5uer A 1.87 BS01 87P A 1 W374 P375 F376 K378 P379 V380 D381 L385 N433 H437 E438 M442 W26 P27 F28 K30 P31 V32 D33 L37 N85 H89 E90 M94 ? Ki=43.0nM, EC50=51nM O60885 501 SHMEQLKCCSGILKEMFAKKHAAYAWPFYKPVDVEALGLHDYCDIIKHPMDMSTIKSKLEAREYRDAQEFGADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKM