1nyx A 2.65 BS01 DRF A 1 I281 F282 C285 Q286 R288 S289 H323 I326 L330 I341 S342 M348 H449 L469 Y473 I65 F66 C69 Q70 R72 S73 H107 I110 L114 I125 S126 M132 H233 L253 Y257 ? 0003677,0004879,0005634,0006355 -logKd/Ki=7.04, IC50=0.092uM EC50=575nM, Ki=90nM P37231 12672231 101 DQLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL