5etm A 1.46 BS01 5RW A 1 T42 P43 P44 L45 Y53 N55 W89 R121 F123 T43 P44 P45 L46 Y54 N56 W90 R122 F124 R82 R92 D95 D97 R83 R93 D96 D98 2.7.6.3 0000287,0003848,0005524,0009396,0016301,0016310,0046654,0046656 Kd=3.9uM -logKd/Ki=5.41, Kd=3.9uM P26281 27094768 201 MTVAYIAIGSNLASPLEQVNAALKALGDIPESHILTVSSFYRTPPLGPQDQPDYLNAAVALETSLAPEELLNHTQRIELQQGRVRKAERWGPRTLDLDIMLFGNEVINTERLTVPHYDMKNRGFMLWPLFEIAPELVFPDGEMLRQILHTRAFDKLNKW 5etr A 1.32 BS02 5RW A 1 T43 A44 V46 Y48 Q51 F54 N56 G90 R92 F123 T43 A44 V46 Y48 Q51 F54 N56 G90 R92 F123 R83 R92 D95 D97 R83 R92 D95 D97 2.7.6.3 0003848,0005524,0009396,0016301,0016310,0046654,0046656,0046872 Kd=0.3uM Q2G0Q5 27094768 202 MIQAYLGLGSNIGDRESQLNDAIKILNEYDGISVSNISPIYETAPVGYTEQPNFLNLCVEIQTTLTVLQLLECCLKTEECLHRIRKERWGPRTLDVDILLYGEEMIDLPKLSVPHPRMNERAFVLIPLNDIAANVVEPRSKLKVKDLVFVDDSVKRY 5etr B 1.32 BS02 5RW B 1 T43 A44 V46 Y48 Q51 F54 N56 G90 R92 F123 T43 A44 V46 Y48 Q51 F54 N56 G90 R92 F123 R83 R92 D95 D97 R83 R92 D95 D97 2.7.6.3 0003848,0005524,0009396,0016301,0016310,0046654,0046656,0046872 Kd=0.3uM -logKd/Ki=6.52, Kd=0.30uM Q2G0Q5 27094768 202 MIQAYLGLGSNIGDRESQLNDAIKILNEYDGISVSNISPIYETAPVGYTEQPNFLNLCVEIQTTLTVLQLLECCLKTEECLHRIRKERWGPRTLDVDILLYGEEMIDLPKLSVPHPRMNERAFVLIPLNDIAANVVEPRSKLKVKDLVFVDDSVKRY 7ala A 1.846 BS02 5RW A 1 D127 L157 T240 E243 D70 L100 T173 E176 3.5.4.16 0003934,0046654 P30793 33229582 302 PRSEEDNELNLPNLAAAYSSILSSLGENPQRQGLLKTPWRAASAMQFFTKGYQETISDVLNDAIFDEDHDEMVIVKDIDMFSMCEHHLVPFVGKVHIGYLPNKQVLGLSKLARIVEIYSRRLQVQERLTKQIAVAITEALRPAGVGVVVEATHMCSKTVTSTMLGVFREDPKTREEFLTLIR 7ala A 1.846 BS03 5RW B 1 R235 R241 R168 R174 3.5.4.16 0003934,0046654 P30793 33229582 302 PRSEEDNELNLPNLAAAYSSILSSLGENPQRQGLLKTPWRAASAMQFFTKGYQETISDVLNDAIFDEDHDEMVIVKDIDMFSMCEHHLVPFVGKVHIGYLPNKQVLGLSKLARIVEIYSRRLQVQERLTKQIAVAITEALRPAGVGVVVEATHMCSKTVTSTMLGVFREDPKTREEFLTLIR 7ala B 1.846 BS02 5RW B 1 L157 V233 T240 E243 L79 V151 T158 E161 3.5.4.16 0003934,0046654 P30793 33229582 302 LPNLAAAYSSILSSLGENPQRQGLLKTPWRAASAMQFFTKGYQETISHDEMVIVKDIDMFSMCEHHLVPFVGKVHIGYLPNKQVLGLSKLARIVEIYSRRLQVQERLTKQIAVAITEALRPAGVGVVVEATHMCMVMRGNSKTVTSTMLGVFREDPKTREEFLTLIR 7ala B 1.846 BS03 5RW C 1 S228 R235 R241 S146 R153 R159 3.5.4.16 0003934,0046654 P30793 33229582 302 LPNLAAAYSSILSSLGENPQRQGLLKTPWRAASAMQFFTKGYQETISHDEMVIVKDIDMFSMCEHHLVPFVGKVHIGYLPNKQVLGLSKLARIVEIYSRRLQVQERLTKQIAVAITEALRPAGVGVVVEATHMCMVMRGNSKTVTSTMLGVFREDPKTREEFLTLIR 7ala C 1.846 BS02 5RW C 1 D127 L157 T240 E243 D70 L100 T179 E182 3.5.4.16 0003934,0046654 P30793 33229582 302 PRSEEDNELNLPNLAAAYSSILSSLGENPQRQGLLKTPWRAASAMQFFTKGYQETISDVLNDAIFDEDHDEMVIVKDIDMFSMCEHHLVPFVGKVHIGYLPNKQVLGLSKLARIVEIYSRRLQVQERLTKQIAVAITEALRPAGVGVVVEATHMCMVMKMNSKTVTSTMLGVFREDPKTREEFLTLIR 7ala C 1.846 BS03 5RW D 1 R235 R241 R174 R180 3.5.4.16 0003934,0046654 P30793 33229582 302 PRSEEDNELNLPNLAAAYSSILSSLGENPQRQGLLKTPWRAASAMQFFTKGYQETISDVLNDAIFDEDHDEMVIVKDIDMFSMCEHHLVPFVGKVHIGYLPNKQVLGLSKLARIVEIYSRRLQVQERLTKQIAVAITEALRPAGVGVVVEATHMCMVMKMNSKTVTSTMLGVFREDPKTREEFLTLIR 7ala D 1.846 BS02 5RW D 1 D127 L157 T240 E243 D65 L95 T171 E174 3.5.4.16 0003934,0046654 P30793 33229582 302 RPRLNLPNLAAAYSSILSSLGENPQRQGLLKTPWRAASAMQFFTKGYQETISDVLNDAIFDEDHDEMVIVKDIDMFSMCEHHLVPFVGKVHIGYLPNKQVLGLSKLARIVEIYSRRLQVQERLTKQIAVAITEALRPAGVGVVVEATHMCMVNSKTVTSTMLGVFREDPKTREEFLTLIR 7ala D 1.846 BS03 5RW E 1 S228 R235 R241 S159 R166 R172 3.5.4.16 0003934,0046654 P30793 33229582 302 RPRLNLPNLAAAYSSILSSLGENPQRQGLLKTPWRAASAMQFFTKGYQETISDVLNDAIFDEDHDEMVIVKDIDMFSMCEHHLVPFVGKVHIGYLPNKQVLGLSKLARIVEIYSRRLQVQERLTKQIAVAITEALRPAGVGVVVEATHMCMVNSKTVTSTMLGVFREDPKTREEFLTLIR 7ala E 1.846 BS01 5RW A 1 R235 R241 R165 R171 3.5.4.16 0003934,0046654 P30793 33229582 302 PRSEEDNELNLPNLAAAYSSILSSLGENPQRQGLLKTPWRAASAMQFFTKGYQETISDVHDEMVIVKDIDMFSMCEHHLVPFVGKVHIGYLPNKQVLGLSKLARIVEIYSRRLQVQERLTKQIAVAITEALRPAGVGVVVEATHMCMVMRGVSKTVTSTMLGVFREDPKTREEFLTLIR 7ala E 1.846 BS03 5RW E 1 D127 L157 T240 E243 D61 L91 T170 E173 3.5.4.16 0003934,0046654 P30793 33229582 302 PRSEEDNELNLPNLAAAYSSILSSLGENPQRQGLLKTPWRAASAMQFFTKGYQETISDVHDEMVIVKDIDMFSMCEHHLVPFVGKVHIGYLPNKQVLGLSKLARIVEIYSRRLQVQERLTKQIAVAITEALRPAGVGVVVEATHMCMVMRGVSKTVTSTMLGVFREDPKTREEFLTLIR