1uv5 A 2.8 BS01 BRW A 1 I62 A83 L132 Y134 V135 P136 R141 L188 D200 A382 I28 A49 L98 Y100 V101 P102 R107 L154 D166 A348 D181 K183 N186 D200 S219 D147 K149 N152 D166 S185 2.7.11.1,2.7.11.26 0004672,0005524,0006468 -logKd/Ki=8.30, IC50=0.005uM IC50=1500nM P49841 14700633 1383 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQGKAFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHA