3at4 A 2.2 BS01 CCK A 1 L45 V53 V66 K68 F113 H115 V116 M163 I174 D175 L44 V52 V65 K67 F112 H114 V115 M162 I173 D174 D156 K158 N161 D175 P184 S194 D155 K157 N160 D174 P183 S193 2.7.11.1 0004672,0004674,0005524,0006468 Kd=2.26nM -logKd/Ki=8.10, IC50=8.0nM P68400 21735094 336 SGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQA 3e3b X 3.2 BS01 CCK X 1 L46 V54 V67 K69 F114 I117 M164 I175 D176 L46 V54 V67 K69 F114 I117 M164 I175 D176 N162 D176 S195 N162 D176 S195 2.7.11.1 0000785,0001669,0004672,0004674,0005515,0005524,0005634,0005654,0005737,0005829,0005956,0006302,0006338,0006468,0006915,0007283,0016055,0016310,0021987,0031519,0032435,0044024,0051726,0097421,0106310,1901524,1903955,1905818,2001234 -logKd/Ki=7.96, IC50=11nM P19784 19193990 351 MPGPAAGSRARVYAEVNSLRSREYWDYEAHVPSWGNQDDYQLVRKLGRGKYSEVFEAINITNNERVVVKILKPVKKKKIKREVKILENLRGGTNIIKLIDTVKDPVSKTPALVFEYINNTDFKQLYQILTDFDIRFYMYELLKALDYCHSKGIMHRDVKPHNVMIDHQQKKLRLIDWGLAEFYHPAQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRREPFFHGQDNYDQLVRIAKVLGTEELYGYLKKYHIDLDPHFNDILGQHSRKRWENFIHSENRHLVSPEALDLLDKLLRYDHQQRLTAKEAMEHPYFYPVVKEQSQ