1ewj A 2.5 BS01 BLM A 1 L56 A57 S58 W59 R65 S86 G87 R90 W99 G111 L113 R115 N119 L55 A56 S57 W58 R64 S85 G86 R89 W98 G110 L112 R114 N118 ? 0046677 -logKd/Ki=7.49, Kd=32nM P13081 11134052 1001 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj A 2.5 BS02 BLM B 1 F30 W35 I37 F29 W34 I36 ? 0046677 -logKd/Ki=7.49, Kd=32nM P13081 11134052 1002 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj B 2.5 BS01 BLM A 1 F30 W35 F29 W34 ? 0046677 -logKd/Ki=7.49, Kd=32nM P13081 11134052 1001 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj B 2.5 BS02 BLM B 1 L56 A57 S58 W59 S61 R65 G87 R90 W99 G111 R115 N119 L55 A56 S57 W58 S60 R64 G86 R89 W98 G110 R114 N118 ? 0046677 -logKd/Ki=7.49, Kd=32nM P13081 11134052 1002 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj C 2.5 BS01 BLM C 1 L56 S58 W59 S61 R65 S86 G87 R90 W99 G111 L113 R115 N119 E120 L55 S57 W58 S60 R64 S85 G86 R89 W98 G110 L112 R114 N118 E119 ? 0046677 P13081 11134052 1004 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj C 2.5 BS02 BLM D 1 F30 W35 I37 F29 W34 I36 ? 0046677 P13081 11134052 1003 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj D 2.5 BS01 BLM C 1 F30 W35 F29 W34 ? 0046677 P13081 11134052 1004 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj D 2.5 BS02 BLM D 1 P55 L56 S58 W59 S61 R65 R90 W99 L113 R115 N119 P54 L55 S57 W58 S60 R64 R89 W98 L112 R114 N118 ? 0046677 P13081 11134052 1003 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj E 2.5 BS01 BLM E 1 P55 L56 A57 S58 W59 S61 R65 G87 R90 W99 G111 L113 R115 N119 P54 L55 A56 S57 W58 S60 R64 G86 R89 W98 G110 L112 R114 N118 ? 0046677 P13081 11134052 2001 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj E 2.5 BS02 BLM F 1 F30 W35 F48 F29 W34 F47 ? 0046677 P13081 11134052 2002 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj F 2.5 BS01 BLM E 1 F30 W35 F48 F29 W34 F47 ? 0046677 P13081 11134052 2001 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj F 2.5 BS02 BLM F 1 P55 L56 S58 W59 S61 R65 R90 W99 L113 R115 N119 E120 P54 L55 S57 W58 S60 R64 R89 W98 L112 R114 N118 E119 ? 0046677 P13081 11134052 2002 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj G 2.5 BS01 BLM G 1 L56 A57 S58 W59 S61 R65 S86 G87 R90 W99 G111 L113 R115 N119 L55 A56 S57 W58 S60 R64 S85 G86 R89 W98 G110 L112 R114 N118 ? 0046677 P13081 11134052 2004 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj G 2.5 BS02 BLM H 1 F30 W35 F48 F29 W34 F47 ? 0046677 P13081 11134052 2003 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj H 2.5 BS01 BLM G 1 F30 W35 I37 F29 W34 I36 ? 0046677 P13081 11134052 2004 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1ewj H 2.5 BS02 BLM H 1 L56 A57 S58 W59 R65 S86 G87 R90 W99 M103 G111 L113 R115 L55 A56 S57 W58 R64 S85 G86 R89 W98 M102 G110 L112 R114 ? 0046677 P13081 11134052 2003 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNE 1jie A 1.8 BS01 BLM A 1 D60 N61 T62 W65 Y86 T89 P101 R109 G113 C115 H117 D60 N61 T62 W65 Y86 T89 P101 R109 G113 C115 H117 ? 0046677 Q53793 11706014 402 MVKFLGAVPVLTAVDVPANVSFWVDTLGFEKDFGDRDFAGVRRGDIRLHISRTEHQIVADNTSAWIEVTDPDALHEEWARAVSTDYADTSGPAMTPVGESPAGREFAVRDPAGNCVHFTAGE 1jie A 1.8 BS02 BLM B 1 D32 F33 F38 R47 S51 D32 F33 F38 R47 S51 ? 0046677 Q53793 11706014 401 MVKFLGAVPVLTAVDVPANVSFWVDTLGFEKDFGDRDFAGVRRGDIRLHISRTEHQIVADNTSAWIEVTDPDALHEEWARAVSTDYADTSGPAMTPVGESPAGREFAVRDPAGNCVHFTAGE 1jie B 1.8 BS01 BLM A 1 F233 F238 R247 S251 F33 F38 R47 S51 ? 0046677 Q53793 11706014 402 MVKFLGAVPVLTAVDVPANVSFWVDTLGFEKDFGDRDFAGVRRGDIRLHISRTEHQIVADNTSAWIEVTDPDALHEEWARAVSTDYADTSGPAMTPVGESPAGREFAVRDPAGNCVHFTAGE 1jie B 1.8 BS02 BLM B 1 D260 N261 W265 Y286 A302 R309 G313 C315 D60 N61 W65 Y86 A102 R109 G113 C115 ? 0046677 Q53793 11706014 401 MVKFLGAVPVLTAVDVPANVSFWVDTLGFEKDFGDRDFAGVRRGDIRLHISRTEHQIVADNTSAWIEVTDPDALHEEWARAVSTDYADTSGPAMTPVGESPAGREFAVRDPAGNCVHFTAGE 1jif A 1.6 BS01 BLM B 1 F33 F38 H49 S51 F33 F38 H49 S51 ? 0046677 -logKd/Ki=6.20, Kd=630nM Q53793 11706014 401 MVKFLGAVPVLTAVDVPANVSFWVDTLGFEKDFGDRDFAGVRRGDIRLHISRTEHQIVADNTSAWIEVTDPDALHEEWARAVSTDYADTSGPAMTPVGESPAGREFAVRDPAGNCVHFTAGE 1jif A 1.6 BS02 BLM B 2 D60 W65 Y86 P101 R109 G113 C115 D60 W65 Y86 P101 R109 G113 C115 ? 0046677 -logKd/Ki=6.20, Kd=630nM Q53793 11706014 402 MVKFLGAVPVLTAVDVPANVSFWVDTLGFEKDFGDRDFAGVRRGDIRLHISRTEHQIVADNTSAWIEVTDPDALHEEWARAVSTDYADTSGPAMTPVGESPAGREFAVRDPAGNCVHFTAGE 1jif B 1.6 BS01 BLM B 1 D260 W265 Y286 A302 R309 G313 C315 D60 W65 Y86 A102 R109 G113 C115 ? 0046677 -logKd/Ki=6.20, Kd=630nM Q53793 11706014 401 MVKFLGAVPVLTAVDVPANVSFWVDTLGFEKDFGDRDFAGVRRGDIRLHISRTEHQIVADNTSAWIEVTDPDALHEEWARAVSTDYADTSGPAMTPVGESPAGREFAVRDPAGNCVHFTAGE 1jif B 1.6 BS02 BLM B 2 F233 F238 S251 F33 F38 S51 ? 0046677 -logKd/Ki=6.20, Kd=630nM Q53793 11706014 402 MVKFLGAVPVLTAVDVPANVSFWVDTLGFEKDFGDRDFAGVRRGDIRLHISRTEHQIVADNTSAWIEVTDPDALHEEWARAVSTDYADTSGPAMTPVGESPAGREFAVRDPAGNCVHFTAGE 1niq B -1.00 BS01 BLM B 1 S58 W59 C63 R65 R90 W99 M103 L113 R115 S57 W58 C62 R64 R89 W98 M102 L112 R114 ? 0046677 P13081 2402 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNELLAGIS 1niq B -1.00 BS02 BLM B 2 N8 F30 D32 W35 I37 E46 N7 F29 D31 W34 I36 E45 ? 0046677 P13081 3402 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNELLAGIS 1niq C -1.00 BS01 BLM B 1 N8 F30 D32 W35 I37 E46 N7 F29 D31 W34 I36 E45 ? 0046677 P13081 2402 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNELLAGIS 1niq C -1.00 BS02 BLM B 2 S58 W59 C63 R65 R90 E98 W99 M103 L113 R115 S57 W58 C62 R64 R89 E97 W98 M102 L112 R114 ? 0046677 P13081 3402 TDQATPNLPSRDFDSTAAFYERLGFGIVFRDAGWMILQRGDLMLEFFAHPGLDPLASWFSCCLRLDDLAEFYRQCKSVGIQETSSGYPRIHAPELQEWGGTMAALVDPDGTLLRLIQNELLAGIS 1xrk A 1.5 BS01 BLM A 1 D60 N61 Q63 W65 F86 W102 R109 G113 C115 D59 N60 Q62 W64 F85 W101 R108 G112 C114 ? 0046677 P17493 15640151 402 AKLTSAVPVLTARDVAEAVEFWTDRLGFSRVFVEDDFAGVVRDDVTLFISAVQDQVVPDNTQAWVWVRGLDELYAEWSEVVSTNFRDASGPAMTEIVEQPWGREFALRDPAGNCVHFVAE 1xrk A 1.5 BS02 BLM B 1 F33 F38 S51 F32 F37 S50 ? 0046677 P17493 15640151 401 AKLTSAVPVLTARDVAEAVEFWTDRLGFSRVFVEDDFAGVVRDDVTLFISAVQDQVVPDNTQAWVWVRGLDELYAEWSEVVSTNFRDASGPAMTEIVEQPWGREFALRDPAGNCVHFVAE 1xrk B 1.5 BS01 BLM A 1 F33 E35 F38 F32 E34 F37 ? 0046677 P17493 15640151 402 AKLTSAVPVLTARDVAEAVEFWTDRLGFSRVFVEDDFAGVVRDDVTLFISAVQDQVVPDNTQAWVWVRGLDELYAEWSEVVSTNFRDASGPAMTEIVEQPWGREFALRDPAGNCVHFVAEE 1xrk B 1.5 BS02 BLM B 1 D60 N61 Q63 W65 F86 W102 R109 G113 C115 D59 N60 Q62 W64 F85 W101 R108 G112 C114 ? 0046677 P17493 15640151 401 AKLTSAVPVLTARDVAEAVEFWTDRLGFSRVFVEDDFAGVVRDDVTLFISAVQDQVVPDNTQAWVWVRGLDELYAEWSEVVSTNFRDASGPAMTEIVEQPWGREFALRDPAGNCVHFVAEE 2a4w A 1.5 BS01 BLM A 1 V107 W108 G109 Y112 V106 W107 G108 Y111 ? -logKd/Ki=8.29, Kd=5.1nM O05205 16756991 750 SARISLFAVVVEDMAKSLEFYRKLGVEIPAEADSAPHTEAVLDGGIRLAWDTVETVRSYDPEWQAPTGGHRFAIAFEFPDTASVDKKYAELVDAGYEGHLKPWNAVWGQRYAIVKDPDGNVVDLFAPL 2a4w B 1.5 BS01 BLM A 1 H238 D252 Y260 H37 D51 Y59 ? -logKd/Ki=8.29, Kd=5.1nM O05205 16756991 750 SARISLFAVVVEDMAKSLEFYRKLGVEIPAEADSAPHTEAVLDGGIRLAWDTVETVRSYDPEWQAPTGGHRFAIAFEFPDTASVDKKYAELVDAGYEGHLKPWNAVWGQRYAIVKDPDGNVVDLFAPLPL 2a4x A 1.4 BS01 BLM A 1 W108 Q110 Y112 F126 W107 Q109 Y111 F125 ? O05205 16756991 700 SARISLFAVVVEDMAKSLEFYRKLGVEIPAEADSAPHTEAVLDGGIRLAWDTVETVRSYDPEWQAPTGGHRFAIAFEFPDTASVDKKYAELVDAGYEGHLKPWNAVWGQRYAIVKDPDGNVVDLFAPLPLE 2zw7 A 2.8 BS02 BLM A 1 T45 L87 T90 T96 W132 Q157 Y159 W280 T37 L79 T82 T88 W124 Q149 Y151 W272 ? 0005737,0008999,0016740,0016747,0017198,1990189 Q53796 19889644 402 TAHLRTARLELTPLDPAADARHLHHAYGDEEVMRWWTRPACADPAETERYLTSCAAAPGARLWTIRAPDGTVPGMAGLLGGTDVPGLTWLLRRDSWGHGYATEAAAAVVGHALEDGGLDRVEAWIEAGNRRSLAVAARVGLTERARLAQHYPHRPGPHEMVVLGKARAEEPLTTLAVITELPVRDVAATLRLVEAALGARTAFAIGDPPEFAEAALTPWSAGPRFRLAAVPGPGPVEPVRLHLDAAGTADSLHRRAVDAGARVDGPPVRRPWGRSEFVITLPEGHELTVSAPV 2zw7 A 2.8 BS03 BLM B 1 I213 F219 R234 I205 F211 R226 ? 0005737,0008999,0016740,0016747,0017198,1990189 Q53796 19889644 403 TAHLRTARLELTPLDPAADARHLHHAYGDEEVMRWWTRPACADPAETERYLTSCAAAPGARLWTIRAPDGTVPGMAGLLGGTDVPGLTWLLRRDSWGHGYATEAAAAVVGHALEDGGLDRVEAWIEAGNRRSLAVAARVGLTERARLAQHYPHRPGPHEMVVLGKARAEEPLTTLAVITELPVRDVAATLRLVEAALGARTAFAIGDPPEFAEAALTPWSAGPRFRLAAVPGPGPVEPVRLHLDAAGTADSLHRRAVDAGARVDGPPVRRPWGRSEFVITLPEGHELTVSAPV 2zw7 B 2.8 BS01 BLM A 1 F219 R234 F211 R226 ? 0005737,0008999,0016740,0016747,0017198,1990189 Q53796 19889644 402 TAHLRTARLELTPLDPAADARHLHHAYGDEEVMRWWTRPACADPAETERYLTSCAAAPGARLWTIRAPDGTVPGMAGLLGGTDVPGLTWLLRRDSWGHGYATEAAAAVVGHALEDGGLDRVEAWIEAGNRRSLAVAARVGLTERARLAQHYPHRPGPHEMVVLGKARAEEPLTTLAVITELPVRDVAATLRLVEAALGARTAFAIGDPPEFAEAALTPWSAGPRFRLAAVPGPGPVEPVRLHLDAAGTADSLHRRAVDAGARVDGPPVRRPWGRSEFVITLPEGHELTVSAPV 2zw7 B 2.8 BS02 BLM B 1 W44 T45 L87 T90 W132 Q157 H158 W280 W36 T37 L79 T82 W124 Q149 H150 W272 ? 0005737,0008999,0016740,0016747,0017198,1990189 Q53796 19889644 403 TAHLRTARLELTPLDPAADARHLHHAYGDEEVMRWWTRPACADPAETERYLTSCAAAPGARLWTIRAPDGTVPGMAGLLGGTDVPGLTWLLRRDSWGHGYATEAAAAVVGHALEDGGLDRVEAWIEAGNRRSLAVAARVGLTERARLAQHYPHRPGPHEMVVLGKARAEEPLTTLAVITELPVRDVAATLRLVEAALGARTAFAIGDPPEFAEAALTPWSAGPRFRLAAVPGPGPVEPVRLHLDAAGTADSLHRRAVDAGARVDGPPVRRPWGRSEFVITLPEGHELTVSAPV