1rpf A 2.2 BS01 C3P A 1 H12 K41 V43 N44 T45 H119 F120 H12 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 -logKd/Ki=3.99, Ki=103uM Ki=103000nM P61823 7756988 125 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 3djv A 1.6 BS01 C3P A 1 K41 V43 N44 T45 H119 F120 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 Ki=27.9uM -logKd/Ki=4.55, Ki=27.9uM Ki=27900nM P00669 19643512 125 KESAAAKFERQHMDSGNSPSSSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 3djv B 1.6 BS01 C3P B 1 K41 V43 N44 T45 H119 F120 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 Ki=27.9uM -logKd/Ki=4.55, Ki=27.9uM Ki=27900nM P00669 19643512 201 KESAAAKFERQHMDSGNSPSSSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 5et4 A 2.1 BS01 C3P A 1 Q11 H12 K41 V43 N44 T45 H119 F120 Q11 H12 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=103000nM P61823 30287244 500 KETAAAHFEHQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 5et4 B 2.1 BS01 C3P B 1 H12 K41 V43 N44 T45 H119 F120 H12 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=103000nM P61823 30287244 500 KETAAAHFEHQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 5et4 C 2.1 BS01 C3P C 1 Q11 H12 V43 N44 T45 H119 F120 Q11 H12 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=103000nM P61823 30287244 201 KETAAAHFEHQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 5et4 D 2.1 BS01 C3P D 1 H12 K41 V43 N44 T45 H119 F120 H12 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=103000nM P61823 30287244 400 KETAAAHFEHQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 5ogh A 1.16 BS01 C3P A 1 H12 K41 V43 N44 T45 H119 F120 H12 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=103000nM P61823 30287244 201 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 5ogh A 1.16 BS02 C3P A 2 K1 E2 R10 K1 E2 R10 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=103000nM P61823 30287244 202 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV