4ftu A 2.1 BS01 7HK A 1 Q13 L15 Y20 V23 K38 Y86 C87 G90 L137 D148 Q11 L13 Y18 V21 K36 Y76 C77 G80 L127 D138 D130 K132 E134 N135 D148 T170 D120 K122 E124 N125 D138 T160 2.7.11.1 0000077,0004672,0004674,0005524,0006468 IC50=12nM, Ki=10nM O14757 301 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS