5k0b A 2.36 BS01 6PS A 1 M40 G66 M89 E90 I91 S119 H142 W143 M38 G64 M87 E88 I89 S117 H140 W141 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 -logKd/Ki=6.05, IC50=0.9uM P22734 27685665 301 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPS 5k0b B 2.36 BS01 6PS B 1 M40 G66 M89 E90 I91 S119 H142 W143 M39 G65 M88 E89 I90 S118 H141 W142 D141 K144 D169 N170 E199 D140 K143 D168 N169 E198 2.1.1.6 0000287,0006584,0008171,0016206 P22734 27685665 301 GDTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPS 5k0b C 2.36 BS01 6PS C 1 G66 M89 E90 I91 S119 H142 W143 G64 M87 E88 I89 S117 H140 W141 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 P22734 27685665 301 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPSSP 5k0b D 2.36 BS01 6PS D 1 G66 M89 E90 I91 S119 H142 W143 G64 M87 E88 I89 S117 H140 W141 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 P22734 27685665 301 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPSSPS 5k0b E 2.36 BS01 6PS E 1 M40 G66 Y68 M89 E90 I91 S119 H142 W143 M38 G64 Y66 M87 E88 I89 S117 H140 W141 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 P22734 27685665 301 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPSSP 5k0b F 2.36 BS01 6PS F 1 M40 G66 M89 E90 I91 S119 H142 W143 M38 G64 M87 E88 I89 S117 H140 W141 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 P22734 27685665 301 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPS 5k0b G 2.36 BS01 6PS G 1 M40 G66 M89 E90 I91 S119 H142 W143 M38 G64 M87 E88 I89 S117 H140 W141 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 P22734 27685665 301 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPS 5k0b H 2.36 BS01 6PS H 1 G66 M89 E90 I91 S119 H142 W143 G64 M87 E88 I89 S117 H140 W141 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 P22734 27685665 301 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEINPDCAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEECGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPSSP