3h26 A 2.5 BS01 B56 A 1 D101 N120 I122 M145 D184 F189 G216 K220 R254 D90 N109 I111 M134 D173 F178 G205 K209 R243 V28 D54 K220 R254 V27 D53 K209 R243 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 ic50=32.4uM -logKd/Ki=4.49, IC50=32.4uM Kd=5260nM, IC50=32400nM Q81VW8 19899766 901 KWDYDLRCGEYTLNLNEKTLIMGILNVTPDSFSDGGSYNEVDAAVRHAKEMRDEGAHIIDIGGSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK 3h26 B 2.5 BS01 B56 B 1 D101 N120 I122 M145 D184 F189 G216 K220 R254 D97 N116 I118 M141 D180 F185 G212 K216 R250 V28 D54 K220 R254 V36 D58 K216 R250 2.5.1.15 0004156,0005829,0009396,0016740,0042558,0044237,0046654,0046656,0046872 ic50=32.4uM Kd=5260nM, IC50=32400nM Q81VW8 19899766 902 HHSSGLVPMKWDYDLRCGEYTLNLNEKTLIMGILNVTPDGGSYNEVDAAVRHAKEMRDEGAHIIDIGGEVSVEEEIKRVVPMIQAVSKEVKLPISIDTYKAEVAKQAIEAGAHIINDIWGAKAEPKIAEVAAHYDVPIILMHNRDNMNYRNLMADMIADLYDSIKIAKDAGVRDENIILDPGIGFAKTPEQNLEAMRNLEQLNVLGYPVLLGTSRKSFIGHVLDLPVEERLEGTGATVCLGIEKGCEFVRVHDVKEMSRMAKMMDAMIGK