6fdz U 2.55 BS01 C87 U 1 S22 A26 V28 A42 K44 M91 F93 C94 G97 L144 F158 S15 A19 V21 A35 K37 M84 F86 C87 G90 L137 F151 D137 K139 Q141 N142 D157 S176 D130 K132 Q134 N135 D150 S169 2.7.11.1 0004672,0004674,0005524,0006468,0010506 Q6PHR2 301 PPRLDGFILTERLGSGTYATVYKAYAKKDTREVVAIKCVAKKSLNKASVENLLTEIEILKGIRHPHIVQLKDFQWDSDNIYLIMEFCAGGDLSRFIHTRRILPEKVARVFMQQLASALQFLHERNISHLDLKPQNILLSSLEKPHLKLADFGFAQHMSPWDEKHVLRGSPLYMAPEMVCQYDARVDLWSMGVILYEALFGQPPFASRSFSELEEKIRSNRVIELPLRPLLSRDCRDLLQRLLERDPSRRISFQDFFAHPWVDLEH 7nns B 2.14 BS01 C87 B 1 V214 K235 Y285 H286 G289 D293 K340 L343 V11 K32 Y82 H83 G86 D90 K137 L140 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 IC50=8nM, Kd=25nM Q04771 507 VARDITLLECVGKGRYGEVWRGSWQGENVAVKIFSSRDEKSWFRETELYNTVMLRHENILGFIASDMTSRHSSTQLWLITHYHEMGSLYDYLQLTTLDTVSCLRIVLSIASGLAHLHIEIFGTQGKPAIAHRDLKSKNILVKKNGQCCIADLGLAVMHSQSTNQLDVGNNPRVGTKRYMAPEVLDETIQVDCFDSYKRVDIWAFGLVLWEVARRMVSNGIVEDYKPPFYDVVPNDPSFEDMRKVVCVDQQRPNIPNRWFSDPTLTSLAKLMKECWYQNPSARLTALRIKKTLTKID 8bxh A 1.3 BS01 C87 A 1 G858 G861 V863 A880 K882 Y931 L932 G935 L983 D994 G26 G29 V31 A48 K50 Y99 L100 G103 L151 D162 2.7.10.2 0004672,0004713,0005524,0006468 O60674 38843875 1201 NLYFQSMDPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG