1al8 A 2.2 BS02 DHP A 1 Y24 W108 Y129 F172 H254 R257 Y24 W108 Y129 F166 H239 R242 S106 Y129 T155 D157 K230 H254 S106 Y129 T155 D157 K215 H239 1.1.3.15 0003973,0005777,0009853,0009854,0010181,0016491,0051707 Ki=4.8uM -logKd/Ki=5.32, Ki=4.8uM P05414 9144771 361 MEITNVNEYEAIAKQKLPKMVYDYYASGAEDQWTLAENRNAFSRILFRPRILIDVTNIDMTTTILGFKISMPIMIAPTAMQKMAHPEGEYATARAASAAGTIMTLSSWATSSVEEVASTGPGIRFFQLYVYKDRNVVAQLVRRAERAGFKAIALTVDTPRLIKNRFVLPPFLTLKNFEGIDLGLSSYVAGQIDRSLSWKDVAWLQTITSLPILVKGVITAEDARLAVQHGAAGIIVSNHGARQLDYVPATIMALEEVVKAAQGRIPVFLDGGVRRGTDVFKALALGAAGVFIGRPVVFSLAAEGEAGVKKVLQMMRDEFELTMALSGCRSLKEISRSHIAADWD