6iup A 2.0 BS01 AX0 A 1 C477 V481 A501 K503 V550 C552 A553 L619 D630 C26 V30 A50 K52 V97 C99 A100 L157 D168 D612 R616 N617 D630 D150 R154 N155 D168 2.7.10.1 0004672,0004713,0005524,0006468 ic50=23.1nM -logKd/Ki=7.64, IC50=23.1nM IC50=23nM P22455 31335138 801 LDLPLDPLWEFPRDRLVLGKPLGEGCFGQVVRAEAFGMDPARPDQASTVAVKMLKASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPRSSEGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLARGVHHIDYYKKTSNGRLPVKWMAPEALFDEVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAV