5f1h A 1.82 BS01 5U6 A 1 F44 F45 F47 V49 I53 A54 N100 Y106 F23 F24 F26 V28 I32 A33 N79 Y85 ? Kd=14.1nM -logKd/Ki=7.85, Kd=14.1nM Kd=47nM, IC50=75nM Q9H8M2 26914985 201 STPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMSKERLLALKRSMS 5f1h B 1.82 BS01 5U6 B 1 F44 F45 P48 V49 I53 N100 Y106 F24 F25 P28 V29 I33 N80 Y86 ? Kd=14.1nM Kd=47nM, IC50=75nM Q9H8M2 26914985 201 ESTPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMSKERLLALKRSM 5mq1 A 1.5 BS01 5U6 A 1 A154 F155 I164 N211 Y217 A23 F24 I33 N80 Y86 ? IC50=3410nM, Kd=418nM Q9NPI1 700 EQTPLQEALNQLMRQLQRKDPSAFFSFPVTDFIAPGYSMIIKHPMDFSTMKEKIKNNDYQSIEELKDNFKLMCTNAMIYNKPETIYYKAAKKLLHSGMKILSQERIQS 6tn8 A 1.63 BS01 5U6 A 1 A233 K235 E248 L281 T283 Y285 H286 L343 D354 A30 K32 E45 L78 T80 Y82 H83 L140 D151 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 IC50=5090nM Q04771 505 VARDITLLECVGKGRYGEVWRGSWQGENVAVKIFSSRDEKSWFRETELYNTVMLRHENILGFIASDMTSRHSSTQLWLITHYHEMGSLYDYLQLTTLDTVSCLRIVLSIASGLAHLHIEIFGTQGKPAIAHRDLKSKNILVKKNGQCCIADLGLAVMHSQSTNQLDVGNNPRVGTKRYMAPEVLDETIQVDCFDSYKRVDIWAFGLVLWEVARRMVSNGIVEDYKPPFYDVVPNDPSFEDMRKVVCVDQQRPNIPNRWFSDPTLTSLAKLMKECWYQNPSARLTALRIKKTLTKID 6v1f A 2.0 BS01 5U6 A 1 F155 F156 P159 I164 N211 Y217 F24 F25 P28 I33 N80 Y86 ? Kd=418nM IC50=3410nM, Kd=418nM Q9NPI1 32091206 301 EQTPLQEALNQLMRQLQRKDPSAFFSFPVTDFIAPGYSMIIKHPMDFSTMKEKIKNNDYQSIEELKDNFKLMCTNAMIYNKPETIYYKAAKKLLHSGMKILSQERIQSLKQSIDFMA 6v1l A 2.1 BS01 5U6 A 1 W81 P82 F83 L92 L94 N140 W38 P39 F40 L49 L51 N97 ? Kd=418nM IC50=>100000nM, Kd=>10000nM O60885 32091206 201 NPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPT