5i43 A 1.95 BS06 67M A 1 G178 G179 I180 A182 H183 L214 H218 Q219 H222 H228 P238 Y240 G72 G73 I74 A76 H77 L108 H112 Q113 H116 H122 P132 Y134 H218 Q219 H222 H228 H112 Q113 H116 H122 3.4.24.65 0004222,0006508,0008237,0008270,0031012 -logKd/Ki=7.20, IC50=63nM P39900 27356908 306 PVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHQIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 5i43 B 1.95 BS01 67M B 1 I180 A182 H183 L214 H218 Q219 H222 H228 V235 F237 P238 T239 Y240 I76 A78 H79 L110 H114 Q115 H118 H124 V131 F133 P134 T135 Y136 H218 Q219 H222 H228 H114 Q115 H118 H124 3.4.24.65 0004222,0006508,0008237,0008270,0031012 P39900 27356908 301 MGPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHQIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 5i43 C 1.95 BS01 67M C 1 G179 I180 A182 H183 L214 T215 H218 Q219 H222 H228 P238 Y240 G74 I75 A77 H78 L109 T110 H113 Q114 H117 H123 P133 Y135 H218 Q219 H222 H228 H113 Q114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 P39900 27356908 301 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHQIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 5i43 D 1.95 BS01 67M D 1 G178 G179 I180 A182 L214 H218 Q219 H222 H228 P238 Y240 G73 G74 I75 A77 L109 H113 Q114 H117 H123 P133 Y135 H218 Q219 H222 H228 H113 Q114 H117 H123 3.4.24.65 0004222,0006508,0008237,0008270,0031012 P39900 27356908 301 GPVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHQIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG