1jiz A 2.6 BS06 CGS A 1 I81 L82 A83 T116 H119 E120 H123 H129 P139 Y141 I82 L83 A84 T117 H120 E121 H124 H130 P140 Y142 H119 E120 H123 H129 H120 E121 H124 H130 3.4.24.65 0004222,0006508,0008237,0008270,0031012 -logKd/Ki=8.70, IC50=2.0nM P39900 11575929 998 GFREMPGGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYGD 1jiz B 2.6 BS06 CGS B 1 I81 L82 T116 H119 E120 H123 H129 P139 I82 L83 T117 H120 E121 H124 H130 P140 H119 E120 H123 H129 H120 E121 H124 H130 3.4.24.65 0004222,0006508,0008237,0008270,0031012 P39900 11575929 999 GFREMPGGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHEIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYGD 2w0d A 2.0 BS06 CGS A 1 I180 L181 A182 H218 H222 H228 P238 Y240 I75 L76 A77 H113 H117 H123 P133 Y135 H218 A219 H222 H228 H113 A114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50~2nM -logKd/Ki=8.70, IC50=2.0nM P39900 19239231 1273 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHAIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 2w0d A 2.0 BS07 CGS C 1 G179 I180 G74 I75 H218 A219 H222 H228 H113 A114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50~2nM -logKd/Ki=8.70, IC50=2.0nM P39900 19239231 1273 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHAIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 2w0d B 2.0 BS06 CGS B 1 I180 L181 A182 H218 H222 H228 P238 I75 L76 A77 H113 H117 H123 P133 H218 A219 H222 H228 H113 A114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50~2nM P39900 19239231 1269 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHAIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 2w0d C 2.0 BS06 CGS C 1 I180 A182 H218 H222 H228 P238 Y240 I76 A78 H114 H118 H124 P134 Y136 H218 A219 H222 H228 H114 A115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50~2nM P39900 19239231 1273 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHAIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 2w0d D 2.0 BS06 CGS D 1 I180 L181 A182 T215 H218 H222 H228 P238 Y240 I76 L77 A78 T111 H114 H118 H124 P134 Y136 H218 A219 H222 H228 H114 A115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 ic50~2nM P39900 19239231 1273 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDFHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHAIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 3ayk A -1.00 BS04 CGS A 1 N80 L81 A82 H118 H122 P138 S139 Y140 N74 L75 A76 H112 H116 P132 S133 Y134 H118 E119 H122 H128 H112 E113 H116 H122 3.4.24.7 0004222,0006508,0008237,0008270,0031012 Ki=33nM, IC50=15nM P03956 10353819 173 PRWEQTHLTYRIENYTPDLPRADVDHAIEKAFQLWSNVTPLTFTKVSEGQADIMISFVRGDHRDNSPFDGPGGNLAHAFQPGPGIGGDAHFDEDERWTNNFREYNLHRVAAHELGHSLGLSHSTDIGALMYPSYTFSGDVQLAQDDIDGIQAIYGRS 4ayk A -1.00 BS04 CGS A 1 N80 L81 A82 R114 H118 H122 H128 P138 S139 N80 L81 A82 R114 H118 H122 H128 P138 S139 H118 E119 H122 H128 H118 E119 H122 H128 3.4.24.7 0004222,0006508,0008237,0008270,0031012 Ki=33nM, IC50=15nM P03956 10353819 173 VLTEGNPRWEQTHLTYRIENYTPDLPRADVDHAIEKAFQLWSNVTPLTFTKVSEGQADIMISFVRGDHRDNSPFDGPGGNLAHAFQPGPGIGGDAHFDEDERWTNNFREYNLHRVAAHELGHSLGLSHSTDIGALMYPSYTFSGDVQLAQDDIDGIQAIYGRSQNPVQP