2h96 A 3.0 BS02 893 A 1 V40 M108 L110 M111 D112 A113 V158 L168 V34 M102 L104 M105 D106 A107 V152 L162 D151 K153 N156 D169 T188 D145 K147 N150 D163 T182 2.7.11.24 0004672,0004707,0005524,0006468 -logKd/Ki=6.64, IC50=0.23uM IC50=230nM P45983 16854050 901 DNNFYSVEIGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAILERNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIIGLLNVFTPQKSLEEFQDVYIVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTAGTSFMMEPEVVTRYYRAPEVILGMGYKENVDLWSVGCIMGEMVCHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRTYVENRPKYAGYSFEKLFPDVLFPADSEHNKLKASQARDLLSKMLVIDASKRISVDEALQHPYINVWYDPSEAEAPPPKIPDKQLDEREHTIEEWKELIYKEVMDLE 2h96 B 3.0 BS02 893 B 1 I32 V40 A53 M108 L110 M111 D112 A113 N114 V158 L168 I26 V34 A47 M102 L104 M105 D106 A107 N108 V152 L162 N156 D169 N150 D163 2.7.11.24 0004672,0004707,0005524,0006468 IC50=230nM P45983 16854050 902 DNNFYSVEIGDSTFTVLKRYQNLKPIGSGAQGIVCAAYDAILERNVAIKKLSRPFQNQTHAKRAYRELVLMKCVNHKNIIGLLNVFTPQKSLEEFQDVYIVMELMDANLCQVIQMELDHERMSYLLYQMLCGIKHLHSAGIIHRDLKPSNIVVKSDCTLKILDFGLARTAGTSFMMEPEVVTRYYRAPEVILGMGYKENVDLWSVGCIMGEMVCHKILFPGRDYIDQWNKVIEQLGTPCPEFMKKLQPTVRTYVENRPKYAGYSFEKLFPDVLFPADSEHNKLKASQARDLLSKMLVIDASKRISVDEALQHPYINVWYDPSEAEAPPPKIPDKQLDEREHTIEEWKELIYKEVMDL