5i3m A 2.17 BS01 67F A 1 I180 A182 H183 L214 T215 H218 Q219 H222 H228 F237 P238 T239 Y240 I74 A76 H77 L108 T109 H112 Q113 H116 H122 F131 P132 T133 Y134 H218 Q219 H222 H228 H112 Q113 H116 H122 3.4.24.65 0004222,0006508,0008237,0008270,0031012 -logKd/Ki=7.40, IC50=40nM P39900 27356908 301 PVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHQIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 5i3m B 2.17 BS01 67F B 1 I180 A182 L214 T215 H218 Q219 H222 H228 P238 Y240 I74 A76 L108 T109 H112 Q113 H116 H122 P132 Y134 H218 Q219 H222 H228 H112 Q113 H116 H122 3.4.24.65 0004222,0006508,0008237,0008270,0031012 P39900 27356908 301 PVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHQIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 5i3m C 2.17 BS01 67F C 1 G179 I180 A182 H183 L214 H218 Q219 H228 P238 Y240 G73 I74 A76 H77 L108 H112 Q113 H122 P132 Y134 H218 Q219 H222 H228 H112 Q113 H116 H122 3.4.24.65 0004222,0006508,0008237,0008270,0031012 P39900 27356908 301 PVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHQIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG 5i3m D 2.17 BS01 67F D 1 I180 A182 H183 L214 H218 Q219 H222 H228 V235 F237 P238 T239 Y240 I74 A76 H77 L108 H112 Q113 H116 H122 V129 F131 P132 T133 Y134 H218 Q219 H222 H228 H112 Q113 H116 H122 3.4.24.65 0004222,0006508,0008237,0008270,0031012 P39900 27356908 301 PVWRKHYITYRINNYTPDMNREDVDYAIRKAFQVWSNVTPLKFSKINTGMADILVVFARGAHGDDHAFDGKGGILAHAFGPGSGIGGDAHFDEDEFWTTHSGGTNLFLTAVHQIGHSLGLGHSSDPKAVMFPTYKYVDINTFRLSADDIRGIQSLYG