5tbp A 2.6 BS01 7A4 A 1 A272 Q275 L276 L301 R302 W305 A10 Q13 L14 L39 R40 W43 ? 0003677,0003707,0005634,0006355,0008270 -logKd/Ki=5.18, Kd=6.67uM Kd=2380nM, IC50=2400nM P19793 28714476 501 DPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAPHQ 5tbp A 2.6 BS02 7A4 A 2 A271 A272 Q275 R316 L326 A327 A9 A10 Q13 R54 L64 A65 ? 0003677,0003707,0005634,0006355,0008270 -logKd/Ki=5.18, Kd=6.67uM Kd=2380nM, IC50=2400nM P19793 28714476 502 DPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAPHQ 5tbp A 2.6 BS03 7A4 A 3 F439 I447 F177 I185 ? 0003677,0003707,0005634,0006355,0008270 -logKd/Ki=5.18, Kd=6.67uM Kd=2380nM, IC50=2400nM P19793 28714476 503 DPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAPHQ 5tbp B 2.6 BS01 7A4 B 1 D273 R302 W305 D28 R57 W60 ? 0003677,0003707,0005634,0006355,0008270 Kd=2380nM, IC50=2400nM P19793 28714476 501 NEDMPVERILEAELAPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 5tbp B 2.6 BS02 7A4 D 1 F439 L451 F194 L206 ? 0003677,0003707,0005634,0006355,0008270 Kd=2380nM, IC50=2400nM P19793 28714476 501 NEDMPVERILEAELAPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 5tbp C 2.6 BS01 7A4 A 3 D273 R302 W305 D28 R57 W60 ? 0003677,0003707,0005634,0006355,0008270 -logKd/Ki=5.18, Kd=6.67uM Kd=2380nM, IC50=2400nM P19793 28714476 503 EDMPVERILEAELAVPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 5tbp D 2.6 BS01 7A4 B 1 L436 F439 I447 L174 F177 I185 ? 0003677,0003707,0005634,0006355,0008270 Kd=2380nM, IC50=2400nM P19793 28714476 501 DPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAPHQ 5tbp D 2.6 BS02 7A4 D 1 A272 Q275 L276 L301 R302 W305 A10 Q13 L14 L39 R40 W43 ? 0003677,0003707,0005634,0006355,0008270 Kd=2380nM, IC50=2400nM P19793 28714476 501 DPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAPHQ 5tbp D 2.6 BS03 7A4 D 2 A271 A272 Q275 F313 R316 L326 A327 F438 A9 A10 Q13 F51 R54 L64 A65 F176 ? 0003677,0003707,0005634,0006355,0008270 Kd=2380nM, IC50=2400nM P19793 28714476 502 DPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAPHQ