4rak A 2.04 BS01 652 A 1 F271 T272 L274 A275 S278 M312 T316 R319 F329 L330 L345 I353 F54 T55 L57 A58 S61 M95 T99 R102 F112 L113 L128 I136 ? 0003677,0004879,0006629 Ki=14nM -logKd/Ki=7.85, Ki=14nM EC50=250nM, Ki=14nM P55055 25435151 503 VQLTAAQELMIQQLVAAQLQCNKRSFSDQPKVTPWPLGADPQSRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRKLPPLLSEIW 4rak B 2.04 BS01 652 B 1 F268 F271 T272 L274 A275 S278 I309 M312 L313 E315 T316 R319 F329 L330 F340 F349 H435 W457 F42 F45 T46 L48 A49 S52 I83 M86 L87 E89 T90 R93 F103 L104 F114 F123 H209 W231 ? 0003677,0004879,0006629 Ki=14nM EC50=250nM, Ki=14nM P55055 25435151 502 QLTAAQELMIQQLVAAQLQCNKRSFSDQPKVTPWPDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRLQDKKLPPLLSEIWD