2vgo A 1.7 BS01 AD5 A 1 G100 V107 A120 L154 L170 E171 F172 A173 G176 E177 L223 G14 V21 A34 L68 L84 E85 F86 A87 G90 E91 L137 D216 K218 E220 N221 D234 T252 D130 K132 E134 N135 D148 T166 2.7.11.1 0004672,0005524,0006468 ic50=500nM -logKd/Ki=6.30, IC50=500nM Q6DE08 18483302 1357 KFTIDDFDIGRPLGKGKFGNVYLAREKQNKFIMALKVLFKSQLEKEGVEHQLRREIEIQSHLRHPNILRMYNYFHDRKRIYLMLEFAPRGELYKELQKHGRFDEQRSATFMEELADALHYCHERKVIHRDIKPENLLMGYKGELKIADFGWSVHAPSLRRRTMCGTLDYLPPEMIEGKTHDEKVDLWCAGVLCYEFLVGMPPFDSPSHTETHRRIVNVDLKFPPFLSDGSKDLISKLLRYHPPQRLPLKGVMEHPWVKANSRRVLPPVY 2vgo B 1.7 BS01 AD5 B 1 G102 V107 L154 F172 A173 P174 G176 E177 G25 V30 L75 F93 A94 P95 G97 E98 D216 K218 E220 N221 D234 T252 D137 K139 E141 N142 D155 T173 2.7.11.1 0004672,0005524,0006468 ic50=500nM Q6DE08 18483302 1359 TALAEMPKRKFTIDDFDIGRPLGKGKFGNVYLAREKQNKFIMALKVLFKSQLEKVEHQLRREIEIQSHLRHPNILRMYNYFHDRKRIYLMLEFAPRGELYKELQKHGRFDEQRSATFMEELADALHYCHERKVIHRDIKPENLLMGYKGELKIADFGWSVHAPSLRRRTMCGTLDYLPPEMIEGKTHDEKVDLWCAGVLCYEFLVGMPPFDSPSHTETHRRIVNVDLKFPPFLSDGSKDLISKLLRYHPPQRLPLKGVMEHPWVKANSRRVLPPVYQS 5ljj A 3.0 BS01 AD5 A 1 I531 A551 E603 G605 N606 I607 D608 L654 Q672 P673 I17 A37 E89 G91 N92 I93 D94 L140 Q158 P159 D647 K649 N652 D664 T686 D133 K135 N138 D150 T167 2.7.12.1 0004672,0005524,0006468 -logKd/Ki=7.21, Kd=62nM P33981 27699881 901 FQSMSVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMEYGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDTDSQVGTVNYMPPEAIKDMISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQT 8bak A 1.65 BS01 AD5 A 1 L579 Q626 E627 F628 V629 K630 G632 K640 L680 L44 Q91 E92 F93 V94 K95 G97 K105 L145 2.7.10.2 0004672,0005524,0006468 O60674 36678572 906 VFHKIRNEDLIFNESLGQGTFTKIFKGVRREVGDYGQLHETEVLLKVLDKAHRNYSESFFEAASMMSKLSHKHLVLNYGVCFCGDENILVQEFVKFGSLDTYLKKNKNCINILWKLEVAKQLAWAMHFLEENTLIHGNVCAKNILLIREEDRKTGNPPFIKLSDPGISITVLPKDILQERIPWVPPECIENPKNLNLATDKWSFGTTLWEICSGGDKPLSALDSQRKLQFYEDRHQLPAPKAAELANLINNCMDYEPDHRPSFRAIIRDLNSLF 8ex1 A 1.5 BS01 AD5 A 1 L551 L579 E627 F628 V629 K630 G632 L680 L15 L43 E91 F92 V93 K94 G96 L144 2.7.10.2 0004672,0005524,0006468 O60674 36678572 901 FHKIRNEDLIFNESLGQGTFTKIFKGVRREVGDYGQLHETEVLLKVLDKAHRNYSESFFEAASMMSKLSHKHLVLNYGVCVCGDENILVQEFVKFGSLDTYLKKNKNCINILWKLEVAKQLAAAMHFLEENTLIHGNVCAKNILLIREEDRKTGNPPFIKLSDPGISITVLPKDILQERIPWVPPECIENPKNLNLATDKWSFGTTLWEICSGGDKPLSALDSQRKLQFYEDRHQLPAPKAAELANLINNCMDYEPDHRPSFRAIIRDLNSL