5zwj A 2.9 BS01 9LL A 1 A743 K745 L777 M790 T854 D855 F856 L858 A42 K44 L76 M89 T153 D154 F155 L157 D837 R841 N842 D855 D136 R140 N141 D154 2.7.10.1 0004672,0004713,0005524,0006468 IC50=3.0nM P00533 29802850 1101 ALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGSLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDE 6p1l A 2.8 BS03 9LL A 1 V726 A743 K745 I759 A763 M766 C775 R776 L788 M790 D855 F856 L858 V26 A43 K45 I57 A61 M64 C73 R74 L86 M88 D153 F154 L156 D837 R841 N842 D855 D135 R139 N140 D153 2.7.10.1 0004672,0004713,0005524,0006468 IC50=3.0nM P00533 31749909 1103 QALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREAPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDM 6p1l C 2.8 BS03 9LL C 1 V726 A743 K745 I759 E762 M766 C775 R776 L788 M790 D855 F856 L858 V25 A42 K44 I51 E54 M58 C67 R68 L80 M82 D147 F148 L150 D837 R841 N842 D855 D129 R133 N134 D147 2.7.10.1 0004672,0004713,0005524,0006468 IC50=3.0nM P00533 31749909 1103 ALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELRNKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEE 6p1l D 2.8 BS03 9LL D 1 A743 K745 I759 M766 C775 R776 L777 L788 M790 D855 F856 L858 A42 K44 I58 M65 C74 R75 L76 L87 M89 D154 F155 L157 D837 R841 N842 D855 D136 R140 N141 D154 2.7.10.1 0004672,0004713,0005524,0006468 IC50=3.0nM P00533 31749909 1103 ALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMDVVDADE 6z4b A 2.5 BS02 9LL A 1 A743 K745 C775 R776 L777 L788 M790 D855 F856 A44 K46 C76 R77 L78 L89 M91 D156 F157 D837 R841 N842 D855 D138 R142 N143 D156 2.7.10.1 0004672,0004713,0005524,0006468 IC50=3.0nM P00533 33335671 1102 NQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQ 6z4b B 2.5 BS02 9LL B 1 V726 A743 K745 I759 E762 M766 R776 L777 L788 D855 F856 V25 A40 K42 I56 E59 M63 R73 L74 L85 D152 F153 D837 R841 N842 D855 D134 R138 N139 D152 2.7.10.1 0004672,0004713,0005524,0006468 IC50=3.0nM P00533 33335671 1102 PNQALLRILKETEFKKIKVLGSGTVYKGLWIPEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGD 7jxm B 2.192 BS02 9LL B 1 V726 A743 K745 I759 C775 R776 L777 L788 M790 D855 F856 L858 V26 A43 K45 I59 C75 R76 L77 L88 M90 D155 F156 L158 2.7.10.1 0004672,0004713,0005524,0006468 IC50=3.0nM P00533 1102 QALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMDDVVD 7jxm D 2.192 BS03 9LL D 1 V726 A743 I744 K745 I759 C775 R776 L777 L788 M790 D855 F856 L858 V27 A44 I45 K46 I60 C76 R77 L78 L89 M91 D156 F157 L159 2.7.10.1 0004672,0004713,0005524,0006468 IC50=3.0nM P00533 1103 NQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMRKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDM