N8 D10 H44 H51 H192 G214 H215 N9 H12 H45 R47 R51 E72 T103 E153 H193 N8 H11 H44 R46 R50 E71 T102 E152 H192 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856,0042802 Kd=54uM P0A794 12269807 1007 AELLLGVNIDHIATLRNARGTAYPDPVQAAFIAEQAGADGITVHLREDRRHITDRDVRILRQTLDTRMNLEMAVTEEMLAIAVETKPHFCCLVPEKRQEVTTEGGLDVAGQRDKMRDACKRLADAGIQVSLFIDADEEQIKAAAEVGAPFIEIHTGCYADAKTDAEQAQELARIAKAATFAASLGLKVNAGHGLTYHNVKAIAAIPEMHELNIGHAIIGRAVMTGLKDAVAEMKRLMLEARG 1q0q A 1.9 BS01 DXP A 1 S151 E152 S186 H209 W212 M214 S222 N227 K228 E231 S151 E152 S186 H209 W212 M214 S222 N227 K228 E231 1.1.1.267 0008299,0016491,0019288,0030145,0030604,0042802,0046872,0051484,0070402,1990065 P45568 15567415 701 MKQLTILGSTGSIGCSTLDVVRHNPEHFRVVALVAGKNVTRMVEQCLEFSPRYAVMDDEASAKLLKTMLQQQGSRTEVLSGQQAACDMAALEDVDQVMAAIVGAAGLLPTLAAIRAGKTILLANKESLVTCGRLFMDAVKQSKAQLLPVDSEHNAIFQSLPQPIQHNLGYADLEQNGVVSILLTGSGGPFRETPLRDLATMTPDQACRHPNWSMGRKISVDSATMMNKGLEYIEARWLFNASASQMEVLIHPQSVIHSMVRYQDGSVLAQLGEPDMRTPIAHTMAWPNRVNSGVKPLDFCKLSALTFAAPDYDRYPCLKLAMEAFEQGQAATTALNAANEITVAAFLAQQIRFTDIAALNLSVLEKMDMREPQCVDDVLSVDANAREVARKEVMRLAS 1q0q B 1.9 BS01 DXP B 1 D150 S151 E152 S186 H209 W212 M214 S222 N227 K228 E231 D150 S151 E152 S186 H209 W212 M214 S222 N227 K228 E231 1.1.1.267 0008299,0016491,0019288,0030145,0030604,0042802,0046872,0051484,0070402,1990065 P45568 15567415 702 MKQLTILGSTGSIGCSTLDVVRHNPEHFRVVALVAGKNVTRMVEQCLEFSPRYAVMDDEASAKLLKTMLQQQGSRTEVLSGQQAACDMAALEDVDQVMAAIVGAAGLLPTLAAIRAGKTILLANKESLVTCGRLFMDAVKQSKAQLLPVDSEHNAIFQSLPQPIQHNLGYADLEQNGVVSILLTGSGGPFRETPLRDLATMTPDQACRHPNWSMGRKISVDSATMMNKGLEYIEARWLFNASASQMEVLIHPQSVIHSMVRYQDGSVLAQLGEPDMRTPIAHTMAWPNRVNSGVKPLDFCKLSALTFAAPDYDRYPCLKLAMEAFEQGQAATTALNAANEITVAAFLAQQIRFTDIAALNLSVLEKMDMREPQCVDDVLSVDANAREVARKEVMRLAS 3gk0 A 2.28 BS01 DXP G 1 T29 Y31 T27 Y29 N16 H19 H52 R54 R58 E79 T110 E160 H200 N14 H17 H50 R52 R56 E77 T108 E158 H198 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856 Q3JQ80 23382856 259 FFLTTPAAIDLGVNIDHVATLRNARGTAYPDPVRAALAAEDAGADAITLHLREDRRHIVDADVRTLRPRVKTRMNLECAVTPEMLDIACEIRPHDACLVPEKRSELTTEGGLDVVGHFDAVRAACKQLADAGVRVSLFIDPDEAQIRAAHETGAPVIELHTGRYADAHDAAEQQREFERIATGVDAGIALGLKVNAGHGLHYTNVQAIAALPGIAELNIGHAIVAHAVFVGWDNAVREMKAIMVAARVAALH 3gk0 C 2.28 BS01 DXP C 1 H223 A224 H214 A215 N16 H19 H52 R54 R58 E79 T110 E160 H200 N7 H10 H43 R45 R49 E70 T101 E151 H191 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856 Q3JQ80 23382856 258 AIDLGVNIDHVATLRNARGTAYPDPVRAALAAEDAGADAITLHLREDRRHIVDADVRTLRPRVKTRMNLECAVTPEMLDIACEIRPHDACLVPEKRSELTTEGGLDVVGHFDAVRAACKQLADAGVRVSLFIDPDEAQIRAAHETGAPVIELHTGRYADAHDAAEQQREFERIATGVDAGIALGLKVNAGHGLHYTNVQAIAALPGIAELNIGHAIVAHAVFVGWDNAVREMKAIMVAARVAAL 3gk0 D 2.28 BS01 DXP F 1 T29 Y31 T21 Y23 N16 H19 H52 R54 R58 E79 T110 E160 H200 N8 H11 H44 R46 R50 E71 T102 E152 H192 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856 Q3JQ80 23382856 258 AAIDLGVNIDHVATLRNARGTAYPDPVRAALAAEDAGADAITLHLREDRRHIVDADVRTLRPRVKTRMNLECAVTPEMLDIACEIRPHDACLVPEKRSELTTEGGLDVVGHFDAVRAACKQLADAGVRVSLFIDPDEAQIRAAHETGAPVIELHTGRYADAHDAAEQQREFERIATGVDAGIALGLKVNAGHGLHYTNVQAIAALPGIAELNIGHAIVAHAVFVGWDNAVREMKAIMVAARVAALH 3gk0 F 2.28 BS01 DXP F 1 Y204 H223 A224 Y195 H214 A215 N16 H19 H52 R54 R58 E79 T110 E160 H200 N7 H10 H43 R45 R49 E70 T101 E151 H191 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856 Q3JQ80 23382856 258 AIDLGVNIDHVATLRNARGTAYPDPVRAALAAEDAGADAITLHLREDRRHIVDADVRTLRPRVKTRMNLECAVTPEMLDIACEIRPHDACLVPEKRSELTTEGGLDVVGHFDAVRAACKQLADAGVRVSLFIDPDEAQIRAAHETGAPVIELHTGRYADAHDAAEQQREFERIATGVDAGIALGLKVNAGHGLHYTNVQAIAALPGIAELNIGHAIVAHAVFVGWDNAVREMKAIMVAARVAAL 3gk0 G 2.28 BS01 DXP G 1 H203 H223 A224 H228 H194 H214 A215 H219 N16 H19 H52 R54 R58 E79 T110 E160 H200 N7 H10 H43 R45 R49 E70 T101 E151 H191 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856 Q3JQ80 23382856 259 AIDLGVNIDHVATLRNARGTAYPDPVRAALAAEDAGADAITLHLREDRRHIVDADVRTLRPRVKTRMNLECAVTPEMLDIACEIRPHDACLVPEKRSELTTEGGLDVVGHFDAVRAACKQLADAGVRVSLFIDPDEAQIRAAHETGAPVIELHTGRYADAHDAAEQQREFERIATGVDAGIALGLKVNAGHGLHYTNVQAIAALPGIAELNIGHAIVAHAVFVGWDNAVREMKAIMVAARVAALH 3gk0 H 2.28 BS01 DXP C 1 T29 Y31 T21 Y23 N16 H19 H52 R54 R58 E79 T110 E160 H200 N8 H11 H44 R46 R50 E71 T102 E152 H192 2.6.99.2 0005737,0005829,0008615,0016740,0016769,0033856 Q3JQ80 23382856 258 AAIDLGVNIDHVATLRNARGTAYPDPVRAALAAEDAGADAITLHLREDRRHIVDADVRTLRPRVKTRMNLECAVTPEMLDIACEIRPHDACLVPEKRSELTTEGGLDVVGHFDAVRAACKQLADAGVRVSLFIDPDEAQIRAAHETGAPVIELHTGRYADAHDAAEQQREFERIATGVDAGIALGLKVNAGHGLHYTNVQAIAALPGIAELNIGHAIVAHAVFVGWDNAVREMKAIMVAARVAALH 3ll3 A 2.002 BS02 DXP A 1 H127 N295 E341 A348 H128 N296 E342 A349 2.7.1.12 0005524,0005975,0016301,0016310,0016773,0046316 Q5FM28 3264 SLKYIIGMDVGTTATKGVLYDINGKAVASVSKGYPLIQTKVGQAEEDPKLIFDAVQEIIFDLTQKIDGKIAAISWSSQMHSLIGLGSDDELLTNSITWADNCAKSIVQDAKNRGFAQQIYRKTGMPMHPMAPIYKLLWLKNKKTEVFSQAQKWIGIKEYIIFRLTGKLVTDTTMAAGTGILNLKTLTWDQELLDILKIKKEQLPKIAQPTKVIFPIKTEYVKKLGIDSDTKIILGASDGYLSTIGVNAIDSDHCALNVGTSGAIRTIVDQPKIDPSASYFCYPADKTHYLLGGPVNNGGIVFNWARQTLFDADETPQDFLDVAQTAPAGSRNLIFLPYLGGERAPIWDANARGSFVGLTRMHQKPEMARAVIEGIIFNLYDAASNLIKNTKKPVAINATGGFLKSDFVRQLCANIFNVPIVTMKEQQSGTLAAMFLARQALGLNQDLSEIGQFAQADKVYFPNPKEAATYQKLFPLYCEIRNALAASYGKFS 3ll3 B 2.002 BS02 DXP B 1 H127 N295 G339 E341 A348 H127 N295 G338 E340 A347 2.7.1.12 0005524,0005975,0016301,0016310,0016773,0046316 Q5FM28 3265 LKYIIGMDVGTTATKGVLYDINGKAVASVSKGYPLIQTKVGQAEEDPKLIFDAVQEIIFDLTQKIDGKIAAISWSSQMHSLIGLGSDDELLTNSITWADNCAKSIVQDAKNRGFAQQIYRKTGMPMHPMAPIYKLLWLKNKKTEVFSQAQKWIGIKEYIIFRLTGKLVTDTTMAAGTGILNLKTLTWDQELLDILKIKKEQLPKIAQPTKVIFPIKTEYVKKLGIDSDTKIILGASDGYLSTIGVNAIDSDHCALNVGTSGAIRTIVDQPKIDPSASYFCYPADKTHYLLGGPVNNGGIVFNWARQTLFADETPQDFLDVAQTAPAGSRNLIFLPYLGGERAPIWDANARGSFVGLTRMHQKPEMARAVIEGIIFNLYDAASNLIKNTKKPVAINATGGFLKSDFVRQLCANIFNVPIVTMKEQQSGTLAAMFLARQALGLNQDLSEIGQFAQADKVYFPNPKEAATYQKLFPLYCEIRNALAASYGKFS 5z9y A 1.48 BS01 DXP A 1 T43 K98 G159 L205 L206 A207 S208 T39 K85 G146 L192 L193 A194 S195 2.8.1.10 0005737,0009228,0009229,0016740,0016783,1990107 P9WG73 29428731 301 KLVIGDRSFASRLIMGTGGATNLAVLEQALIASGTELTTVAIGLLDLLNRLGITPLPNTAGSRSAAEAVLTAQLAREALNTNWVKLEVIADERTLWPDAVELVRAAEQLVDDGFVVLPYTTDDPVLARRLEDTGCAAVMPLGSPIGTGLGIANPHNIEMIVAGARVPVVLDAGIGTASDAALAMELGCDAVLLASAVTRAADPPAMAAAMAAAVTAGYLARCAGRIPKRFWA 5z9y B 1.48 BS01 DXP B 1 T43 K98 L205 A207 S208 T39 K85 L192 A194 S195 2.8.1.10 0005737,0009228,0009229,0016740,0016783,1990107 P9WG73 29428731 301 KLVIGDRSFASRLIMGTGGATNLAVLEQALIASGTELTTVAIGLLDLLNRLGITPLPNTAGSRSAAEAVLTAQLAREALNTNWVKLEVIADERTLWPDAVELVRAAEQLVDDGFVVLPYTTDDPVLARRLEDTGCAAVMPLGSPIGTGLGIANPHNIEMIVAGARVPVVLDAGIGTASDAALAMELGCDAVLLASAVTRAADPPAMAAAMAAAVTAGYLARCAGRIPKRFWAQA