1xqc A 2.05 BS01 AEJ A 1 M343 A350 D351 E353 W383 L387 F404 I424 L525 M27 A34 D35 E37 W67 L71 F88 I108 L207 ? ic50=63nM -logKd/Ki=7.20, IC50=63nM EC50=23.2nM, IC50=63nM P03372 15658851 1001 ALSLTADQMVSALLDAEPPILYSESMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMPLYDLLLEMLDAHR 1xqc B 2.05 BS01 AEJ B 1 A350 D351 E353 W383 M421 G521 L525 A34 D35 E37 W67 M105 G203 L207 ? ic50=63nM EC50=23.2nM, IC50=63nM P03372 15658851 2001 ALSLTADQMVSALLDAEPPILYSESMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLPLYDLLLEMLDAHR 1xqc C 2.05 BS01 AEJ C 1 M343 A350 D351 E353 W383 G521 L525 M27 A34 D35 E37 W67 G203 L207 ? ic50=63nM EC50=23.2nM, IC50=63nM P03372 15658851 3001 ALSLTADQMVSALLDAEPPILYSESMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMPLYDLLLEMLDAHR 1xqc D 2.05 BS01 AEJ D 1 A350 D351 E353 L354 W383 M421 L536 A34 D35 E37 L38 W67 M105 L209 ? ic50=63nM EC50=23.2nM, IC50=63nM P03372 15658851 4001 ALSLTADQMVSALLDAEPPILYSESMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLESAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKSVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLPLYDLLLEMLDAHR