6iuo A 2.3 BS01 AWX A 1 C477 Q480 V481 A501 E520 V550 C552 A553 L619 C34 Q37 V38 A56 E75 V105 C107 A108 L161 D612 R616 N617 D630 D154 R158 N159 D172 2.7.10.1 0004672,0004713,0005524,0006468 -logKd/Ki=7.79, IC50=16.3nM IC50=>200nM P22455 31335138 801 GLLAGLVSLDLPLDPLWEFPRDRLVLGKPLGEGCFGQVVRAEAFGMARPDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLLPVKWMAPEALFDEVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAV