5eyk	A	1.93	BS02	5U5	A	1	L99 G100 K122 E141 Q145 L154 M156 L170 F172 A173 P174 G176 E177 L223	L12 G13 K35 E54 Q58 L67 M69 L83 F85 A86 P87 G89 E90 L136	D216 K218 E220 N221 D234 T252	D129 K131 E133 N134 D147 T161	2.7.11.1	0004672,0005524,0006468		ic50=3nM	-logKd/Ki=8.52, IC50=3nM		Q6DE08	27496137	401 	FTIDDFDIVRPLGKGKFGNVYLAREKQNKFIMALKVLFKSQLEKEGVEHQLRREIEIQSHLRHPNILRMYNYFHDRKRIYLMLEFAPRGELYKELQKHGRFDEQRSATFMEELADALHYCHERKVIHRDIKPENLLMGYKGELKIADFGWSVHARRTMCGTLDYLPPEMIEGKTHDEKVDLWCAGVLCYEFLVGMPPFDSPSHTETHRRIVNVDLKFPPFLSDGSKDLISKLLRYHPPQRLPLKGVMEHPWVKANSRRVLPPVY
5eyk	B	1.93	BS01	5U5	B	1	L99 G100 K101 K122 E141 Q145 L154 L168 L170 F172 A173 G176 E177 L223	L19 G20 K21 K42 E61 Q65 L74 L88 L90 F92 A93 G96 E97 L143	D216 K218 E220 N221 D234 T252	D136 K138 E140 N141 D154 T172	2.7.11.1	0004672,0005524,0006468		ic50=3nM			Q6DE08	27496137	401 	AEMPKRKFTIDDFDIVRPLGKGKFGNVYLAREKQNKFIMALKVLFKSQLEKEGVEHQLRREIEIQSHLRHPNILRMYNYFHDRKRIYLMLEFAPRGELYKELQKHGRFDEQRSATFMEELADALHYCHERKVIHRDIKPENLLMGYKGELKIADFGWSVHAPSLRRRTMCGTLDYLPPEMIEGKTHDEKVDLWCAGVLCYEFLVGMPPFDSPSHTETHRRIVNVDLKFPPFLSDGSKDLISKLLRYHPPQRLPLKGVMEHPWVKANSRRVLPPVYQ
5eym	A	2.7	BS01	5U5	A	1	L74 A95 K97 I141 M143 H145 M146 G149 Q153 L197	L34 A52 K54 I98 M100 H102 M103 G106 Q110 L151	D190 K192 S194 N195 D208 D217 T226	D144 K146 S148 N149 D162 D171 T174	2.7.12.2	0000165,0000187,0004672,0004674,0004708,0004712,0004713,0005078,0005515,0005524,0005634,0005737,0005739,0005769,0005770,0005783,0005794,0005813,0005816,0005829,0005856,0005886,0005925,0006468,0006935,0007165,0007507,0008285,0010628,0014044,0016020,0016310,0021697,0030182,0030216,0030295,0030878,0032872,0035987,0038133,0042552,0043410,0043539,0044342,0045893,0048009,0048538,0048679,0048870,0050772,0060020,0060324,0060425,0060440,0060502,0060674,0060711,0070371,0070374,0071902,0090170,0090398,0097110,0106310,1903226,2000641			-logKd/Ki=7.60, IC50=25nM	IC50=25nM	Q02750	27496137	401 	ELDEQQRKRLEAFLTQKQKVGELKDDDFEKISELGAGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMTRSYMSPERLVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGL
5eym	B	2.7	BS02	5U5	B	1	L74 V82 A95 K97 I141 M143 H145 M146 G149 Q153 L197	L34 V39 A52 K54 I98 M100 H102 M103 G106 Q110 L151	D190 K192 S194 N195 D208 D217 T226	D144 K146 S148 N149 D162 D171 T174	2.7.12.2	0000165,0000187,0004672,0004674,0004708,0004712,0004713,0005078,0005515,0005524,0005634,0005737,0005739,0005769,0005770,0005783,0005794,0005813,0005816,0005829,0005856,0005886,0005925,0006468,0006935,0007165,0007507,0008285,0010628,0014044,0016020,0016310,0021697,0030182,0030216,0030295,0030878,0032872,0035987,0038133,0042552,0043410,0043539,0044342,0045893,0048009,0048538,0048679,0048870,0050772,0060020,0060324,0060425,0060440,0060502,0060674,0060711,0070371,0070374,0071902,0090170,0090398,0097110,0106310,1903226,2000641				IC50=25nM	Q02750	27496137	401 	ELDEQQRKRLEAFLTQKQKVGELKDDDFEKISELGAGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDSMTRSYMSPERLVQSDIWSMGLSLVEMAVGRYPIPPPDAKELELMFPMAIFELLDYIVNEPPPKLPSGVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGL
5mai	A	2.15	BS01	5U5	A	1	I17 C70 L86 E87 Y88 C89 L139 I149	I17 C70 L86 E87 Y88 C89 L139 I149	D132 K134 E136 N137 D150 S171	D132 K134 E136 N137 D150 S152	2.7.10.2,2.7.11.1	0004672,0004674,0005524,0006468					Q14680	29191878	402 	PKDYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTLGSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFSLAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDNVMALYKKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR