5uy8	A	2.39	BS01	8UM	A	1	K266 M312 S313 F315 D339 K358 N489	K263 M309 S310 F312 D336 K355 N486			2.1.2.3,3.5.4.10	0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761		ic50<5nM	-logKd/Ki=8.30, IC50<5nM	EC50=4.0nM, IC50=<5.0nM	P31939	29072452	601 	GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH
5uy8	A	2.39	BS05	8UM	B	1	N431 S450 R451 I452 P543 F544 D546 N547	N428 S447 R448 I449 P540 F541 D543 N544			2.1.2.3,3.5.4.10	0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761		ic50<5nM	-logKd/Ki=8.30, IC50<5nM	EC50=4.0nM, IC50=<5.0nM	P31939	29072452	601 	GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH
5uy8	B	2.39	BS01	8UM	A	1	N431 S450 R451 I452 P543 F544 D546 N547	N428 S447 R448 I449 P540 F541 D543 N544			2.1.2.3,3.5.4.10	0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761		ic50<5nM	-logKd/Ki=8.30, IC50<5nM	EC50=4.0nM, IC50=<5.0nM	P31939	29072452	601 	GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH
5uy8	B	2.39	BS03	8UM	B	1	K266 M312 S313 F315 D339 K358 N489	K263 M309 S310 F312 D336 K355 N486			2.1.2.3,3.5.4.10	0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761		ic50<5nM	-logKd/Ki=8.30, IC50<5nM	EC50=4.0nM, IC50=<5.0nM	P31939	29072452	601 	GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH
5uy8	C	2.39	BS01	8UM	C	1	K266 M312 S313 F315 D339 K358 N489	K263 M309 S310 F312 D336 K355 N486			2.1.2.3,3.5.4.10	0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761		ic50<5nM		EC50=4.0nM, IC50=<5.0nM	P31939	29072452	601 	GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH
5uy8	C	2.39	BS05	8UM	D	1	N431 S450 R451 I452 P543 F544 D546 N547	N428 S447 R448 I449 P540 F541 D543 N544			2.1.2.3,3.5.4.10	0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761		ic50<5nM		EC50=4.0nM, IC50=<5.0nM	P31939	29072452	601 	GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH
5uy8	D	2.39	BS01	8UM	C	1	N431 S450 R451 I452 P543 F544 D546 N547	N428 S447 R448 I449 P540 F541 D543 N544			2.1.2.3,3.5.4.10	0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761		ic50<5nM		EC50=4.0nM, IC50=<5.0nM	P31939	29072452	601 	GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH
5uy8	D	2.39	BS03	8UM	D	1	K266 M312 S313 F315 D339 N489	K263 M309 S310 F312 D336 N486			2.1.2.3,3.5.4.10	0003360,0003824,0003937,0004643,0005737,0005829,0005886,0006139,0006164,0006177,0006189,0016020,0016740,0016787,0021549,0021987,0031100,0042803,0044208,0045296,0046452,0046654,0070062,0097294,0098761		ic50<5nM		EC50=4.0nM, IC50=<5.0nM	P31939	29072452	601 	GQLALFSVSDKTGLVEFARNLTALGLNLVASGGTAKALRDAGLAVRDVSELTGFPEMLGGRVKTLHPAVHAGILARNIPEDNADMARLDFNLIRVVACNLYPFVKTVASPGVTVEEAVEQIDIGGVTLLRAAAKNHARVTVVCEPEDYVVVSTEMQSSESKDTSLETRRQLALKAFTHTAQYDEAISDYFRKQYSKGVSQMPLRYGMNPHQTPAQLYTLQPKLPITVLNGAPGFINLCDALNAWQLVKELKEALGIPAAASFKHVSPAGAAVGIPLSEDEAKVCMVYDLYKTLTPISAAYARARGADRMSSFGDFVALSDVCDVPTAKIISREVSDGIIAPGYEEEALTILSKKKNGNYCVLQMDQSYKPDENEVRTLFGLHLSQKRNNGVVDKSLFSNVVTKNKDLPESALRDLIVATIAVKYTQSNSVCYAKNGQVIGIGAGQQSRIHCTRLAGDKANYWWLRHHPQVLSMKFKTGVKRAEISNAIDQYVTGTIGEDEDLIKWKALFEEVPELLTEAEKKEWVEKLTEVSISSDAFFPFRDNVDRAKRSGVAYIAAPSGSAADKVVIEACDELGIILAHTNLRLFHH