6ilq A 2.408 BS02 AE0 A 1 C285 R288 S289 A292 I326 M329 I341 E343 M364 C58 R61 S62 A65 I99 M102 I114 E116 M137 ? 0003677,0004879,0005634,0006355 ic50=0.44uM -logKd/Ki=6.36, IC50=0.44uM IC50=440nM, EC50=1730nM P37231 30594432 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTSPFVIYDMNSLMMVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETSLHPLLQEIYKDL