1uvr A 2.81 BS01 BI8 A 1 L88 G89 A109 L159 S160 Y161 E166 E209 L212 T222 D223 L18 G19 A39 L89 S90 Y91 E96 E139 L142 T152 D153 D205 K207 E209 N210 D223 T245 D135 K137 E139 N140 D153 T171 2.7.11.1 0004672,0004674,0005524,0006468 -logKd/Ki=6.00, IC50=1uM O15530 14962382 1372 PPQPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPARANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEYLIFQKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT 2vd5 A 2.8 BS01 BI8 A 1 I77 M148 E149 Y150 Y151 N200 L202 D213 I67 M138 E139 Y140 Y141 N190 L192 D203 D195 K197 N200 D213 T234 D185 K187 N190 D203 T224 2.7.11.1 0004672,0004674,0005524,0006468 Q09013 19309729 1417 QQLVLDPGFLGLEPLLDLLLGVHQELGASELAQDKYVADFLQWAEPIVVRLKEVRLQRDDFEILKVIGRGAFSEVAVVKMKQTGQVYAMKIMNKWDMLKRGEVSCFREERDVLVNGDRRWITQLHFAFQDENYLYLVMEYYVGGDLLTLLSKFGERIPAEMARFYLAEIVMAIDSVHRLGYVHRDIKPDNILLDRCGHIRLADFGSCLKLRADGTVRSLVAVGTPDYLSPEILQAVGGGPGTGSYGPECDWWALGVFAYEMFYGQTPFYADSTAETYGKIVHYKEHLSLPGVPEEARDFIQRLLCPPETRLGRGGAGDFRTHPFFFGLDWDGLRDSVPPFTPDDTCNFDEDGLTAMVSGGGETLSDILGVHLPFVGYSYSCMALRDSEVP 2vd5 B 2.8 BS01 BI8 B 1 I77 V85 A98 K100 T132 M148 E149 Y150 Y151 N200 L202 D213 I67 V75 A88 K90 T122 M138 E139 Y140 Y141 N190 L192 D203 D195 K197 N200 D213 T234 D185 K187 N190 D203 T224 2.7.11.1 0004672,0004674,0005524,0006468 Q09013 19309729 1417 QQLVLDPGFLGLEPLLDLLLGVHQELGASELAQDKYVADFLQWAEPIVVRLKEVRLQRDDFEILKVIGRGAFSEVAVVKMKQTGQVYAMKIMNKWDMLKRGEVSCFREERDVLVNGDRRWITQLHFAFQDENYLYLVMEYYVGGDLLTLLSKFGERIPAEMARFYLAEIVMAIDSVHRLGYVHRDIKPDNILLDRCGHIRLADFGSCLKLRADGTVRSLVAVGTPDYLSPEILQAVGGSYGPECDWWALGVFAYEMFYGQTPFYADSTAETYGKIVHYKEHLSLVPEEARDFIQRLLCPPETRLGRGGAGDFRTHPFFFGLDWDGLRDSVPPFTPDTDTCNFDDGLTAMVGGETLSDIGVHLPFVGYSYSCMALRDSEVP