5eth A 2.803 BS01 5RT A 1 C320 H323 L324 A327 M365 V376 F378 F388 I400 F401 V480 C52 H55 L56 A59 M97 V108 F110 F120 I132 F133 V212 ? 0003677,0004879,0005634,0006355 -logKd/Ki=7.25, IC50=0.056uM IC50=56nM P51449 27080181 501 EIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIF 5eth B 2.803 BS01 5RT B 1 W317 C320 H323 L324 V361 M365 F378 F388 I400 F401 V480 W51 C54 H57 L58 V95 M99 F112 F122 I134 F135 V214 ? 0003677,0004879,0005634,0006355 IC50=56nM P51449 27080181 501 LTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQ