3djf A 2.302 BS01 BC3 A 1 A118 A119 G120 Y202 E203 V219 G220 M221 N245 H259 A111 A112 G113 Y195 E196 V212 G213 M214 N238 H252 S35 H66 H88 Y90 E91 A118 M221 S222 N245 S247 H259 S31 H59 H81 Y83 E84 A111 M214 S215 N238 S240 H252 2.4.2.1 0003824,0004731,0005737,0006139,0009116,0016757,0047975 ic50=0.8uM -logKd/Ki=6.10, IC50=0.8uM Q9BMI9 20129792 290 VTANIENVKKVAHHIQKLTSIVPEIGIICGSGLGKLADGVKDKITIPYTKIPNFPQTSHSGNLIFGTLSGRKVVVMQGRFHMYEGYSNDTVALPIRVMKLLGVKILMVSNAAGGLNRSLKLGDFVILKDHIYLPGLGLNNILVGPNQEAFGTRFPALSNAYDRDLRKLAVQVAEENGFGNLVHQGVYVMNGGPCYETPAECTMLLNMGCDVVGMSTIPEVVIARHCGIQVFAVSLVTNISVLDVESDLKPNHEEVLATGAQRAELMQSWFEKIIEKLPKD 3djf B 2.302 BS01 BC3 B 1 A118 A119 G120 Y202 E203 V219 G220 M221 N245 A112 A113 G114 Y196 E197 V213 G214 M215 N239 S35 H66 H88 Y90 E91 A118 M221 S222 N245 S247 S32 H60 H82 Y84 E85 A112 M215 S216 N239 S241 2.4.2.1 0003824,0004731,0005737,0006139,0009116,0016757,0047975 ic50=0.8uM -logKd/Ki=6.10, IC50=0.8uM Q9BMI9 20129792 289 SVTANIENVKKVAHHIQKLTSIVPEIGIICGSGLADGVKDKITIPYTKIPNFPQTSVVGHSGNLIFGTLSGRKVVVMQGRFHMYEGYSNDTVALPIRVMKLLGVKILMVSNAAGGLNRSLKLGDFVILKDHIYLPGLGLNNILVGPNQEAFGTRFPALSNAYDRDLRKLAVQVAEENGFGNLVHQGVYVMNGGPCYETPAECTMLLNMGCDVVGMSTIPEVVIARHCGIQVFAVSLVTNISVLDVESAQRAELMQSWFEKIIEKLPKD 3djf C 2.302 BS01 BC3 C 1 A118 A119 G120 Y202 E203 M221 N245 H259 A115 A116 G117 Y199 E200 M218 N242 H256 S35 H66 H88 Y90 E91 A118 M221 S222 N245 S247 H259 S32 H63 H85 Y87 E88 A115 M218 S219 N242 S244 H256 2.4.2.1 0003824,0004731,0005737,0006139,0009116,0016757,0047975 ic50=0.8uM Q9BMI9 20129792 290 SVTANIENVKKVAHHIQKLTSIVPEIGIICGSGLGKLADGVKDKITIPYTKIPNFPQTSVVGHSGNLIFGTLSGRKVVVMQGRFHMYEGYSNDTVALPIRVMKLLGVKILMVSNAAGGLNRSLKLGDFVILKDHIYLPGLGLNNILVGPNQEAFGTRFPALSNAYDRDLRKLAVQVAEENGFGNLVHQGVYVMNGGPCYETPAECTMLLNMGCDVVGMSTIPEVVIARHCGIQVFAVSLVTNISVLDVESDLKPNHEEVLATGAQRAELMQSWFEKIIEKLPKD