5usq A 2.55 BS01 8LY A 1 I211 A230 K232 Y249 L278 V279 S280 Y282 H283 D290 L340 D351 I12 A31 K33 Y50 L79 V80 S81 Y83 H84 D91 L141 D152 D333 K335 N338 D351 T375 D134 K136 N139 D152 T176 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 -logKd/Ki=7.00, IC50=100nM EC50=1000nM, IC50=100nM P36897 28359790 500 TIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQ