5f9e A 2.0 BS01 5VS A 1 L386 G387 F391 V394 A407 K409 T442 M458 E459 Y460 L461 N509 L511 D522 F664 L13 G14 F18 V21 A34 K36 T69 M85 E86 Y87 L88 N136 L138 D149 F291 D504 K506 D508 N509 D522 T542 D131 K133 D135 N136 D149 T169 2.7.11.13 0004672,0004674,0004697,0005524,0006468 ic50=0.46nM -logKd/Ki=9.34, IC50=0.46nM IC50=16nM Q04759 27117263 1001 KLKIEDFELHKMLGKGSFGKVFLAEFKKTNQFFAIKALKKDVVLMDDDVECTMVEKRVLSLAWEHPFLTHMFCTFQTKENLFFVMEYLNGGDLMYHIQSCHKFDLSRATFYAAEIILGLQFLHSKGIVYRDLKLDNILLDKDGHIKIADFGMCKENMLGDAKTNEFCGTPDYIAPEILLGQKYNHSVDWWSFGVLLYEMLIGQSPFHGQDEEELFHSIRMDNPFYPRWLEKEAKDLLVKLFVREPEKRLGVRGDIRQHPLFREINWEELERKEIDPPFRPKVKSPFDCSNFDKEFLNEKPRLSFADRALINSMDQNMFRNFSFMNPGMERLISHHH 5f9e B 2.0 BS01 5VS B 1 L386 F391 V394 A407 K409 T442 E459 L461 L12 F17 V20 A33 K35 T68 E85 L87 D504 K506 D508 N509 D522 T542 D130 K132 D134 N135 D148 T168 2.7.11.13 0004672,0004674,0004697,0005524,0006468 ic50=0.46nM IC50=16nM Q04759 27117263 1001 LKIEDFELHKMLGKGSFGKVFLAEFKKTNQFFAIKALKKDVVLMDDDVECTMVEKRVLSLAWEHPFLTHMFCTFQTKENLFFVMEYLNGGDLMYHIQSCHKFDLSRATFYAAEIILGLQFLHSKGIVYRDLKLDNILLDKDGHIKIADFGMCKENMLGDAKTNEFCGTPDYIAPEILLGQKYNHSVDWWSFGVLLYEMLIGQSPFHGQDEEELFHSIRMDNPFYPRWLEKEAKDLLVKLFVREPEKRLGVRGDIRQHPLFREINWEELERKEIDPPFRPKVKNMFRNFSFMNPG