3r22 A 2.9 BS01 D37 A 1 L139 G140 K141 V147 L194 Y212 A213 G216 T217 R220 L263 L14 G15 K16 V22 L69 Y87 A88 G91 T92 R95 L138 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T158 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 -logKd/Ki=7.77, IC50=17nM IC50=17nM O14965 21798738 1 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK