3nj4 A 2.5 BS02 AFX A 1 H55 T57 E59 D131 T157 K186 D190 H301 G352 H353 M358 H54 T56 E58 D130 T156 K185 D189 H300 G351 H352 M357 H55 S78 S83 D131 E156 N181 K186 D190 N191 C195 H301 H353 S361 Q365 H54 S77 S82 D130 E155 N180 K185 D189 N190 C194 H300 H352 S360 Q364 3.13.2.1 0004013,0005515,0005634,0005737,0005783,0005829,0006730,0016787,0033353,0042470,0070062 ic50=0.48uM P23526 21226494 601 SDKLPYKVADIGLAAWGRKALDIAENEMPGLMRMRERYSASKPLKGARIAGCLHMTVETAVLIETLVTLGAEVQWSSCNIFSTQDHAAAAIAKAGIPVYAWKGETDEEYLWCIEQTLYFKDGPLNMILDDGGDLTNLIHTKYPQLLPGIRGISEETTTGVHNLYKMMANGILKVPAINVNDSVTKSKFDNLYGCRESLIDGIKRATDVMIAGKVAVVAGYGDVGKGCAQALRGFGARVIITEIDPINALQAAMEGYEVTTMDEACQEGNIFVTTTGCIDIILGRHFEQMKDDAIVCNIGHFDVEIDVKWLNENAVEKVNIKPQVDRYRLKNGRRIILLAEGRLVNLGCAMGHPSFVMSNSFTNQVMAQIELWTHPDKYPVGVHFLPKKLDEAVAEAHLGKLNVKLTKLTEKQAQYLGMSCDGPFKPDHYRY 3nj4 B 2.5 BS03 AFX B 1 H55 T57 E59 E156 T157 K186 D190 L347 G352 H353 M358 H53 T55 E57 E154 T155 K184 D188 L345 G350 H351 M356 H55 S78 S83 D131 E156 N181 K186 D190 N191 C195 H301 H353 S361 Q365 H53 S76 S81 D129 E154 N179 K184 D188 N189 C193 H299 H351 S359 Q363 3.13.2.1 0004013,0005515,0005634,0005737,0005783,0005829,0006730,0016787,0033353,0042470,0070062 ic50=0.48uM P23526 21226494 602 DKLPYKVADIGLAAWGRKALDIAENEMPGLMRMRERYSASKPLKGARIAGCLHMTVETAVLIETLVTLGAEVQWSSCNIFSTQDHAAAAIAKAGIPVYAWKGETDEEYLWCIEQTLYFKDGPLNMILDDGGDLTNLIHTKYPQLLPGIRGISEETTTGVHNLYKMMANGILKVPAINVNDSVTKSKFDNLYGCRESLIDGIKRATDVMIAGKVAVVAGYGDVGKGCAQALRGFGARVIITEIDPINALQAAMEGYEVTTMDEACQEGNIFVTTTGCIDIILGRHFEQMKDDAIVCNIGHFDVEIDVKWLNENAVEKVNIKPQVDRYRLKNGRRIILLAEGRLVNLGCAMGHPSFVMSNSFTNQVMAQIELWTHPDKYPVGVHFLPKKLDEAVAEAHLGKLNVKLTKLTEKQAQYLGMSCDGPFKPDHYRY 3nj4 C 2.5 BS02 AFX C 1 H55 T57 D131 E156 T157 K186 D190 G352 H353 M358 H54 T56 D130 E155 T156 K185 D189 G351 H352 M357 H55 S78 S83 D131 E156 N181 K186 D190 N191 C195 H301 H353 S361 Q365 H54 S77 S82 D130 E155 N180 K185 D189 N190 C194 H300 H352 S360 Q364 3.13.2.1 0004013,0005515,0005634,0005737,0005783,0005829,0006730,0016787,0033353,0042470,0070062 ic50=0.48uM P23526 21226494 603 SDKLPYKVADIGLAAWGRKALDIAENEMPGLMRMRERYSASKPLKGARIAGCLHMTVETAVLIETLVTLGAEVQWSSCNIFSTQDHAAAAIAKAGIPVYAWKGETDEEYLWCIEQTLYFKDGPLNMILDDGGDLTNLIHTKYPQLLPGIRGISEETTTGVHNLYKMMANGILKVPAINVNDSVTKSKFDNLYGCRESLIDGIKRATDVMIAGKVAVVAGYGDVGKGCAQALRGFGARVIITEIDPINALQAAMEGYEVTTMDEACQEGNIFVTTTGCIDIILGRHFEQMKDDAIVCNIGHFDVEIDVKWLNENAVEKVNIKPQVDRYRLKNGRRIILLAEGRLVNLGCAMGHPSFVMSNSFTNQVMAQIELWTHPDKYPVGVHFLPKKLDEAVAEAHLGKLNVKLTKLTEKQAQYLGMSCDGPFKPDHYRY 3nj4 D 2.5 BS03 AFX D 1 H55 T57 E59 E156 T157 K186 D190 G352 H353 M358 H53 T55 E57 E154 T155 K184 D188 G350 H351 M356 H55 S78 S83 D131 E156 N181 K186 D190 N191 C195 H301 H353 S361 Q365 H53 S76 S81 D129 E154 N179 K184 D188 N189 C193 H299 H351 S359 Q363 3.13.2.1 0004013,0005515,0005634,0005737,0005783,0005829,0006730,0016787,0033353,0042470,0070062 ic50=0.48uM P23526 21226494 604 DKLPYKVADIGLAAWGRKALDIAENEMPGLMRMRERYSASKPLKGARIAGCLHMTVETAVLIETLVTLGAEVQWSSCNIFSTQDHAAAAIAKAGIPVYAWKGETDEEYLWCIEQTLYFKDGPLNMILDDGGDLTNLIHTKYPQLLPGIRGISEETTTGVHNLYKMMANGILKVPAINVNDSVTKSKFDNLYGCRESLIDGIKRATDVMIAGKVAVVAGYGDVGKGCAQALRGFGARVIITEIDPINALQAAMEGYEVTTMDEACQEGNIFVTTTGCIDIILGRHFEQMKDDAIVCNIGHFDVEIDVKWLNENAVEKVNIKPQVDRYRLKNGRRIILLAEGRLVNLGCAMGHPSFVMSNSFTNQVMAQIELWTHPDKYPVGVHFLPKKLDEAVAEAHLGKLNVKLTKLTEKQAQYLGMSCDGPFKPDHYRY