1csi A 1.7 BS02 CMX A 1 R46 L273 H274 A277 V314 V315 G317 Y318 G319 H320 A321 K366 A367 K368 N373 D375 R44 L271 H272 A275 V312 V313 G315 Y316 G317 H318 A319 K364 A365 K366 N371 D373 S244 H274 H320 R329 D375 S242 H272 H318 R327 D373 2.3.3.1 0004108,0005739,0005759,0005975,0006099,0006101,0016740,0036440,0042802,0046912 Ki=1.6nM -logKd/Ki=8.80, Ki=1.6nM P23007 8011640 700 STNLKDVLASLIPKEQARIKTFRQQHGNTAVGQITVDMSYGGMRGMKGLIYETSVLDPDEGIRFRGFSIPECQKLLPKAGGGEEPLPEGLFWLLVTGQIPTPEQVSWVSKEWAKRAALPSHVVTMLDNFPTNLHPMSQLSAAITALNSESNFARAYAEGINRTKYWEFVYEDAMDLIAKLPCVAAKIYRNLYRAGSSIGAIDSKLDWSHNFTNMLGYTDPQFTELMRLYLTIHSDHEGGNVSAHTSHLVGSALSDPYLSFAAAMNGLAGPLHGLANQEVLLWLSQLQKDLGADASDEKLRDYIWNTLNSGRVVPGYGHAVLRKTDPRYTCQREFALKHLPSDPMFKLVAQLYKIVPNVLLEQGKAKNPWPNVDAHSGVLLQYYGMTEMNYYTVLFGVSRALGVLAQLIWSRALGFPLERPKSMSTAGLEKLSAGG 2h12 A 1.85 BS02 CMX A 1 A271 H272 A275 K307 L308 G310 F311 G312 R314 Y360 R364 L366 N369 D371 A253 H254 A257 K289 L290 G292 F293 G294 R296 Y342 R346 L348 N351 D353 S242 H272 H313 R322 D371 S224 H254 H295 R304 D353 2.3.3.16 0004108,0005737,0006099,0016740,0036440,0046912 P20901 17087502 5001 STATISVDGKSAEMPVLSGTLGPDVIDIRKLPAQLGVFTFDPGYGETAACNSKITFIDGDKGVLLHRGYPIAQLAENASYEEVIYLLLNGELPNKAQYDTFTNTLTNHTLLHEQIRNFFNGFRRDAHPMAILCGTVGALSAFYPANRDLAAMRLIAKIPTIAAWAYKYTQGEAFIYPRNDLNYAENFLSMMFARMSEPYKVNPVLARAMNRILILHADHEQNASTSTVRLAGSTGANPFACIAAGIAALWGPAHGGANEAVLKMLARIGKKENIPAFIAQVKDKNSGVKLMGFGHRVYKNFDPRAKIMQQTCHEVLTELGIKDDPLLDLAVELEKIALSDDYFVQRKLYPNVDFYSGIILKAMGIPTSMFTVLFAVARTTGWVSQWKEMIEEPGQRISRPRQLYIGAPQRDYVPLAKR 2h12 B 1.85 BS02 CMX B 1 A271 H272 A275 K307 L308 G310 F311 G312 H313 R314 Y360 R364 L366 N369 D371 A261 H262 A265 K297 L298 G300 F301 G302 H303 R304 Y350 R354 L356 N359 D361 S242 H272 H313 R322 D371 S232 H262 H303 R312 D361 2.3.3.16 0004108,0005737,0006099,0016740,0036440,0046912 P20901 17087502 5002 STATISVDGKSAEMPVLSGTLGPDVIDIRKLPAQLGVFTFDPGYGETAACNSKITFIDGDKGVLLHRGYPIAQLAENASYEEVIYLLLNGELPNKAQYDTFTNTLTNHTLLHEQIRNFFNGFRRDAHPMAILCGTVGALSAFYPDANDIAIPANRDLAAMRLIAKIPTIAAWAYKYTQGEAFIYPRNDLNYAENFLSMMFARMSEPYKVNPVLARAMNRILILHADHEQNASTSTVRLAGSTGANPFACIAAGIAALWGPAHGGANEAVLKMLARIGKKENIPAFIAQVKDKNSGVKLMGFGHRVYKNFDPRAKIMQQTCHEVLTELGIKDDPLLDLAVELEKIALSDDYFVQRKLYPNVDFYSGIILKAMGIPTSMFTVLFAVARTTGWVSQWKEMIEEPGQRISRPRQLYIGAPQRDYVPLAKR 2h12 C 1.85 BS02 CMX C 1 A271 H272 A275 K307 L308 G310 F311 G312 H313 R314 Y360 R364 L366 N369 D371 A261 H262 A265 K297 L298 G300 F301 G302 H303 R304 Y350 R354 L356 N359 D361 S242 H272 H313 R322 D371 S232 H262 H303 R312 D361 2.3.3.16 0004108,0005737,0006099,0016740,0036440,0046912 P20901 17087502 5003 STATISVDGKSAEMPVLSGTLGPDVIDIRKLPAQLGVFTFDPGYGETAACNSKITFIDGDKGVLLHRGYPIAQLAENASYEEVIYLLLNGELPNKAQYDTFTNTLTNHTLLHEQIRNFFNGFRRDAHPMAILCGTVGALSAFYPDANDIAIPANRDLAAMRLIAKIPTIAAWAYKYTQGEAFIYPRNDLNYAENFLSMMFARMSEPYKVNPVLARAMNRILILHADHEQNASTSTVRLAGSTGANPFACIAAGIAALWGPAHGGANEAVLKMLARIGKKENIPAFIAQVKDKNSGVKLMGFGHRVYKNFDPRAKIMQQTCHEVLTELGIKDDPLLDLAVELEKIALSDDYFVQRKLYPNVDFYSGIILKAMGIPTSMFTVLFAVARTTGWVSQWKEMIEEPGQRISRPRQLYIGAPQRDYVPLAKR 2h12 D 1.85 BS02 CMX D 1 A271 H272 A275 L308 M309 G310 F311 G312 R314 Y360 R364 L366 N369 D371 A252 H253 A256 L289 M290 G291 F292 G293 R295 Y341 R345 L347 N350 D352 S242 H272 H313 R322 D371 S223 H253 H294 R303 D352 2.3.3.16 0004108,0005737,0006099,0016740,0036440,0046912 P20901 17087502 5004 STATISVDGKSAEMPVLSGTLGPDVIDIRKLPAQLGVFTFDPGYGETAACNSKITFIDGDKGVLLHRGYPIAQLAENASYEEVIYLLLNGELPNKAQYDTFTNTLTNHTLLHEQIRNFFNGFRRDAHPMAILCGTVGALSAFYPNRDLAAMRLIAKIPTIAAWAYKYTQGEAFIYPRNDLNYAENFLSMMFARMSEPYKVNPVLARAMNRILILHADHEQNASTSTVRLAGSTGANPFACIAAGIAALWGPAHGGANEAVLKMLARIGKKENIPAFIAQVKDKNSGVKLMGFGHRVYKNFDPRAKIMQQTCHEVLTELGIKDDPLLDLAVELEKIALSDDYFVQRKLYPNVDFYSGIILKAMGIPTSMFTVLFAVARTTGWVSQWKEMIEEPGQRISRPRQLYIGAPQRDYVPLAKR 2h12 E 1.85 BS02 CMX E 1 A271 H272 A275 L308 G310 F311 G312 H313 R314 Y360 R364 L366 N369 D371 A261 H262 A265 L298 G300 F301 G302 H303 R304 Y350 R354 L356 N359 D361 S242 H272 H313 R322 D371 S232 H262 H303 R312 D361 2.3.3.16 0004108,0005737,0006099,0016740,0036440,0046912 P20901 17087502 5005 STATISVDGKSAEMPVLSGTLGPDVIDIRKLPAQLGVFTFDPGYGETAACNSKITFIDGDKGVLLHRGYPIAQLAENASYEEVIYLLLNGELPNKAQYDTFTNTLTNHTLLHEQIRNFFNGFRRDAHPMAILCGTVGALSAFYPDANDIAIPANRDLAAMRLIAKIPTIAAWAYKYTQGEAFIYPRNDLNYAENFLSMMFARMSEPYKVNPVLARAMNRILILHADHEQNASTSTVRLAGSTGANPFACIAAGIAALWGPAHGGANEAVLKMLARIGKKENIPAFIAQVKDKNSGVKLMGFGHRVYKNFDPRAKIMQQTCHEVLTELGIKDDPLLDLAVELEKIALSDDYFVQRKLYPNVDFYSGIILKAMGIPTSMFTVLFAVARTTGWVSQWKEMIEEPGQRISRPRQLYIGAPQRDYVPLAKR 2h12 F 1.85 BS02 CMX F 1 A271 H272 A275 K307 L308 G310 F311 G312 R314 Y360 R364 L366 N369 D371 A255 H256 A259 K291 L292 G294 F295 G296 R298 Y344 R348 L350 N353 D355 S242 H272 H313 R322 D371 S226 H256 H297 R306 D355 2.3.3.16 0004108,0005737,0006099,0016740,0036440,0046912 P20901 17087502 5006 STATISVDGKSAEMPVLSGTLGPDVIDIRKLPAQLGVFTFDPGYGETAACNSKITFIDGDKGVLLHRGYPIAQLAENASYEEVIYLLLNGELPNKAQYDTFTNTLTNHTLLHEQIRNFFNGFRRDAHPMAILCGTVGALSAFYPDPANRDLAAMRLIAKIPTIAAWAYKYTQGEAFIYPRNDLNYAENFLSMMFARMSEPYKVNPVLARAMNRILILHADHEQNASTSTVRLAGSTGANPFACIAAGIAALWGPAHGGANEAVLKMLARIGKKENIPAFIAQVKDKNSGVKLMGFGHRVYKNFDPRAKIMQQTCHEVLTELGIKDDPLLDLAVELEKIALSDDYFVQRKLYPNVDFYSGIILKAMGIPTSMFTVLFAVARTTGWVSQWKEMIEEPGQRISRPRQLYIGAPQRDYVPLAKR 6xbq A 1.64 BS02 CMX A 1 Q39 Q60 A70 K73 W74 H83 H84 L107 F122 P125 K126 L132 Q39 Q60 A70 K73 W74 H83 H84 L107 F122 P125 K126 L132 H7 E43 Q60 H84 E134 H7 E43 Q60 H84 E134 ? 0004493,0046491,0046872 Q9L2C2 204 SLTRIDHIGIACHDLDATVEFYRATYGFEVFHTEVNEEQGVREAMLKINDTSDGGASYLQLLEPTREDSAVGKWLAKNGEGVHHIAFGTADVDADAADIRDKGVRVLYDEPRRGSMGSRITFLHPKDCHGVLTELVTSAAVESP