5tig A 2.7 BS01 7DH B 1 F50 R61 F50 R61 P1 R39 F50 R61 P1 R39 F50 R61 5.3.2.6 0009056,0016853,0042184,0042203 -logKd/Ki=4.22, Ki=60uM Q01468 29303557 101 PIAQIHILEGRSDEQKETLIREVSEAISRSLDAPLTSVRVIITEMAKGHFGIGGELASKVRR 5tig B 2.7 BS01 7DH B 1 P1 S37 P1 S37 P1 R39 F50 P1 R39 F50 5.3.2.6 0009056,0016853,0042184,0042203 -logKd/Ki=4.22, Ki=60uM Q01468 29303557 101 PIAQIHILEGRSDEQKETLIREVSEAISRSLDAPLTSVRVIITEMAKGHFGIGGELAS 5tig C 2.7 BS01 7DH C 1 P1 S37 P1 S37 P1 R39 F50 P1 R39 F50 5.3.2.6 0009056,0016853,0042184,0042203 Q01468 29303557 101 PIAQIHILEGRSDEQKETLIREVSEAISRSLDAPLTSVRVIITEMAKGHFGIGGELASK 5tig F 2.7 BS01 7DH F 1 P1 S37 P1 S37 P1 R39 F50 P1 R39 F50 5.3.2.6 0009056,0016853,0042184,0042203 Q01468 29303557 101 PIAQIHILEGRSDEQKETLIREVSEAISRSLDAPLTSVRVIITEMAKGHFGIGGELASKV 5tig O 2.7 BS01 7DH O 1 P1 S37 P1 S37 P1 R39 F50 P1 R39 F50 5.3.2.6 0009056,0016853,0042184,0042203 Q01468 29303557 101 PIAQIHILEGRSDEQKETLIREVSEAISRSLDAPLTSVRVIITEMAKGHFGIGGELASK 5tig P 2.7 BS01 7DH O 1 F50 I52 F50 I52 P1 R39 F50 P1 R39 F50 5.3.2.6 0009056,0016853,0042184,0042203 Q01468 29303557 101 PIAQIHILEGRSDEQKETLIREVSEAISRSLDAPLTSVRVIITEMAKGHFGIGGELAS 5tig P 2.7 BS02 7DH P 1 P1 S37 P1 S37 P1 R39 F50 P1 R39 F50 5.3.2.6 0009056,0016853,0042184,0042203 Q01468 29303557 101 PIAQIHILEGRSDEQKETLIREVSEAISRSLDAPLTSVRVIITEMAKGHFGIGGELAS 5tig Q 2.7 BS01 7DH R 1 L8 R11 F50 L8 R11 F50 P1 R39 F50 P1 R39 F50 5.3.2.6 0009056,0016853,0042184,0042203 Q01468 29303557 101 PIAQIHILEGRSDEQKETLIREVSEAISRSLDAPLTSVRVIITEMAKGHFGIGGELASK