2c8x B 2.17 BS03 C5M B 1 H57 Y60A W60D L99 D189 A190 S195 V213 W215 G216 G226 F227 H43 Y47 W50 L96 D191 A192 S197 V217 W219 G220 G230 F231 H57 D102 E192 G193 D194 S195 G196 H43 D99 E194 G195 D196 S197 G198 3.4.21.5 0004252,0005509,0006508,0007596 ic50=220nM -logKd/Ki=6.66, IC50=220nM IC50=220nM P00734 16480269 1251 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKEGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFGE