1n0t A 2.1 BS01 AT1 A 1 E13 Y61 P89 L90 T91 R96 G141 S142 T143 E193 Y220 E9 Y57 P85 L86 T87 R92 G137 S138 T139 E189 Y216 ? 0015276,0016020 ic50=12.2uM -logKd/Ki=4.91, IC50=12.2uM P19491 12519060 264 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1n0t B 2.1 BS01 AT1 B 1 E13 Y61 P89 L90 T91 R96 S142 T143 E193 Y220 E9 Y57 P85 L86 T87 R92 S138 T139 E189 Y216 ? 0015276,0016020 ic50=12.2uM P19491 12519060 265 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1n0t C 2.1 BS01 AT1 C 1 E13 Y61 P89 L90 T91 R96 S142 T143 E193 M196 Y220 E9 Y57 P85 L86 T87 R92 S138 T139 E189 M192 Y216 ? 0015276,0016020 ic50=12.2uM P19491 12519060 266 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1n0t D 2.1 BS01 AT1 D 1 E13 Y61 P89 L90 T91 R96 G141 S142 T143 E193 M196 Y220 E9 Y57 P85 L86 T87 R92 G137 S138 T139 E189 M192 Y216 ? 0015276,0016020 ic50=12.2uM P19491 12519060 266 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 1vso A 1.85 BS01 AT1 A 1 E13 Y61 P88 L89 T90 R95 G140 S141 E190 Y216 E9 Y57 P79 L80 T81 R86 G131 S132 E178 Y204 ? 0015276,0016020 Ki=18980nM -logKd/Ki=4.72, Ki=18.98uM Ki=2900nM P22756 17581823 258 TLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNG