1rne A 2.4 BS01 C60 A 1 Q13 D32 G34 Y75 S76 T77 F117 D215 G217 A218 S219 Y220 S222 A300 Q15 D34 G36 Y79 S80 T81 F120 D215 G217 A218 S219 Y220 S222 A303 D32 S35 N37 W39 Y75 D215 A218 D34 S37 N39 W41 Y79 D215 A218 3.4.23.15 0004190,0006508 ic50=2nM -logKd/Ki=8.70, IC50=2nM IC50=0.830000nM, Ki=0.7nM P00797 1807356 350 NTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSNVWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRYSTGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAEFDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYNRLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMKGVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEALGAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVFQESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTEFDRRNNRIGFALAR